CA2605796A1 - Compositions pharmaceutiques et methodes comprenant une combinaison d'un modulateur selectif du recepteur de l'oestrogene et d'un inhibiteur de l'aromatase - Google Patents
Compositions pharmaceutiques et methodes comprenant une combinaison d'un modulateur selectif du recepteur de l'oestrogene et d'un inhibiteur de l'aromatase Download PDFInfo
- Publication number
- CA2605796A1 CA2605796A1 CA002605796A CA2605796A CA2605796A1 CA 2605796 A1 CA2605796 A1 CA 2605796A1 CA 002605796 A CA002605796 A CA 002605796A CA 2605796 A CA2605796 A CA 2605796A CA 2605796 A1 CA2605796 A1 CA 2605796A1
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- CA
- Canada
- Prior art keywords
- phenyl
- pharmaceutically acceptable
- pyrrolidin
- cis
- ethoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
- A61K31/5685—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone having an oxo group in position 17, e.g. androsterone
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
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- A—HUMAN NECESSITIES
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Landscapes
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- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
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- Neurosurgery (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US67480705P | 2005-04-25 | 2005-04-25 | |
| US60/674,807 | 2005-04-25 | ||
| PCT/IB2006/001040 WO2006114702A2 (fr) | 2005-04-25 | 2006-04-13 | Compositions pharmaceutiques et methodes comprenant une combinaison d'un modulateur selectif du recepteur de l'oestrogene et d'un inhibiteur de l'aromatase |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2605796A1 true CA2605796A1 (fr) | 2006-11-02 |
Family
ID=36693972
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002605796A Abandoned CA2605796A1 (fr) | 2005-04-25 | 2006-04-13 | Compositions pharmaceutiques et methodes comprenant une combinaison d'un modulateur selectif du recepteur de l'oestrogene et d'un inhibiteur de l'aromatase |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP1937251A2 (fr) |
| JP (1) | JP2006306872A (fr) |
| AR (1) | AR054258A1 (fr) |
| CA (1) | CA2605796A1 (fr) |
| TW (1) | TW200716094A (fr) |
| WO (1) | WO2006114702A2 (fr) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI0711525A2 (pt) | 2006-06-02 | 2011-11-01 | Pear Tree Women S Health Care | composição farmacêutica e método para tratar sintomas de vaginite atrófica |
| EP2070943A1 (fr) * | 2007-12-14 | 2009-06-17 | Crystal Pharma, S.A. | Procédé de préparation des 6-Alkylidenandrost-1,4-dien-3-ones |
| JP5777163B2 (ja) * | 2009-07-03 | 2015-09-09 | 国立研究開発法人理化学研究所 | Ｐｅｔ用標識化合物 |
| PT2753312T (pt) * | 2011-09-08 | 2017-02-03 | Mereo Biopharma 2 Ltd | Utilização de um inibidor da aromatase para o tratamento de hipogonadismo e doenças relacionadas |
| JP7131773B2 (ja) * | 2016-04-29 | 2022-09-06 | ボード オブ リージェンツ，ザ ユニバーシティ オブ テキサス システム | ホルモン受容体に関連する転写活性の標的尺度 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5552412A (en) * | 1995-01-09 | 1996-09-03 | Pfizer Inc | 5-substitued-6-cyclic-5,6,7,8-tetrahydronaphthalen2-ol compounds which are useful for treating osteoporosis |
| AR034142A1 (es) * | 2000-09-08 | 2004-02-04 | Sloan Kettering Inst Cancer | Una composicion farmaceutica, metodo para fabricar un medicamento en base a dicha composicion y uso de la composicion |
| NZ524104A (en) * | 2000-09-08 | 2004-12-24 | Pharmacia Italia S | Exemestane as chemopreventing agent |
| WO2003017973A1 (fr) * | 2001-08-31 | 2003-03-06 | Pantarhei Bioscience B.V. | Traitement de troubles gynecologiques benins et vecteur d'administration a cet effet |
| EP1435967A2 (fr) * | 2001-10-10 | 2004-07-14 | Pharmacia Italia S.p.A. | Procedes de prevention et de traitement de la deperdition osseuse avec des composes steroides |
| WO2005070434A2 (fr) * | 2004-01-13 | 2005-08-04 | Wyeth | Traitement de l'osteoporose liee a la therapie par un inhibiteur de l'aromatase |
| WO2006048749A1 (fr) * | 2004-11-04 | 2006-05-11 | Pfizer Products Inc. | Anticorps ctla-4 et inhibiteur de l'aromatase ou traitement combine du cancer du sein |
-
2006
- 2006-04-13 EP EP06744583A patent/EP1937251A2/fr not_active Withdrawn
- 2006-04-13 WO PCT/IB2006/001040 patent/WO2006114702A2/fr not_active Ceased
- 2006-04-13 CA CA002605796A patent/CA2605796A1/fr not_active Abandoned
- 2006-04-24 JP JP2006118713A patent/JP2006306872A/ja active Pending
- 2006-04-24 AR AR20060101616A patent/AR054258A1/es not_active Application Discontinuation
- 2006-04-24 TW TW095114529A patent/TW200716094A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2006114702A2 (fr) | 2006-11-02 |
| TW200716094A (en) | 2007-05-01 |
| JP2006306872A (ja) | 2006-11-09 |
| EP1937251A2 (fr) | 2008-07-02 |
| WO2006114702A3 (fr) | 2007-01-04 |
| AR054258A1 (es) | 2007-06-13 |
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