BRPI0810679A2 - Derivados de 4-aza indol e seu uso como fungicidas - Google Patents

Derivados de 4-aza indol e seu uso como fungicidas

Info

Publication number
BRPI0810679A2
BRPI0810679A2 BRPI0810679-7A2A BRPI0810679A BRPI0810679A2 BR PI0810679 A2 BRPI0810679 A2 BR PI0810679A2 BR PI0810679 A BRPI0810679 A BR PI0810679A BR PI0810679 A2 BRPI0810679 A2 BR PI0810679A2
Authority
BR
Brazil
Prior art keywords
fungicides
indol derivatives
aza
aza indol
derivatives
Prior art date
Application number
BRPI0810679-7A2A
Other languages
English (en)
Inventor
Patrice Selles
Fredrik Cederbaum
Florence Marie-Emilie Bonnaterre
William Guy Whittingham
Jane Elizabeth Wibley
Mafalda Nina
Original Assignee
Syngenta Ltd
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Ltd, Syngenta Participations Ag filed Critical Syngenta Ltd
Publication of BRPI0810679A2 publication Critical patent/BRPI0810679A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A01N43/42Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647Triazoles; Hydrogenated triazoles
    • A01N43/6531,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BRPI0810679-7A2A 2007-04-26 2008-04-16 Derivados de 4-aza indol e seu uso como fungicidas BRPI0810679A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0708141.7A GB0708141D0 (en) 2007-04-26 2007-04-26 Improvements in or relating to organic compounds
PCT/GB2008/001348 WO2008132434A2 (en) 2007-04-26 2008-04-16 4-aza indole derivatives and their use as fungicides

Publications (1)

Publication Number Publication Date
BRPI0810679A2 true BRPI0810679A2 (pt) 2014-10-07

Family

ID=38170765

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0810679-7A2A BRPI0810679A2 (pt) 2007-04-26 2008-04-16 Derivados de 4-aza indol e seu uso como fungicidas

Country Status (20)

Country Link
US (1) US8084395B2 (pt)
EP (1) EP2136640A2 (pt)
JP (1) JP2010525039A (pt)
KR (1) KR20100015918A (pt)
CN (1) CN101784191A (pt)
AR (1) AR066310A1 (pt)
AU (1) AU2008244055A1 (pt)
BR (1) BRPI0810679A2 (pt)
CA (1) CA2682773A1 (pt)
CL (1) CL2008001214A1 (pt)
CO (1) CO6140003A2 (pt)
CR (1) CR11076A (pt)
EC (1) ECSP099699A (pt)
GB (1) GB0708141D0 (pt)
IL (1) IL201195A0 (pt)
MX (1) MX2009011337A (pt)
RU (1) RU2009143567A (pt)
TW (1) TW200847926A (pt)
WO (1) WO2008132434A2 (pt)
ZA (1) ZA200906887B (pt)

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ATE541845T1 (de) * 2007-08-29 2012-02-15 Schering Corp 2,3-substituierte azaindolderivate zur behandlung von virusinfektionen
WO2010046215A2 (en) * 2008-10-21 2010-04-29 Syngenta Participations Ag Diaza-indole derivatives and their use as fungicides
DE102008052943A1 (de) * 2008-10-23 2010-04-29 Merck Patent Gmbh Azaindolderivate
EP2198710A1 (de) 2008-12-19 2010-06-23 Bayer CropScience AG Verwendung von 5-Pyridin-4yl-(1,3)Thiazole zur Bekämpfung phytopathogener Pilze
US9593108B2 (en) 2009-04-06 2017-03-14 Ptc Therapeutics, Inc. Compounds and methods for antiviral treatment
EP2245936A1 (en) 2009-04-27 2010-11-03 Bayer CropScience AG Use of 4-aza indole derivatives for the reduction of mycotoxin contamination
AR081810A1 (es) 2010-04-07 2012-10-24 Bayer Cropscience Ag Piridinilpirazoles biciclicos
JP5790440B2 (ja) 2010-12-01 2015-10-07 住友化学株式会社 ピリミジン化合物およびその有害生物防除用途
WO2012084678A1 (en) * 2010-12-23 2012-06-28 Syngenta Participations Ag Novel imidazoles useful as plant fungicides
EP2487159A1 (en) 2011-02-11 2012-08-15 MSD Oss B.V. RorgammaT inhibitors
US9055745B2 (en) 2011-04-13 2015-06-16 Natureza, Inc. Compositions for internal and external insecticides, ovicides, repellents and wound healing
CN103159663B (zh) * 2011-12-09 2014-09-17 中国科学院大连化学物理研究所 一种由联二烯衍生物制备吡咯衍生物的方法
WO2014026330A1 (en) 2012-08-15 2014-02-20 Merck Sharp & Dohme Corp. 3-AMINOCYCLOALKYL COMPOUNDS AS RORgammaT INHIBITORS AND USES THEREOF
WO2014026329A1 (en) 2012-08-15 2014-02-20 Merck Sharp & Dohme Corp. N-alkylated indole and indazole compounds as rorgammat inhibitors and uses thereof
WO2014026327A1 (en) 2012-08-15 2014-02-20 Merck Sharp & Dohme Corp. 4-heteroaryl substituted benzoic acid compounds as rorgammat inhibitors and uses thereof
JP2016135742A (ja) * 2013-03-29 2016-07-28 日本農薬株式会社 縮合複素環化合物又はその塩類及び該化合物を含有する農園芸用殺虫剤並びにその使用方法
RS58361B1 (sr) * 2013-07-31 2019-03-29 Merck Patent Gmbh Piridini, pirimidini i pirazini, kao inhibitori btk i njihova upotreba
AR103232A1 (es) 2014-12-22 2017-04-26 Bristol Myers Squibb Co ANTAGONISTAS DE TGFbR
CA2975997A1 (en) 2015-02-11 2016-08-18 Merck Sharp & Dohme Corp. Substituted pyrazole compounds as rorgammat inhibitors and uses thereof
US10344000B2 (en) 2015-10-27 2019-07-09 Merck Sharp & Dohme Corp. Substituted bicyclic pyrazole compounds as RORgammaT inhibitors and uses thereof
EP3368535B1 (en) 2015-10-27 2020-12-02 Merck Sharp & Dohme Corp. Heteroaryl substituted benzoic acids as rorgammat inhibitors and uses thereof
JP2018535958A (ja) 2015-10-27 2018-12-06 メルク・シャープ・アンド・ドーム・コーポレーションMerck Sharp & Dohme Corp. RORγT阻害薬としての置換インダゾール化合物及びその使用
WO2018003976A1 (ja) * 2016-07-01 2018-01-04 日本農薬株式会社 N‐アルキルスルホニル縮合複素環化合物又はその塩類及び該化合物を含有する殺虫剤並びにその使用方法
BR112019013266B1 (pt) * 2016-12-27 2022-10-11 Nihon Nohyaku Co., Ltd Composto de 4h-pirrolopiridina ou o sal deste, uso do mesmo, métodos para uso de um inseticida agrícola e hortícola e para controle de pragas agrícolas e hortícolas, composição compreendendo o dito composto e seu uso
CN111164081B (zh) * 2017-09-26 2022-08-12 住友化学株式会社 杂环化合物和含有该杂环化合物的有害节肢动物防除剂
WO2019077345A1 (en) 2017-10-18 2019-04-25 Redag Crop Protection Ltd BENZIMIDAZOLE COMPOUNDS AS AGRICULTURAL CHEMICALS
FI3728252T3 (fi) 2017-12-18 2023-10-18 Bristol Myers Squibb Co 4-atsaindoliyhdisteitä
CN110156775A (zh) * 2018-02-12 2019-08-23 新发药业有限公司 一种吡昔替尼的简便制备方法
LT3796975T (lt) 2018-05-22 2023-12-11 Orsobio, Inc. Sulfonilaminobenzamido dariniai
TWI748194B (zh) 2018-06-28 2021-12-01 德商菲尼克斯 Fxr有限責任公司 含有雙環核心部分之新穎lxr調節劑
EP3921317B1 (en) 2019-02-07 2023-08-02 Bayer Aktiengesellschaft 3-amino-2-[2-(acylamino)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one as csnk1 inhibitors
EP3976610A1 (en) * 2019-05-29 2022-04-06 Syngenta Crop Protection AG Microbiocidal derivatives
WO2022023340A1 (en) 2020-07-29 2022-02-03 Bayer Aktiengesellschaft Substituted heterocyclic compounds and therapeutic uses thereof
EP4188928B1 (en) 2020-07-29 2024-07-24 Bayer Aktiengesellschaft Substituted 1 h-pyrrolo[3,2-b]pyridin compounds and methods of use thereof
CN112661694B (zh) * 2020-12-11 2023-04-11 西安凯立新材料股份有限公司 一种4-(二甲氧基甲基)-哌啶的制备方法
EP4267571A1 (en) * 2020-12-22 2023-11-01 Novartis AG Pyrrolo[3,2-b]pyridine derivatives useful in treating conditions associated with cgas
EP4469457A4 (en) * 2022-01-27 2026-01-21 Broad Inst Inc CSNK1 SUBSTITUTE HETEROCYCLIC INHIBITORS
CN115124527B (zh) * 2022-05-31 2024-03-12 武汉智汇农耀科技有限公司 一种杂环酰胺-氮杂吲哚类化合物及其制备方法和应用、一种除草剂
CN118440080B (zh) * 2024-05-08 2024-12-20 广东省科学院微生物研究所(广东省微生物分析检测中心) 三苯胺类阳离子化合物及其制备方法和应用

Family Cites Families (3)

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Publication number Priority date Publication date Assignee Title
BR9812944A (pt) 1997-10-20 2000-08-08 Hoffmann La Roche Inibidores bicìclicos da cinase
WO2004014922A1 (en) * 2002-08-10 2004-02-19 Astex Technology Limited 3-(carbonyl) 1h-indazole compounds as cyclin dependent kinases (cdk) inhibitors
CA2640502A1 (en) * 2006-01-30 2007-08-02 Max-Planck Gesellschaft Zur Foerderung Der Wissenschaften E.V. Pesticidal composition comprising indole derivates

Also Published As

Publication number Publication date
ZA200906887B (en) 2012-03-28
CO6140003A2 (es) 2010-03-19
WO2008132434A3 (en) 2009-10-15
US20100184598A1 (en) 2010-07-22
IL201195A0 (en) 2010-05-17
EP2136640A2 (en) 2009-12-30
CN101784191A (zh) 2010-07-21
RU2009143567A (ru) 2011-06-10
US8084395B2 (en) 2011-12-27
TW200847926A (en) 2008-12-16
AU2008244055A1 (en) 2008-11-06
GB0708141D0 (en) 2007-06-06
ECSP099699A (es) 2009-11-30
AR066310A1 (es) 2009-08-12
CA2682773A1 (en) 2008-11-06
CL2008001214A1 (es) 2008-11-03
MX2009011337A (es) 2009-11-05
KR20100015918A (ko) 2010-02-12
JP2010525039A (ja) 2010-07-22
WO2008132434A2 (en) 2008-11-06
CR11076A (es) 2009-12-30

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B11E Dismissal acc. art. 34 of ipl - requirements for examination incomplete
B11T Dismissal of application maintained [chapter 11.20 patent gazette]