BRPI0916692A2 - processo para a preparação de um composto, e, composto - Google Patents

processo para a preparação de um composto, e, composto

Info

Publication number
BRPI0916692A2
BRPI0916692A2 BRPI0916692A BRPI0916692A BRPI0916692A2 BR PI0916692 A2 BRPI0916692 A2 BR PI0916692A2 BR PI0916692 A BRPI0916692 A BR PI0916692A BR PI0916692 A BRPI0916692 A BR PI0916692A BR PI0916692 A2 BRPI0916692 A2 BR PI0916692A2
Authority
BR
Brazil
Prior art keywords
compound
preparing
Prior art date
Application number
BRPI0916692A
Other languages
English (en)
Inventor
Hans J Sanders
Jeroen Van Rheenen
Josephus H M Lange
Original Assignee
Abbott Healthcare Products Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Healthcare Products Bv filed Critical Abbott Healthcare Products Bv
Publication of BRPI0916692A2 publication Critical patent/BRPI0916692A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BRPI0916692A 2008-08-01 2009-07-30 processo para a preparação de um composto, e, composto BRPI0916692A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08161619 2008-08-01
PCT/EP2009/059844 WO2010012797A2 (en) 2008-08-01 2009-07-30 Synthesis of 3,4-diaryl-4,5-dihydro-(1h)-pyrazole-1- carboxamidine derivatives

Publications (1)

Publication Number Publication Date
BRPI0916692A2 true BRPI0916692A2 (pt) 2016-05-17

Family

ID=40380031

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0916692A BRPI0916692A2 (pt) 2008-08-01 2009-07-30 processo para a preparação de um composto, e, composto

Country Status (12)

Country Link
EP (1) EP2321280A2 (pt)
JP (1) JP2011529868A (pt)
KR (1) KR20110042095A (pt)
CN (1) CN102089284A (pt)
AR (1) AR072539A1 (pt)
AU (1) AU2009275838A1 (pt)
BR (1) BRPI0916692A2 (pt)
CA (1) CA2729969A1 (pt)
EA (1) EA201170284A1 (pt)
MX (1) MX2011001211A (pt)
TW (1) TW201010981A (pt)
WO (1) WO2010012797A2 (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR079935A1 (es) 2010-01-29 2012-02-29 Abbott Healthcare Products Bv Sintesis de derivados de pirazolin carboxamidina sustituida
WO2020236411A1 (en) * 2019-05-17 2020-11-26 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services A scalable synthesis of dual-target inhibitor of cannabinoid-1 receptor and inducible nitric oxide synthase
CN111686806B (zh) * 2020-05-29 2022-09-30 黑龙江大学 一种聚[2-(3-噻吩基)乙醇]/石墨相氮化碳复合可见光催化剂的制备方法及应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2074179A1 (en) * 1990-01-31 1991-08-01 Charles R. Harrison Arthropodicidal pyrazolines, pyrazolidines and hyrazines
DE4005114A1 (de) * 1990-02-17 1991-08-22 Bayer Ag Substituierte pyrazolinderivate
PL208098B1 (pl) * 2000-03-23 2011-03-31 Solvay Pharm Bv Pochodne 4,5-dihydro-1H-pirazolu, kompozycja farmaceutyczna, sposób wytwarzania związków oraz ich zastosowanie
KR100950430B1 (ko) * 2001-09-21 2010-04-02 솔베이 파마슈티칼스 비. 브이 효력있는 cb1-길항 작용을 가지는4,5-디하이드로-1h-피라졸 유도체

Also Published As

Publication number Publication date
TW201010981A (en) 2010-03-16
AR072539A1 (es) 2010-09-01
JP2011529868A (ja) 2011-12-15
MX2011001211A (es) 2011-03-29
WO2010012797A2 (en) 2010-02-04
CA2729969A1 (en) 2010-02-04
EA201170284A1 (ru) 2011-06-30
AU2009275838A1 (en) 2010-02-04
CN102089284A (zh) 2011-06-08
EP2321280A2 (en) 2011-05-18
KR20110042095A (ko) 2011-04-22
WO2010012797A3 (en) 2010-04-22

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal acc. article 33 of ipl - extension of time limit for request of examination expired