BRPI0918726A2 - derivados de 1-amino-alquilciclohexano para o tratamento de deficiência cognitiva em tinido - Google Patents
derivados de 1-amino-alquilciclohexano para o tratamento de deficiência cognitiva em tinidoInfo
- Publication number
- BRPI0918726A2 BRPI0918726A2 BRPI0918726A BRPI0918726A BRPI0918726A2 BR PI0918726 A2 BRPI0918726 A2 BR PI0918726A2 BR PI0918726 A BRPI0918726 A BR PI0918726A BR PI0918726 A BRPI0918726 A BR PI0918726A BR PI0918726 A2 BRPI0918726 A2 BR PI0918726A2
- Authority
- BR
- Brazil
- Prior art keywords
- tinnitus
- amino
- treatment
- cognitive impairment
- alkylcyclohexane derivatives
- Prior art date
Links
- 208000028698 Cognitive impairment Diseases 0.000 title 1
- 208000009205 Tinnitus Diseases 0.000 title 1
- 208000010877 cognitive disease Diseases 0.000 title 1
- 231100000886 tinnitus Toxicity 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Emergency Medicine (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US19162608P | 2008-09-10 | 2008-09-10 | |
| EP08015947 | 2008-09-10 | ||
| PCT/EP2009/006366 WO2010028769A1 (en) | 2008-09-10 | 2009-09-02 | 1-amino-alkylcyclohexane derivatives for the treatment of cognitive impairment in tinnitus |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0918726A2 true BRPI0918726A2 (pt) | 2015-12-01 |
Family
ID=40342435
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0918726A BRPI0918726A2 (pt) | 2008-09-10 | 2009-09-02 | derivados de 1-amino-alquilciclohexano para o tratamento de deficiência cognitiva em tinido |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20110178179A1 (pt) |
| EP (1) | EP2344144A1 (pt) |
| JP (1) | JP2012501304A (pt) |
| KR (1) | KR20110050739A (pt) |
| CN (1) | CN102123703A (pt) |
| AU (1) | AU2009291244A1 (pt) |
| BR (1) | BRPI0918726A2 (pt) |
| CA (1) | CA2731660A1 (pt) |
| IL (1) | IL211641A0 (pt) |
| MX (1) | MX2011002481A (pt) |
| RU (1) | RU2011113733A (pt) |
| WO (1) | WO2010028769A1 (pt) |
| ZA (1) | ZA201101174B (pt) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2548552B1 (en) * | 2007-09-12 | 2015-11-18 | Merz Pharma GmbH & Co. KGaA | Titration package for 1-amino-alkylcyclohexanes |
| US20150374705A1 (en) | 2012-02-14 | 2015-12-31 | Shanghai Institues for Biological Sciences | Substances for treatment or relief of pain |
| CN106535883A (zh) * | 2014-04-28 | 2017-03-22 | 杏林制药株式会社 | 耳鸣患者的治疗用药剂 |
| WO2020163588A1 (en) * | 2019-02-08 | 2020-08-13 | Board Of Trustees Of Southern Illinois University | Neuronal nicotinic acetylcholine receptor partial agonists as therapeutics for chronic tinnitus |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW200418446A (en) * | 2002-10-24 | 2004-10-01 | Merz Pharma Gmbh & Co Kgaa | Combination therapy using 1-aminocyclohexane derivatives and acetylcholinesterase inhibitors |
| US20060002999A1 (en) * | 2004-06-17 | 2006-01-05 | Forest Laboratories, Inc. | Immediate release formulations of 1-aminocyclohexane compounds, memantine and neramexane |
| US20070123555A1 (en) * | 2005-09-30 | 2007-05-31 | Cypress Bioscience, Inc. | Prevention and treatment of hearing disorders |
| US20070141148A1 (en) * | 2005-11-30 | 2007-06-21 | Merz Pharma Gmbh & Co. Kgaa | Neramexane MR matrix tablet |
-
2009
- 2009-09-02 BR BRPI0918726A patent/BRPI0918726A2/pt not_active Application Discontinuation
- 2009-09-02 CA CA2731660A patent/CA2731660A1/en not_active Abandoned
- 2009-09-02 WO PCT/EP2009/006366 patent/WO2010028769A1/en not_active Ceased
- 2009-09-02 EP EP09778288A patent/EP2344144A1/en not_active Withdrawn
- 2009-09-02 AU AU2009291244A patent/AU2009291244A1/en not_active Abandoned
- 2009-09-02 RU RU2011113733/15A patent/RU2011113733A/ru unknown
- 2009-09-02 KR KR1020117008126A patent/KR20110050739A/ko not_active Ceased
- 2009-09-02 MX MX2011002481A patent/MX2011002481A/es unknown
- 2009-09-02 US US12/998,033 patent/US20110178179A1/en not_active Abandoned
- 2009-09-02 CN CN2009801312987A patent/CN102123703A/zh active Pending
- 2009-09-02 JP JP2011524271A patent/JP2012501304A/ja active Pending
-
2011
- 2011-02-14 ZA ZA2011/01174A patent/ZA201101174B/en unknown
- 2011-03-08 IL IL211641A patent/IL211641A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL211641A0 (en) | 2011-05-31 |
| CN102123703A (zh) | 2011-07-13 |
| RU2011113733A (ru) | 2012-10-20 |
| AU2009291244A1 (en) | 2010-03-18 |
| CA2731660A1 (en) | 2010-03-18 |
| EP2344144A1 (en) | 2011-07-20 |
| US20110178179A1 (en) | 2011-07-21 |
| WO2010028769A1 (en) | 2010-03-18 |
| JP2012501304A (ja) | 2012-01-19 |
| KR20110050739A (ko) | 2011-05-16 |
| ZA201101174B (en) | 2011-10-26 |
| MX2011002481A (es) | 2011-04-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
| B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] |