BRPI1014876A2 - "diamidas de azetidinila como inibidores de monoacilglicerol lipase." - Google Patents

"diamidas de azetidinila como inibidores de monoacilglicerol lipase."

Info

Publication number
BRPI1014876A2
BRPI1014876A2 BRPI1014876A BRPI1014876A BRPI1014876A2 BR PI1014876 A2 BRPI1014876 A2 BR PI1014876A2 BR PI1014876 A BRPI1014876 A BR PI1014876A BR PI1014876 A BRPI1014876 A BR PI1014876A BR PI1014876 A2 BRPI1014876 A2 BR PI1014876A2
Authority
BR
Brazil
Prior art keywords
lipase inhibitors
monoacylglycerol lipase
diamides
azetidinyl
azetidinyl diamides
Prior art date
Application number
BRPI1014876A
Other languages
English (en)
Inventor
Bin Zhu
Christopher M Flores
Haiyan Bian
John Mabus
Jose Clemente
Kristen M Chevalier
Li Liu
Mark E Mcdonnell
Mark J Macielag
Peter J Connolly
Philip M Pitis
Shu-Chen Lin
Sui-Po Zhang
Yue-Mei
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of BRPI1014876A2 publication Critical patent/BRPI1014876A2/pt

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    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
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BRPI1014876A 2009-04-22 2010-04-22 "diamidas de azetidinila como inibidores de monoacilglicerol lipase." BRPI1014876A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US17165809P 2009-04-22 2009-04-22
US17164909P 2009-04-22 2009-04-22
PCT/US2010/032089 WO2010124114A1 (en) 2009-04-22 2010-04-22 Azetidinyl diamides as monoacylglycerol lipase inhibitors

Publications (1)

Publication Number Publication Date
BRPI1014876A2 true BRPI1014876A2 (pt) 2016-04-12

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Family Applications (8)

Application Number Title Priority Date Filing Date
BRPI1013540-5A BRPI1013540A2 (pt) 2009-04-22 2010-04-22 azetidinil diamidas como inibidores de monoacilglicerol lipases
BRPI1015238A BRPI1015238A2 (pt) 2009-04-22 2010-04-22 diamidas de azetidilina como inibidores de monoaciglicerol lipase
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US20110015170A1 (en) 2011-01-20
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BRPI1013545A2 (pt) 2019-09-24
ES2455744T3 (es) 2014-04-16
US20110015171A1 (en) 2011-01-20
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IL215780A0 (en) 2012-01-31
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AU2010239188B2 (en) 2016-03-31
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JP5733840B2 (ja) 2015-06-10
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CN102459167B (zh) 2015-04-01
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BRPI1013540A2 (pt) 2020-11-17
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US20130123232A1 (en) 2013-05-16
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TW201105655A (en) 2011-02-16
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WO2010124112A1 (en) 2010-10-28
BRPI1014281A2 (pt) 2019-09-24
CN102548982A (zh) 2012-07-04
AR076380A1 (es) 2011-06-08
KR20120034616A (ko) 2012-04-12
CA2759713A1 (en) 2010-10-28
AU2010239204A1 (en) 2011-11-10
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JP2012524803A (ja) 2012-10-18
BRPI1014284A2 (pt) 2017-10-10
CN102459240A (zh) 2012-05-16
KR101705697B1 (ko) 2017-02-10
US8722658B2 (en) 2014-05-13
CA2759697A1 (en) 2010-10-28
KR20110137831A (ko) 2011-12-23
AU2010238738A1 (en) 2011-11-10
IL215781A0 (en) 2012-01-31
AU2016201405A1 (en) 2016-03-24
EP2421848A1 (en) 2012-02-29
PT2421825E (pt) 2014-03-13
AU2010238736A1 (en) 2011-11-10
WO2010124119A1 (en) 2010-10-28
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US8962607B2 (en) 2015-02-24
EP2421825A1 (en) 2012-02-29
WO2010124116A1 (en) 2010-10-28
RS53235B (sr) 2014-08-29
CN102459166B (zh) 2015-03-25
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US20130123233A1 (en) 2013-05-16
US20100324012A1 (en) 2010-12-23

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