CA2019324A1 - Comprimes de fosinopril - Google Patents

Comprimes de fosinopril

Info

Publication number: CA2019324A1
Authority: CA; Canada
Prior art keywords: tablet formulations; fosinopril; fosinopril tablet; tablets; sodium
Prior art date: 1989-07-10
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

CA2019324A

Other languages

English (en)

Other versions

CA2019324C (fr

Inventor

Robert L. Jerzewski

Thomas M. Wong

Lewis J. Gryziewicz

Nemichand B. Jain

Ajit B. Thakur

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

ER Squibb and Sons LLC

Original Assignee

Individual

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1989-07-10

Filing date

1990-06-19

Publication date

1991-01-10

1990-06-19 Application filed by Individual filed Critical Individual

1991-01-10 Publication of CA2019324A1 publication Critical patent/CA2019324A1/fr

1996-08-20 Application granted granted Critical

1996-08-20 Publication of CA2019324C publication Critical patent/CA2019324C/fr

2010-06-19 Anticipated expiration legal-status Critical

Status Expired - Lifetime legal-status Critical Current

Links

BIDNLKIUORFRQP-XYGFDPSESA-N (2s,4s)-4-cyclohexyl-1-[2-[[(1s)-2-methyl-1-propanoyloxypropoxy]-(4-phenylbutyl)phosphoryl]acetyl]pyrrolidine-2-carboxylic acid Chemical compound C([P@@](=O)(O[C@H](OC(=O)CC)C(C)C)CC(=O)N1[C@@H](C[C@H](C1)C1CCCCC1)C(O)=O)CCCC1=CC=CC=C1 BIDNLKIUORFRQP-XYGFDPSESA-N 0.000 title 1
229960002490 fosinopril Drugs 0.000 title 1
239000007916 tablet composition Substances 0.000 title 1
239000011230 binding agent Substances 0.000 abstract 1
239000007884 disintegrant Substances 0.000 abstract 1
239000002934 diuretic Substances 0.000 abstract 1
230000001882 diuretic effect Effects 0.000 abstract 1
MVPICKVDHDWCJQ-UHFFFAOYSA-N ethyl 3-pyrrolidin-1-ylpropanoate Chemical compound CCOC(=O)CCN1CCCC1 MVPICKVDHDWCJQ-UHFFFAOYSA-N 0.000 abstract 1
239000000945 filler Substances 0.000 abstract 1
229960001880 fosinopril sodium Drugs 0.000 abstract 1
239000008172 hydrogenated vegetable oil Substances 0.000 abstract 1
239000000314 lubricant Substances 0.000 abstract 1
239000000546 pharmaceutical excipient Substances 0.000 abstract 1
229940045902 sodium stearyl fumarate Drugs 0.000 abstract 1
TVTJZMHAIQQZTL-WATAJHSMSA-M sodium;(2s,4s)-4-cyclohexyl-1-[2-[[(1s)-2-methyl-1-propanoyloxypropoxy]-(4-phenylbutyl)phosphoryl]acetyl]pyrrolidine-2-carboxylate Chemical compound [Na+].C([P@@](=O)(O[C@H](OC(=O)CC)C(C)C)CC(=O)N1[C@@H](C[C@H](C1)C1CCCCC1)C([O-])=O)CCCC1=CC=CC=C1 TVTJZMHAIQQZTL-WATAJHSMSA-M 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Chemical & Material Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
General Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Epidemiology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Biophysics (AREA)
Molecular Biology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)

CA002019324A 1989-07-10 1990-06-19 Comprimes de fosinopril Expired - Lifetime CA2019324C (fr)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US37768389A	1989-07-10	1989-07-10
US377,683		1989-07-10

Publications (2)

Publication Number	Publication Date
CA2019324A1 true CA2019324A1 (fr)	1991-01-10
CA2019324C CA2019324C (fr)	1996-08-20

Family

ID=23490122

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CA002019324A Expired - Lifetime CA2019324C (fr)	1989-07-10	1990-06-19	Comprimes de fosinopril

Country Status (8)

Country	Link
EP (1)	EP0408273B1 (fr)
JP (1)	JP2965633B2 (fr)
AT (1)	ATE100321T1 (fr)
CA (1)	CA2019324C (fr)
DD (1)	DD299154A5 (fr)
DE (1)	DE69006125T2 (fr)
DK (1)	DK0408273T3 (fr)
ES (1)	ES2062376T3 (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US9993434B2 (en)	2003-07-31	2018-06-12	Delavau L.L.C.	Calcium carbonate granulation

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5464632C1 (en) *	1991-07-22	2001-02-20	Prographarm Lab	Rapidly disintegratable multiparticular tablet
FR2679451B1 (fr) *	1991-07-22	1994-09-09	Prographarm Laboratoires	Comprime multiparticulaire a delitement rapide.
ES2059260B1 (es) *	1992-10-06	1995-04-16	Espanola Prod Quimicos	Procedimiento de preparacion de comprimidos conteniendo diclofenaco; dispersables en agua.
FR2766089B1 (fr) *	1997-07-21	2000-06-02	Prographarm Lab	Comprime multiparticulaire perfectionne a delitement rapide
FR2784895B1 (fr) *	1998-10-23	2004-12-17	Gattefosse Ets Sa	Comprime a croquer a gout masque et liberation immediate du principe actif et procede de fabrication
UA75569C2 (en) *	1998-12-01	2006-05-15	Reddys Lab Ltd Dr	Pharmaceutical composition of thiadiazolidinedione and method for its manufacture
CA2363053C (fr) *	2001-11-09	2011-01-25	Bernard Charles Sherman	Formulation pour pastilles de bisulfate de clopidogrel
KR20010114199A (ko) *	2001-12-11	2001-12-29	유형선	제약산업에서 사용될 수 있는 고형제제를 위한 직타용부형제의 새로운 의약품 조성물
US20050095287A1 (en) *	2003-10-29	2005-05-05	Matharu Amol S.	Fosinopril composition
EP3165220B2 (fr) *	2004-12-03	2024-11-13	Merck Sharp & Dohme LLC	Composition pharmaceutique contenant un agent d'anti-nucléation
GR1006875B (el) *	2005-06-30	2010-07-12	"Φαρματεν" Φαρμακευτικη Βιομηχανικη Εμπορικη Α.Ε.,	Βελτιωμενες φαρμακευτικες συνθεσεις περιεχουσες αναστολεις του μετατρεπτικου ενζυμου αγγειοτενσινης και μεθοδοι παρασκευης αυτων.
US9138414B1 (en)	2006-09-15	2015-09-22	Delavau Llc	Calcium supplement having enhanced absorption
SI23149A (sl)	2009-09-21	2011-03-31	Silverstone Pharma	Nove benzatinske soli ACE inhibitorjev, postopek za njihovo pripravo in njihova uporaba za zdravljenje kardiovaskularnih bolezni
US10076494B2 (en)	2016-06-16	2018-09-18	Dexcel Pharma Technologies Ltd.	Stable orally disintegrating pharmaceutical compositions

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4217347A (en) *	1977-12-27	1980-08-12	E. R. Squibb & Sons, Inc.	Method of treating hypertension and medicaments therefor
US4384123A (en) *	1980-12-04	1983-05-17	E. R. Squibb & Sons, Inc.	Phosphinylalkanoyl substituted prolines
US4793998A (en) *	1986-10-20	1988-12-27	Warner-Lambert Company	Stabilized drug compositions
AU612137B2 (en) *	1987-04-27	1991-07-04	E.R. Squibb & Sons, Inc.	Method for inhibiting loss of cognitive functions employing an ace inhibitor

1990
- 1990-06-19 CA CA002019324A patent/CA2019324C/fr not_active Expired - Lifetime
- 1990-07-09 ES ES90307449T patent/ES2062376T3/es not_active Expired - Lifetime
- 1990-07-09 AT AT90307449T patent/ATE100321T1/de not_active IP Right Cessation
- 1990-07-09 EP EP90307449A patent/EP0408273B1/fr not_active Expired - Lifetime
- 1990-07-09 DE DE69006125T patent/DE69006125T2/de not_active Expired - Lifetime
- 1990-07-09 DK DK90307449.0T patent/DK0408273T3/da active
- 1990-07-10 JP JP2185179A patent/JP2965633B2/ja not_active Expired - Lifetime
- 1990-10-01 DD DD90344330A patent/DD299154A5/de not_active IP Right Cessation

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US9993434B2 (en)	2003-07-31	2018-06-12	Delavau L.L.C.	Calcium carbonate granulation

Also Published As

Publication number	Publication date
ATE100321T1 (de)	1994-02-15
EP0408273B1 (fr)	1994-01-19
ES2062376T3 (es)	1994-12-16
DK0408273T3 (da)	1994-02-28
EP0408273A1 (fr)	1991-01-16
JP2965633B2 (ja)	1999-10-18
CA2019324C (fr)	1996-08-20
DE69006125D1 (de)	1994-03-03
DE69006125T2 (de)	1994-05-19
JPH0348623A (ja)	1991-03-01
DD299154A5 (de)	1992-04-02

Legal Events

Date	Code	Title	Description
1994-01-21	EEER	Examination request
2010-06-19	MKEX	Expiry
2023-05-26	MKEX	Expiry	Effective date: 20100619

Publication	Publication Date	Title
DE69006125D1 (de)	1994-03-03	Fosinopril enthaltende Tablettenformulierungen.
AU551177B2 (en)	1986-04-17	A device for raising and lowering objects, such as bed frameswork tables or the like
AU1143892A (en)	1992-05-14	(4.3.3.0)propellane-8,11-diamine compounds
AU2701184A (en)	1984-10-25	Divisible polyacrylate based tablet
AU5431390A (en)	1990-11-16	Novel arylpyridazines, their manufacture, use and medicaments containing them
AU7702291A (en)	1991-11-28	Dietary fiber, its process and physiologically active composition containing the same as an active ingredient
AU2378988A (en)	1989-04-20	4-(N-3-pyridylmethyl)-amino-1,2,4-triazinones
AU1056795A (en)	1995-06-06	Removable, washable sweatband for hats
DE3779053D1 (fr)	1992-06-17
GR3007385T3 (fr)	1993-07-30
FI874188A7 (fi)	1988-03-26	Blankett bestaoende av flera delar, som loesgoerbart haolles pao plats av tillfaellig ytbindning i talongomraodet.
IE930197L (en)	1987-12-11	Anti-Inflammatory Compositions
AU5494490A (en)	1990-11-22	3,4-dehydropiperidine derivatives having psychotropic activity
EP0427124A3 (en)	1991-09-18	Antacid tablets
AU7547787A (en)	1988-01-12	Dibenz(b,e)oxepin derivative and pharmaceutical containing the same as active ingredient
GR3015016T3 (en)	1995-05-31	Ultra-wideband achromatic lens.
AU567940B2 (en)	1987-12-10	Controlled release tablet
AU1097988A (en)	1988-08-04	Alkylmelatonins
CA2001782A1 (fr)	1990-05-10	3-(3-propan-2-ylphenyl)butanal et 3-(3-propen-2-ylphenyl)butanal et leur utilisation comme agents odorisants.
AU4719489A (en)	1990-07-12	Controlled-release, low dose aspirin
ES2185666T3 (es)	2003-05-01	Formulacion estabilizada para comprimidos.
NO874241D0 (no)	1987-10-09	Terapeutisk aktive salter.
BG102638A (bg)	1999-07-30	Таблети с високо съдържание на фамцикловир
CA2330904A1 (fr)	2002-07-11	Formulation pour pastilles de fosinopril sodium
EP0948961A3 (fr)	2001-04-04	Comprimé effervescent comprenant du calcium avec un antihistaminique comme principe actif

CA2019324A1 - Comprimes de fosinopril - Google Patents

Info

Links

Classifications

Landscapes

Applications Claiming Priority (2)

Publications (2)

Family

ID=23490122

Family Applications (1)

Country Status (8)

Cited By (1)

Families Citing this family (14)

Family Cites Families (4)

Cited By (1)

Also Published As

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Legal Events