BRPI0911622A2 - derivados de benzoxepina e benzociclo-heptano. - Google Patents

derivados de benzoxepina e benzociclo-heptano.

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Publication number
BRPI0911622A2
BRPI0911622A2 BRPI0911622A BRPI0911622A BRPI0911622A2 BR PI0911622 A2 BRPI0911622 A2 BR PI0911622A2 BR PI0911622 A BRPI0911622 A BR PI0911622A BR PI0911622 A BRPI0911622 A BR PI0911622A BR PI0911622 A2 BRPI0911622 A2 BR PI0911622A2
Authority
BR
Brazil
Prior art keywords
benzoxepine
benzocycloheptane
derivatives
benzocycloheptane derivatives
Prior art date
Application number
BRPI0911622A
Other languages
English (en)
Inventor
Alain Philippe Poncelet
Bruno Schoentjes
Joannes Theodorus Maria Linders
Julien Georges Pierre-Olivier Doyon
Lieven Meerpoel
Luc August Laurentius Ver Donck
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of BRPI0911622A2 publication Critical patent/BRPI0911622A2/pt
Publication of BRPI0911622B1 publication Critical patent/BRPI0911622B1/pt
Publication of BRPI0911622B8 publication Critical patent/BRPI0911622B8/pt

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BRPI0911622A 2008-04-28 2009-04-27 derivados de benzoxepina e benzociclo-heptano, seu processo de preparação, seu uso e composição farmacêutica que os compreende BRPI0911622B8 (pt)

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RU2496769C2 (ru) * 2008-04-28 2013-10-27 Янссен Фармацевтика Нв Производные бензоциклогептана и бензоксепина
US9643947B2 (en) 2013-08-28 2017-05-09 Northwestern University 7-membered fused heterocycles and methods of their synthesis
US10065948B2 (en) 2014-06-02 2018-09-04 Chdi Foundation, Inc. Histone deacetylase inhibitors and compositions and methods of use thereof

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FR2319332A1 (fr) * 1975-07-28 1977-02-25 Roussel Uclaf Nouveaux derives de l'aminobenzocycloheptene et leurs sels, procede de preparation et application a titre de medicaments desdits produits
US4736031A (en) * 1985-06-10 1988-04-05 Takeda Chemical Industries, Ltd. 2-(piperazinylalkyl)-1-benzothiepin, 1-benzoxepin, and 1,5-benzodioxepin derivatives
DE19755480A1 (de) * 1997-12-13 1999-06-24 Gruenenthal Gmbh Substituierte heterocyclische Benzocycloalkene und ihre Verwendung als analgetisch wirksame Substanzen
RU2204390C2 (ru) * 1998-01-14 2003-05-20 Ниппон Синяку Ко., Лтд. Активаторы калиевых каналов
JPWO2004014412A1 (ja) 2002-08-09 2005-12-02 科研製薬株式会社 心筋細胞保護剤
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US20140187557A1 (en) 2014-07-03
RU2496769C2 (ru) 2013-10-27
US20120322796A1 (en) 2012-12-20
CN102076654A (zh) 2011-05-25
RU2010148433A (ru) 2012-06-10
WO2009133052A1 (en) 2009-11-05
ES2433215T3 (es) 2013-12-10
BRPI0911622B1 (pt) 2021-05-11
US20110046139A1 (en) 2011-02-24
US8278466B2 (en) 2012-10-02
EP2297089B1 (en) 2013-07-31
AU2009242219A1 (en) 2009-11-05
PL2297089T3 (pl) 2013-12-31
CA2722122A1 (en) 2009-11-05
JP5754811B2 (ja) 2015-07-29
EP2297089A1 (en) 2011-03-23
US8703973B2 (en) 2014-04-22
US9040725B2 (en) 2015-05-26
BRPI0911622B8 (pt) 2021-05-25
MX2010011767A (es) 2010-11-30
CN102076654B (zh) 2014-07-23
CA2722122C (en) 2017-01-03
AU2009242219B2 (en) 2013-03-21

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