BRPI0821349A2 - compostos antivirais heterocíclicos - Google Patents

compostos antivirais heterocíclicos

Info

Publication number
BRPI0821349A2
BRPI0821349A2 BRPI0821349A BRPI0821349A BRPI0821349A2 BR PI0821349 A2 BRPI0821349 A2 BR PI0821349A2 BR PI0821349 A BRPI0821349 A BR PI0821349A BR PI0821349 A BRPI0821349 A BR PI0821349A BR PI0821349 A2 BRPI0821349 A2 BR PI0821349A2
Authority
BR
Brazil
Prior art keywords
antiviral compounds
heterocyclic antiviral
heterocyclic
compounds
antiviral
Prior art date
Application number
BRPI0821349A
Other languages
English (en)
Inventor
J Billedeau Roland
Kevin Sweeney Zachary
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40262294&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0821349(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BRPI0821349A2 publication Critical patent/BRPI0821349A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4162—1,2-Diazoles condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BRPI0821349A 2007-12-21 2008-12-11 compostos antivirais heterocíclicos BRPI0821349A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1614207P 2007-12-21 2007-12-21
PCT/EP2008/067274 WO2009080534A1 (en) 2007-12-21 2008-12-11 Heterocyclic antiviral compounds

Publications (1)

Publication Number Publication Date
BRPI0821349A2 true BRPI0821349A2 (pt) 2019-09-24

Family

ID=40262294

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0821349A BRPI0821349A2 (pt) 2007-12-21 2008-12-11 compostos antivirais heterocíclicos

Country Status (18)

Country Link
US (1) US8063028B2 (pt)
EP (1) EP2225239B1 (pt)
JP (1) JP5411160B2 (pt)
KR (2) KR101610415B1 (pt)
CN (1) CN101903382B (pt)
AR (1) AR069789A1 (pt)
AU (1) AU2008340422B2 (pt)
BR (1) BRPI0821349A2 (pt)
CA (1) CA2709348C (pt)
CL (1) CL2008003786A1 (pt)
ES (1) ES2526649T3 (pt)
IL (1) IL205863A (pt)
MX (1) MX2010006397A (pt)
PE (1) PE20091177A1 (pt)
RU (1) RU2495878C2 (pt)
TW (1) TWI445533B (pt)
WO (1) WO2009080534A1 (pt)
ZA (1) ZA201003815B (pt)

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US20110053931A1 (en) * 2006-06-08 2011-03-03 John Gaudino Quinoline compounds and methods of use
DE102007026341A1 (de) 2007-06-06 2008-12-11 Merck Patent Gmbh Benzoxazolonderivate
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DE102007061963A1 (de) 2007-12-21 2009-06-25 Merck Patent Gmbh Pyridazinonderivate
DE102008019907A1 (de) 2008-04-21 2009-10-22 Merck Patent Gmbh Pyridazinonderivate
DE102008028905A1 (de) 2008-06-18 2009-12-24 Merck Patent Gmbh 3-(3-Pyrimidin-2-yl-benzyl)-[1,2,4]triazolo[4,3-b]pyridazinderivate
WO2010059771A1 (en) 2008-11-20 2010-05-27 Osi Pharmaceuticals, Inc. Substituted pyrrolo[2,3-b]-pyridines and-pyrazines
MX2011006682A (es) 2008-12-22 2011-07-13 Merck Patent Gmbh Nuevas formas polimorficas de dihidrogeno-fosfato de 6-(1-metil-1h-pirazol-4-il)-2-{3-[5-(2-morfolin-4-il-etoxi)-pirim idin-2-il]-bencil}-2h-piridazin-3-ona y procesos para su preparacion.
US20120232062A1 (en) * 2009-10-20 2012-09-13 Eiger Biopharmaceuticals, Inc. Azaindazoles to treat flaviviridae virus infection
CN102639504A (zh) 2009-11-21 2012-08-15 弗·哈夫曼-拉罗切有限公司 杂环抗病毒化合物
WO2011143646A1 (en) * 2010-05-14 2011-11-17 OSI Pharmaceuticals, LLC Fused bicyclic kinase inhibitors
AR081039A1 (es) 2010-05-14 2012-05-30 Osi Pharmaceuticals Llc Inhibidores biciclicos fusionados de quinasa
US10872283B2 (en) 2018-10-31 2020-12-22 United Services Automobile Association (Usaa) Wireless communications device with concealed value
PY1999323A (es) * 2018-11-28 2020-10-29 Bayer Ag (tio)amidas de piridazina como compuestos fungicidas
CN111153775B (zh) * 2020-01-16 2023-04-28 江苏理工学院 一种三氯生甲酯的制备方法
WO2026042788A1 (ja) * 2024-08-20 2026-02-26 塩野義製薬株式会社 複素環誘導体

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US4569790A (en) 1984-03-28 1986-02-11 Cetus Corporation Process for recovering microbially produced interleukin-2 and purified recombinant interleukin-2 compositions
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Also Published As

Publication number Publication date
EP2225239A1 (en) 2010-09-08
CA2709348A1 (en) 2009-07-02
RU2010129548A (ru) 2012-01-27
KR20100095606A (ko) 2010-08-31
JP5411160B2 (ja) 2014-02-12
WO2009080534A1 (en) 2009-07-02
KR101610607B1 (ko) 2016-04-07
KR20150070440A (ko) 2015-06-24
RU2495878C2 (ru) 2013-10-20
TW200930372A (en) 2009-07-16
ZA201003815B (en) 2011-02-23
US8063028B2 (en) 2011-11-22
IL205863A0 (en) 2010-11-30
AR069789A1 (es) 2010-02-17
CA2709348C (en) 2016-07-19
CN101903382B (zh) 2012-11-28
AU2008340422A1 (en) 2009-07-02
AU2008340422B2 (en) 2014-06-19
ES2526649T3 (es) 2015-01-14
KR101610415B1 (ko) 2016-04-07
CL2008003786A1 (es) 2010-02-19
PE20091177A1 (es) 2009-08-03
MX2010006397A (es) 2010-07-05
EP2225239B1 (en) 2014-10-22
TWI445533B (zh) 2014-07-21
CN101903382A (zh) 2010-12-01
JP2011506535A (ja) 2011-03-03
IL205863A (en) 2016-08-31
US20090170856A1 (en) 2009-07-02

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]
B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2543 DE 01-10-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.