BRPI1015238A2 - diamidas de azetidilina como inibidores de monoaciglicerol lipase - Google Patents

diamidas de azetidilina como inibidores de monoaciglicerol lipase

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Publication number
BRPI1015238A2
BRPI1015238A2 BRPI1015238A BRPI1015238A BRPI1015238A2 BR PI1015238 A2 BRPI1015238 A2 BR PI1015238A2 BR PI1015238 A BRPI1015238 A BR PI1015238A BR PI1015238 A BRPI1015238 A BR PI1015238A BR PI1015238 A2 BRPI1015238 A2 BR PI1015238A2
Authority
BR
Brazil
Prior art keywords
monoaciglycerol
azetidiline
diamides
lipase inhibitors
lipase
Prior art date
Application number
BRPI1015238A
Other languages
English (en)
Inventor
Zhu Bin
M Flores Christopher
Bian Haiyan
Mabus John
Clemente Jose
Liu Li
E Mcdonnell Mark
J Macielag Mark
J Connolly Peter
M Pitis Philip
Lin Shu-Chen
Zhang Sui-Po
Zhang Yue-Mei
M Chevalier Kristen
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of BRPI1015238A2 publication Critical patent/BRPI1015238A2/pt

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    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
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BRPI1015238A 2009-04-22 2010-04-22 diamidas de azetidilina como inibidores de monoaciglicerol lipase BRPI1015238A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US17164909P 2009-04-22 2009-04-22
US17165809P 2009-04-22 2009-04-22
PCT/US2010/032095 WO2010124119A1 (en) 2009-04-22 2010-04-22 Azetidinyl diamides as monoacylglycerol lipase inhibitors

Publications (1)

Publication Number Publication Date
BRPI1015238A2 true BRPI1015238A2 (pt) 2019-09-24

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Application Number Title Priority Date Filing Date
BRPI1014876A BRPI1014876A2 (pt) 2009-04-22 2010-04-22 "diamidas de azetidinila como inibidores de monoacilglicerol lipase."
BRPI1014284A BRPI1014284A2 (pt) 2009-04-22 2010-04-22 azetidinil diamidas como inibidores da monoacilglicerol lipase
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