BRPI0912171A2 - composição farmacêutica - Google Patents

composição farmacêutica

Info

Publication number
BRPI0912171A2
BRPI0912171A2 BRPI0912171A BRPI0912171A BRPI0912171A2 BR PI0912171 A2 BRPI0912171 A2 BR PI0912171A2 BR PI0912171 A BRPI0912171 A BR PI0912171A BR PI0912171 A BRPI0912171 A BR PI0912171A BR PI0912171 A2 BRPI0912171 A2 BR PI0912171A2
Authority
BR
Brazil
Prior art keywords
pharmaceutical composition
pharmaceutical
composition
Prior art date
Application number
BRPI0912171A
Other languages
English (en)
Inventor
Dota Atsuyoshi
Imoto Kenji
Matsuda Mamoru
Kato Masatomo
Takai Miwa
Matsuyama Takahiro
Kurose Tatsuji
Mori Toshiyuki
Hagiwara Yumi
Original Assignee
Santen Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Santen Pharmaceutical Co Ltd filed Critical Santen Pharmaceutical Co Ltd
Publication of BRPI0912171A2 publication Critical patent/BRPI0912171A2/pt
Publication of BRPI0912171A8 publication Critical patent/BRPI0912171A8/pt
Publication of BRPI0912171B1 publication Critical patent/BRPI0912171B1/pt
Publication of BRPI0912171B8 publication Critical patent/BRPI0912171B8/pt

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Classifications

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
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    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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BRPI0912171A 2008-05-12 2009-05-12 composto ativador de receptor de glicocorticoide, e, composição BRPI0912171B8 (pt)

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WO2012108455A1 (ja) * 2011-02-09 2012-08-16 参天製薬株式会社 ３－ヒドロキシ－６Ｈ－ベンゾ［ｃ］クロメン－６－オン誘導体およびその製造方法
WO2013108921A1 (ja) * 2012-01-20 2013-07-25 参天製薬株式会社 １，２－ジヒドロキノリン誘導体またはその塩の工業的製造方法およびその製造中間体
EP2981077B1 (en) * 2013-03-28 2017-09-27 Aisin Seiki Kabushiki Kaisha Periphery monitoring device and program
CN107922356A (zh) 2015-08-25 2018-04-17 参天制药株式会社 [4‑(1,3,3‑三甲基‑2‑氧代‑3,4‑二氢‑1h‑喹喔啉‑7‑基)苯氧基]乙基氧基化合物或其盐
US11433090B2 (en) 2017-06-16 2022-09-06 The Doshisha mTOR-inhibitor-containing medicine for treating or preventing ophthalmic symptoms, disorders, or diseases, and application thereof
WO2018230713A1 (ja) 2017-06-16 2018-12-20 学校法人同志社 カスパーゼ阻害活性を有する化合物、これらの化合物を含む、角膜内皮の症状、障害または疾患を治療または予防するための医薬およびその応用
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PL1944290T3 (pl) 2005-09-14 2014-07-31 Ayumi Pharmaceutical Corp Nowa pochodna 1-2-dihydrochinoliny mająca aktywność wiązania glukokortykoidowego receptora
ES2391910T3 (es) * 2006-11-14 2012-12-03 Santen Pharmaceutical Co., Ltd Derivado de 1,2-dihidroquinolina que tiene un grupo (fenil sustituido o heterociclil sustituido)carboniloxi-alquilo inferior y un grupo fenilo introducido por éster como sustituyentes
JP2008255112A (ja) * 2007-03-13 2008-10-23 Santen Pharmaceut Co Ltd ２，２，４−トリメチル−６−フェニル−１，２−ジヒドロキノリン誘導体からなるグルココルチコイド受容体アゴニスト

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CA2724055A1 (en) 2009-11-19
TW200950781A (en) 2009-12-16
EA201071296A1 (ru) 2011-06-30
AU2009247250B2 (en) 2014-04-10
BRPI0912171A8 (pt) 2017-12-12
MY158747A (en) 2016-11-15
US20110118260A1 (en) 2011-05-19
WO2009139361A1 (ja) 2009-11-19
BRPI0912171B8 (pt) 2021-05-25
MX2010012303A (es) 2011-03-30
EP2319835A4 (en) 2011-12-28
EP2319835B1 (en) 2016-04-13
JP5635743B2 (ja) 2014-12-03
CN105395550B (zh) 2018-07-17
EP2319835A1 (en) 2011-05-11
ES2574987T3 (es) 2016-06-23
TWI510240B (zh) 2015-12-01
EA019091B1 (ru) 2014-01-30
GEP20146061B (en) 2014-03-25
JP2009298775A (ja) 2009-12-24
CN105395550A (zh) 2016-03-16
US8426406B2 (en) 2013-04-23
CN102089283B (zh) 2015-11-25
BRPI0912171B1 (pt) 2020-11-03
KR20110010634A (ko) 2011-02-01
AU2009247250A1 (en) 2009-11-19
UA102101C2 (ru) 2013-06-10
CA2724055C (en) 2016-08-02

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