BRPI0922042A2 - derivados de 1-arilpirazol diméricos - Google Patents

derivados de 1-arilpirazol diméricos

Info

Publication number
BRPI0922042A2
BRPI0922042A2 BRPI0922042A BRPI0922042A BRPI0922042A2 BR PI0922042 A2 BRPI0922042 A2 BR PI0922042A2 BR PI0922042 A BRPI0922042 A BR PI0922042A BR PI0922042 A BRPI0922042 A BR PI0922042A BR PI0922042 A2 BRPI0922042 A2 BR PI0922042A2
Authority
BR
Brazil
Prior art keywords
dimeric
arylpyrazole derivatives
arylpyrazole
derivatives
Prior art date
Application number
BRPI0922042A
Other languages
English (en)
Inventor
Charles Q Meng
Original Assignee
Merial Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merial Ltd filed Critical Merial Ltd
Publication of BRPI0922042A2 publication Critical patent/BRPI0922042A2/pt
Publication of BRPI0922042B1 publication Critical patent/BRPI0922042B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pest Control & Pesticides (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Agronomy & Crop Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
BRPI0922042A 2008-11-19 2009-11-18 derivados de 1-arilpirazol diméricos BRPI0922042B1 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11602108P 2008-11-19 2008-11-19
PCT/US2009/064981 WO2010059719A2 (en) 2008-11-19 2009-11-18 Dimeric 1-arylpyrazole derivatives

Publications (2)

Publication Number Publication Date
BRPI0922042A2 true BRPI0922042A2 (pt) 2016-11-01
BRPI0922042B1 BRPI0922042B1 (pt) 2020-01-28

Family

ID=42034586

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0922042A BRPI0922042B1 (pt) 2008-11-19 2009-11-18 derivados de 1-arilpirazol diméricos

Country Status (12)

Country Link
US (1) US8642636B2 (pt)
EP (1) EP2364300B1 (pt)
JP (1) JP2012509338A (pt)
CN (1) CN102264706A (pt)
AU (1) AU2009316710B2 (pt)
BR (1) BRPI0922042B1 (pt)
CA (2) CA2743553C (pt)
EA (1) EA020923B1 (pt)
ES (1) ES2605811T3 (pt)
MX (1) MX2011005214A (pt)
NZ (1) NZ592985A (pt)
WO (1) WO2010059719A2 (pt)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102001364B1 (ko) 2011-05-13 2019-07-22 어레이 바이오파마 인크. Trka 키나제 저해제로서의 피롤리디닐 유레아 및 피롤리디닐 티오유레아 화합물
WO2014078378A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. Pyrrolidinyl urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
WO2014078328A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. N-bicyclic aryl,n'-pyrazolyl urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
WO2014078331A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. N-(arylalkyl)-n'-pyrazolyl-urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
US9809578B2 (en) 2012-11-13 2017-11-07 Array Biopharma Inc. Pyrazolyl urea, thiourea, guanidine and cyanoguanidine compounds as trkA kinase inhibitors
US9822118B2 (en) 2012-11-13 2017-11-21 Array Biopharma Inc. Bicyclic heteroaryl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
RU2664541C2 (ru) 2012-11-13 2018-08-20 Эррэй Биофарма Инк. Бициклические соединения мочевины, тиомочевины, гуанидина и цианогуанидина, пригодные для лечения боли
WO2014078325A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. N-(monocyclic aryl),n'-pyrazolyl-urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
US9790178B2 (en) 2012-11-13 2017-10-17 Array Biopharma Inc. Pyrrolidinyl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
UA116455C2 (uk) 2012-11-13 2018-03-26 Еррей Біофарма Інк. Сполуки n-піролідинілсечовини, n'-піразолілсечовини, тіосечовини, гуанідину та ціаногуанідину як інгібітори кінази trka
US9981959B2 (en) 2012-11-13 2018-05-29 Array Biopharma Inc. Thiazolyl and oxazolyl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
JP2016164125A (ja) * 2013-07-02 2016-09-08 国立大学法人帯広畜産大学 バベシア症の治療剤及び予防剤
MY191956A (en) 2014-05-15 2022-07-20 Array Biopharma Inc 1-((3s,4r)-4-(3-fluorophenyl)-1-(2-methoxyethyl)pyrrolidin-3-yl)-3-(4-methyl-3-(2-methylpyrimidin-5-yl)-1-phenyl-1h-pyrazol-5-yl)urea as a trka kinase inhibitor
WO2017195173A1 (en) 2016-05-12 2017-11-16 Verdesian Life Sciences, U.S., Llc Compositions for controlling enzyme-induced urea decomposition
KR102480799B1 (ko) 2017-03-28 2022-12-22 베르데시안 라이프 사이언시스 유.에스., 엘엘씨 효소-유도된 우레아 분해를 조절하기 위한 트리아릴메탄 화합물
PL3876722T3 (pl) 2018-11-06 2026-02-23 Corteva Agriscience Llc Zabezpieczone kompozycje zawierające herbicydy pirydynokarboksylanowe i klokwintocet
DK3876726T3 (da) * 2018-11-06 2025-03-03 Corteva Agriscience Llc Sammensætninger, som omfatter pyridincarboxylat-herbicider og azolcarboxylat-safeners
EP3876730B1 (en) 2018-11-07 2025-07-02 Corteva Agriscience LLC Compositions comprising pyridine carboxylate herbicides and 4-hydroxyphenyl-pyruvate dioxygenase (hppd) inhibitor herbicides
EA202191264A1 (ru) 2018-11-07 2021-07-27 КОРТЕВА АГРИСАЙЕНС ЭлЭлСи Композиции, содержащие гербициды на основе пиридинкарбоксилата с гербицидами, представляющими собой ингибиторы фотосистемы ii и необязательно hppd
HUE072472T2 (hu) 2018-11-07 2025-11-28 Corteva Agriscience Llc Piridin-karboxilát herbicideket acetolaktát-szintáz (ALS) gátló herbicidekkel tartalmazó készítmények
EA202191265A1 (ru) 2018-11-07 2021-07-27 КОРТЕВА АГРИСАЙЕНС ЭлЭлСи Композиции, содержащие гербицид на основе пиридинкарбоксилата и гербициды, представляющие собой ингибиторы протопорфириногеноксидазы (protox)
KR102860839B1 (ko) 2018-11-07 2025-09-17 코르테바 애그리사이언스 엘엘씨 피리딘 카르복실레이트 제초제를 합성 옥신 제초제 또는 옥신 수송 억제제와 함께 포함하는 조성물
EP3886854A4 (en) 2018-11-30 2022-07-06 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof
JP7724845B2 (ja) 2020-07-24 2025-08-18 エランコ・ユーエス・インコーポレイテッド イソオキサゾリン化合物及びその中間体を作製するための方法
KR20230061465A (ko) 2020-09-04 2023-05-08 엘랑코 유에스 인코포레이티드 기호성 제형

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3966900A (en) * 1969-03-12 1976-06-29 Airwick Industries, Inc. Evaporator system comprising a stabilized pesticidal phosphoric acid ester and method for stabilizing such ester enclosed in an evaporator
MY129771A (en) * 1999-12-02 2007-04-30 Merial Ltd Control of arthropods in animals
US7262214B2 (en) * 2003-02-26 2007-08-28 Merial Limited 1-N-arylpyrazole derivatives in prevention of arthropod-borne and mosquito-borne diseases
ES2444015T3 (es) 2004-06-26 2014-02-21 Merial Limited Derivados de N-fenilpirazol como plaguicidas

Also Published As

Publication number Publication date
CA2952443A1 (en) 2010-05-27
HK1160852A1 (en) 2012-08-17
EA201100800A1 (ru) 2011-12-30
AU2009316710A1 (en) 2010-05-27
JP2012509338A (ja) 2012-04-19
EP2364300B1 (en) 2016-10-19
MX2011005214A (es) 2011-06-01
ES2605811T3 (es) 2017-03-16
AU2009316710B2 (en) 2015-08-06
BRPI0922042B1 (pt) 2020-01-28
CA2952443C (en) 2019-04-02
US20110245157A1 (en) 2011-10-06
US8642636B2 (en) 2014-02-04
EP2364300A2 (en) 2011-09-14
CA2743553A1 (en) 2010-05-27
WO2010059719A3 (en) 2010-11-18
CA2743553C (en) 2017-03-14
NZ592985A (en) 2013-04-26
WO2010059719A2 (en) 2010-05-27
CN102264706A (zh) 2011-11-30
EA020923B1 (ru) 2015-02-27

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Legal Events

Date Code Title Description
B15I Others concerning applications: loss of priority

Free format text: OBSERVA-SE QUE A PRIORIDADE REQUERIDA US 61/116,021 DE 19.11.2008 POSSUI DEPOSITANTE DIFERENTE DO INFORMADO NA ENTRADA NA FASE NACIONAL E SUA RESPECTIVA CESSAO FOI APRESENTADA EM 19/11/2012 APOS O PRAZO REGULAR DE 60 DIAS DA ENTRADA NA FASE NACIONAL QUE SE ENCERRAVA EM 18/07/2011, MOTIVO PELO QUAL SERA DADA PERDA DESTA PRIORIDADE, CONFORME AS DISPOSICOES PREVISTAS NA LEI 9.279 DE 14/05/1996 (LPI) ART. 16 7O.

B25A Requested transfer of rights approved

Owner name: MERIAL, INC. (US)

B12F Other appeals [chapter 12.6 patent gazette]
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07G Grant request does not fulfill article 229-c lpi (prior consent of anvisa) [chapter 7.7 patent gazette]

Free format text: NOTIFICACAO DE DEVOLUCAO DO PEDIDO POR NAO SE ENQUADRAR NO ART. 229-C DA LPI.

B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 28/01/2020, OBSERVADAS AS CONDICOES LEGAIS.

B25A Requested transfer of rights approved

Owner name: BOEHRINGER INGELHEIM ANIMAL HEALTH USA INC. (US)