CL2004000856A1 - Compuestos derivados 8b-vonil-11b-(alfa-sustituidos)alquil-estra-1,3,5(10)-trienos; composiciones farmaceuticas; compuestos intermediarios; uso para la anticoncepcion, para el tratamiento de carcinomas de ovario y tumores de celulas granulosas. - Google Patents

Compuestos derivados 8b-vonil-11b-(alfa-sustituidos)alquil-estra-1,3,5(10)-trienos; composiciones farmaceuticas; compuestos intermediarios; uso para la anticoncepcion, para el tratamiento de carcinomas de ovario y tumores de celulas granulosas.

Info

Publication number
CL2004000856A1
CL2004000856A1 CL200400856A CL2004000856A CL2004000856A1 CL 2004000856 A1 CL2004000856 A1 CL 2004000856A1 CL 200400856 A CL200400856 A CL 200400856A CL 2004000856 A CL2004000856 A CL 2004000856A CL 2004000856 A1 CL2004000856 A1 CL 2004000856A1
Authority
CL
Chile
Prior art keywords
compounds
vonil
trienos
alquil
estra
Prior art date
Application number
CL200400856A
Other languages
English (en)
Inventor
Brauer Olaf Peters Alexan Nico
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of CL2004000856A1 publication Critical patent/CL2004000856A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/16—Masculine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J75/00—Processes for the preparation of steroids in general

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Diabetes (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
CL200400856A 2003-04-22 2004-04-22 Compuestos derivados 8b-vonil-11b-(alfa-sustituidos)alquil-estra-1,3,5(10)-trienos; composiciones farmaceuticas; compuestos intermediarios; uso para la anticoncepcion, para el tratamiento de carcinomas de ovario y tumores de celulas granulosas. CL2004000856A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10318896A DE10318896A1 (de) 2003-04-22 2003-04-22 8beta-Vinyl-11beta-(omega-substituierte)alkyl-estra-1,3,5(10)-triene

Publications (1)

Publication Number Publication Date
CL2004000856A1 true CL2004000856A1 (es) 2005-03-28

Family

ID=33304956

Family Applications (1)

Application Number Title Priority Date Filing Date
CL200400856A CL2004000856A1 (es) 2003-04-22 2004-04-22 Compuestos derivados 8b-vonil-11b-(alfa-sustituidos)alquil-estra-1,3,5(10)-trienos; composiciones farmaceuticas; compuestos intermediarios; uso para la anticoncepcion, para el tratamiento de carcinomas de ovario y tumores de celulas granulosas.

Country Status (21)

Country Link
US (1) US7375098B2 (es)
EP (1) EP1622924A2 (es)
JP (1) JP2006524202A (es)
KR (1) KR20060005386A (es)
CN (1) CN100381457C (es)
AR (1) AR044056A1 (es)
AU (1) AU2004232462A1 (es)
BR (1) BRPI0409794A (es)
CA (1) CA2522354A1 (es)
CL (1) CL2004000856A1 (es)
CR (1) CR8053A (es)
DE (1) DE10318896A1 (es)
EA (1) EA009606B1 (es)
EC (1) ECSP056180A (es)
MX (1) MXPA05011386A (es)
NO (1) NO20055493L (es)
PE (1) PE20050423A1 (es)
RS (1) RS20050793A (es)
UY (1) UY28284A1 (es)
WO (1) WO2004094451A2 (es)
ZA (1) ZA200509447B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001077139A1 (de) * 2000-04-12 2001-10-18 Schering Aktiengesellschaft 8.beta.-hydrocarbyl-substituierte estratriene als selektiv wirksame estrogene
JP2008512458A (ja) 2004-09-07 2008-04-24 ワイス ６Ｈ−［１］ベンゾピラノ［４，３−ｂ］キノリン及びエストロゲン様物質としてのそれらの使用
US20070144968A1 (en) * 2005-10-05 2007-06-28 Cristian Fazioni Separation of fulvestrant isomers

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1226155E (pt) * 1999-11-02 2007-07-26 Bayer Schering Pharma Ag 18-nor-esteróides como estrogénios selectivamente activos
WO2001077139A1 (de) * 2000-04-12 2001-10-18 Schering Aktiengesellschaft 8.beta.-hydrocarbyl-substituierte estratriene als selektiv wirksame estrogene
DE10151114A1 (de) * 2001-10-15 2003-04-17 Schering Ag 8ß-Substituierte-11ß-aryl-estra-2,3,5(10)-trienderivate

Also Published As

Publication number Publication date
UY28284A1 (es) 2004-11-30
CR8053A (es) 2006-05-29
NO20055493D0 (no) 2005-11-21
ZA200509447B (en) 2009-08-26
BRPI0409794A (pt) 2006-05-30
WO2004094451A2 (de) 2004-11-04
WO2004094451A3 (de) 2004-12-23
RS20050793A (sr) 2008-04-04
AU2004232462A1 (en) 2004-11-04
US7375098B2 (en) 2008-05-20
KR20060005386A (ko) 2006-01-17
CN1777618A (zh) 2006-05-24
US20050065135A1 (en) 2005-03-24
ECSP056180A (es) 2006-04-19
NO20055493L (no) 2006-01-18
EP1622924A2 (de) 2006-02-08
EA200501568A1 (ru) 2006-06-30
PE20050423A1 (es) 2005-08-13
DE10318896A1 (de) 2004-11-25
AR044056A1 (es) 2005-08-24
CA2522354A1 (en) 2004-11-04
CN100381457C (zh) 2008-04-16
MXPA05011386A (es) 2006-04-18
EA009606B1 (ru) 2008-02-28
JP2006524202A (ja) 2006-10-26

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