CH631180A5 - Procedimento per la preparazione delle 5,6-deidropenicilline. - Google Patents

Procedimento per la preparazione delle 5,6-deidropenicilline. Download PDF

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Publication number
CH631180A5
CH631180A5 CH221077A CH221077A CH631180A5 CH 631180 A5 CH631180 A5 CH 631180A5 CH 221077 A CH221077 A CH 221077A CH 221077 A CH221077 A CH 221077A CH 631180 A5 CH631180 A5 CH 631180A5
Authority
CH
Switzerland
Prior art keywords
product
preparation
phenyl
cooch
xii
Prior art date
Application number
CH221077A
Other languages
English (en)
Italian (it)
Inventor
Luciano Re
Alberto Brandt
Luciano Bassignani
Original Assignee
Anic Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Anic Spa filed Critical Anic Spa
Publication of CH631180A5 publication Critical patent/CH631180A5/de

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/09Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4
    • C07D205/095Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4 and with a nitrogen atom directly attached in position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/10Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having two double bonds between ring members or between ring members and non-ring members

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Polyesters Or Polycarbonates (AREA)
  • Polyamides (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
CH221077A 1976-02-23 1977-02-22 Procedimento per la preparazione delle 5,6-deidropenicilline. CH631180A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT20457/76A IT1058858B (it) 1976-02-23 1976-02-23 5.6 deidropenicilline processo per la loro preparazione e intermdi ottenibili in detto processo

Publications (1)

Publication Number Publication Date
CH631180A5 true CH631180A5 (de) 1982-07-30

Family

ID=11167232

Family Applications (1)

Application Number Title Priority Date Filing Date
CH221077A CH631180A5 (de) 1976-02-23 1977-02-22 Procedimento per la preparazione delle 5,6-deidropenicilline.

Country Status (21)

Country Link
US (3) US4133807A (de)
JP (1) JPS52102267A (de)
AU (1) AU514741B2 (de)
BE (1) BE851751A (de)
CA (1) CA1090290A (de)
CH (1) CH631180A5 (de)
CS (1) CS199662B2 (de)
DD (1) DD128359A5 (de)
DE (1) DE2707404C3 (de)
DK (2) DK77177A (de)
FR (1) FR2341582A1 (de)
GB (2) GB1572140A (de)
HU (2) HU179786B (de)
IT (1) IT1058858B (de)
LU (1) LU76816A1 (de)
NL (1) NL171159C (de)
NO (2) NO770568L (de)
SE (1) SE438506B (de)
SU (3) SU683626A3 (de)
YU (3) YU49377A (de)
ZA (1) ZA77890B (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1058858B (it) * 1976-02-23 1982-05-10 Snam Progetti 5.6 deidropenicilline processo per la loro preparazione e intermdi ottenibili in detto processo
JPS5398951A (en) * 1977-02-08 1978-08-29 Shionogi & Co Ltd Azetidinone derivatives and process for their preparation

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4174318A (en) * 1970-11-03 1979-11-13 Glaxo Laboratories Ltd. Alkylative cleavage of azetidinone disulfides
GB1368234A (en) 1970-11-03 1974-09-25 Glaxo Lab Ltd Thiosubstituted szetidinones and other antibiotic precursors
BE791161A (fr) * 1972-01-03 1973-05-09 Beecham Group Ltd Procede pour la preparation d'analogues des cephalosporines
BE791159A (fr) 1972-01-03 1973-05-09 Beecham Group Ltd Procede pour la preparation de cephemes
DE2204105A1 (de) 1972-01-28 1973-08-02 Beecham Group Ltd Seco-penicilline und verfahren zu ihrer herstellung
US4089963A (en) * 1972-03-13 1978-05-16 Astra Pharmaceutical Products, Inc. Esters of amidinopenicillanic acids, pharmaceutical preparations and method for treating infectious diseases
US4219462A (en) * 1974-07-29 1980-08-26 Merck & Co., Inc. 6-Methyl penicillins
IT1058858B (it) * 1976-02-23 1982-05-10 Snam Progetti 5.6 deidropenicilline processo per la loro preparazione e intermdi ottenibili in detto processo
US4136096A (en) * 1977-02-25 1979-01-23 Pfizer Inc. 6-amino-2,2-dimethyl-3-(5-tetrazolyl)penam process and intermediates therefor
US4168314A (en) * 1977-11-17 1979-09-18 Merck & Co., Inc. 6-(1'-Hydroxyethyl)-2-aminoethylthio-pen-2-em-3-carboxylic acid
US4160091A (en) * 1977-11-21 1979-07-03 Eli Lilly And Company Process for preparation of 3-halo-3-methylcephams

Also Published As

Publication number Publication date
YU214982A (en) 1983-01-21
AU2242877A (en) 1978-08-24
LU76816A1 (de) 1977-07-06
ZA77890B (en) 1977-12-28
NL7701962A (nl) 1977-08-25
FR2341582B1 (de) 1980-01-11
NL171159C (nl) 1983-02-16
SE7701907L (sv) 1977-10-03
DE2707404A1 (de) 1977-08-25
NO773766L (no) 1977-08-24
US4353825A (en) 1982-10-12
CA1090290A (en) 1980-11-25
YU214882A (en) 1983-01-21
NO770568L (no) 1977-08-24
US4133807A (en) 1979-01-09
CS199662B2 (en) 1980-07-31
DK558781A (da) 1981-12-16
SU721004A3 (ru) 1980-03-05
HU183632B (en) 1984-05-28
GB1572139A (en) 1980-07-23
DD128359A5 (de) 1977-11-16
SE438506B (sv) 1985-04-22
BE851751A (fr) 1977-08-23
YU49377A (en) 1983-01-21
DK77177A (da) 1977-08-24
JPS52102267A (en) 1977-08-27
DE2707404C3 (de) 1979-03-22
US4288366A (en) 1981-09-08
NL171159B (nl) 1982-09-16
SU712024A3 (ru) 1980-01-25
AU514741B2 (en) 1981-02-26
HU179786B (en) 1982-12-28
DE2707404B2 (de) 1978-07-13
GB1572140A (en) 1980-07-23
IT1058858B (it) 1982-05-10
FR2341582A1 (fr) 1977-09-16
SU683626A3 (ru) 1979-08-30

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