CA2271788A1 - Analogues de peptide yy et leurs utilisations - Google Patents
Analogues de peptide yy et leurs utilisations Download PDFInfo
- Publication number
- CA2271788A1 CA2271788A1 CA002271788A CA2271788A CA2271788A1 CA 2271788 A1 CA2271788 A1 CA 2271788A1 CA 002271788 A CA002271788 A CA 002271788A CA 2271788 A CA2271788 A CA 2271788A CA 2271788 A1 CA2271788 A1 CA 2271788A1
- Authority
- CA
- Canada
- Prior art keywords
- arg
- leu
- seq
- pyy
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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- LRBQNJMCXXYXIU-NRMVVENXSA-N tannic acid Chemical compound OC1=C(O)C(O)=CC(C(=O)OC=2C(=C(O)C=C(C=2)C(=O)OC[C@@H]2[C@H]([C@H](OC(=O)C=3C=C(OC(=O)C=4C=C(O)C(O)=C(O)C=4)C(O)=C(O)C=3)[C@@H](OC(=O)C=3C=C(OC(=O)C=4C=C(O)C(O)=C(O)C=4)C(O)=C(O)C=3)[C@@H](OC(=O)C=3C=C(OC(=O)C=4C=C(O)C(O)=C(O)C=4)C(O)=C(O)C=3)O2)OC(=O)C=2C=C(OC(=O)C=3C=C(O)C(O)=C(O)C=3)C(O)=C(O)C=2)O)=C1 LRBQNJMCXXYXIU-NRMVVENXSA-N 0.000 description 1
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Endocrinology (AREA)
- Toxicology (AREA)
- Zoology (AREA)
- Gastroenterology & Hepatology (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Abstract
L'invention concerne des analogues de PYY ainsi que des compositions et des procédés utiles pour réguler les activités biologiques telles que la prolifération cellulaire, le transport d'éléments nutritifs, la lipolyse et la sécrétion intestinale d'eau et d'électrolyte.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/US1996/018374 WO1998020885A1 (fr) | 1996-11-13 | 1996-11-13 | Analogues de peptide yy et leurs utilisations |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2271788A1 true CA2271788A1 (fr) | 1998-05-22 |
Family
ID=22256144
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002271788A Abandoned CA2271788A1 (fr) | 1996-11-13 | 1996-11-13 | Analogues de peptide yy et leurs utilisations |
Country Status (5)
| Country | Link |
|---|---|
| EP (1) | EP1015007A1 (fr) |
| JP (1) | JP2000505105A (fr) |
| AU (1) | AU1159897A (fr) |
| CA (1) | CA2271788A1 (fr) |
| WO (1) | WO1998020885A1 (fr) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7048906B2 (en) | 1995-05-17 | 2006-05-23 | Cedars-Sinai Medical Center | Methods of diagnosing and treating small intestinal bacterial overgrowth (SIBO) and SIBO-related conditions |
| ES2353728T3 (es) * | 1999-02-10 | 2011-03-04 | Curis, Inc. | Péptido yy (pyy) para tratar trastornos metabólicos de la glucosa. |
| US7601691B2 (en) | 1999-05-17 | 2009-10-13 | Conjuchem Biotechnologies Inc. | Anti-obesity agents |
| PL205971B1 (pl) | 2001-09-24 | 2010-06-30 | Imp Innovations Ltd | Zastosowanie PYY₃-₃₆ do wytwarzania leku na ograniczanie apetytu, zmniejszenie otyłości lub do zapobiegania otyłości |
| CA2510199A1 (fr) | 2002-12-17 | 2004-07-08 | Nastech Pharmaceutical Company Inc. | Compositions et procedes permettant d'ameliorer l'administration aux muqueuses de peptides de liaison du recepteur y2, et procedes pour le traitement et la prevention de l'obesite |
| US7229966B2 (en) | 2002-12-17 | 2007-06-12 | Nastech Pharmaceutical Company Inc. | Compositions and methods for enhanced mucosal delivery of Y2 receptor-binding peptides and methods for treating and preventing obesity |
| US7166575B2 (en) | 2002-12-17 | 2007-01-23 | Nastech Pharmaceutical Company Inc. | Compositions and methods for enhanced mucosal delivery of peptide YY and methods for treating and preventing obesity |
| EP1583549A4 (fr) * | 2003-01-17 | 2006-10-04 | Sod Conseils Rech Applic | Analogues du peptide yy |
| JP5638177B2 (ja) | 2004-02-11 | 2014-12-10 | アミリン・ファーマシューティカルズ, リミテッド・ライアビリティ・カンパニーAmylin Pharmaceuticals, Llc | 膵臓ポリペプチドファミリーモチーフおよびそのモチーフを含むポリペプチド |
| WO2005112633A2 (fr) | 2004-05-14 | 2005-12-01 | Emisphere Technologies, Inc. | Composes et compositions pour administration d’agents actifs |
| CA2566161C (fr) | 2004-05-14 | 2013-10-01 | Emisphere Technologies, Inc. | Composes d'aryle cetone et compositions pour la delivrance d'agents actifs |
| EP3000826A1 (fr) | 2004-12-13 | 2016-03-30 | Amylin Pharmaceuticals, LLC | Motifs de famille de polypeptides pancreatiques, polypeptides et leurs methodes |
| CN101296942A (zh) | 2005-08-11 | 2008-10-29 | 安米林药品公司 | 具有可选择特性的杂合多肽 |
| TWI428346B (zh) | 2006-12-13 | 2014-03-01 | Imp Innovations Ltd | 新穎化合物及其等對進食行為影響 |
| PL2651398T3 (pl) | 2010-12-16 | 2018-05-30 | Novo Nordisk A/S | Stałe kompozycje zawierające agonistę GLP-1 i sól kwasu N-(8-(2-hydroksybenzoilo)amino)kaprylowego |
| EP4324475A1 (fr) | 2012-03-22 | 2024-02-21 | Novo Nordisk A/S | Compositions de peptides glp-1 et leur préparation |
| KR20210086717A (ko) | 2013-05-02 | 2021-07-08 | 노보 노르디스크 에이/에스 | Glp-1 화합물의 경구 투여 |
| US10246497B2 (en) | 2013-11-15 | 2019-04-02 | Novo Nordisk A/S | Selective PYY compounds and uses thereof |
| JP6629198B2 (ja) | 2013-11-15 | 2020-01-15 | ノヴォ ノルディスク アー／エス | ３５位にβ−ホモアルギニン置換を有するＨＰＹＹ（１−３６） |
| CA2988500A1 (fr) | 2015-06-12 | 2016-12-15 | Novo Nordisk A/S | Composes pyy selectifs et leurs utilisations |
| WO2019149880A1 (fr) | 2018-02-02 | 2019-08-08 | Novo Nordisk A/S | Compositions solides comprenant un agoniste de glp -1 et un sel d'acide n- (8- (2-hydroxybenzoyl) amino) caprylique |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5328899A (en) * | 1988-07-15 | 1994-07-12 | The Salk Institute For Biological Studies | NPY peptide analogs |
| US5026685A (en) * | 1988-07-15 | 1991-06-25 | The Salk Institute For Biological Studies | NPY peptide analogs |
-
1996
- 1996-11-13 WO PCT/US1996/018374 patent/WO1998020885A1/fr not_active Ceased
- 1996-11-13 AU AU11598/97A patent/AU1159897A/en not_active Abandoned
- 1996-11-13 JP JP10522501A patent/JP2000505105A/ja active Pending
- 1996-11-13 EP EP96942759A patent/EP1015007A1/fr not_active Withdrawn
- 1996-11-13 CA CA002271788A patent/CA2271788A1/fr not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| EP1015007A1 (fr) | 2000-07-05 |
| WO1998020885A1 (fr) | 1998-05-22 |
| JP2000505105A (ja) | 2000-04-25 |
| AU1159897A (en) | 1998-06-03 |
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Legal Events
| Date | Code | Title | Description |
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| FZDE | Dead |