CL2015002706A1 - Inhibidores tripeptídicos de la epoxicetona proteasa. - Google Patents

Inhibidores tripeptídicos de la epoxicetona proteasa.

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Publication number
CL2015002706A1
CL2015002706A1 CL2015002706A CL2015002706A CL2015002706A1 CL 2015002706 A1 CL2015002706 A1 CL 2015002706A1 CL 2015002706 A CL2015002706 A CL 2015002706A CL 2015002706 A CL2015002706 A CL 2015002706A CL 2015002706 A1 CL2015002706 A1 CL 2015002706A1
Authority
CL
Chile
Prior art keywords
epoxy ketone
ketone protease
tripeptide inhibitors
tripeptide
inhibitors
Prior art date
Application number
CL2015002706A
Other languages
English (en)
Inventor
Dustin Mcminn
Henry Johnson
Simeon Bowers
David C Moebius
Original Assignee
Onyx Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=51581125&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2015002706(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Onyx Therapeutics Inc filed Critical Onyx Therapeutics Inc
Publication of CL2015002706A1 publication Critical patent/CL2015002706A1/es

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    • C07K5/08Tripeptides
    • C07K5/0821Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
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Abstract

COMPUESTOS TRIPEPTIDICOS INHIBIDORES DE LA EPOXICETONA PROTEASA; COMPOSICION FARMACEUTICA QUE LOS COMPRENDE; METODO DE INHIBICION DE INMUNOPROTEASA DE UNA CELULA, UTIL PARA EL TRATAMIENTO DE UN ENFERMEDAD INMUNORRELACIONADA TAL COMO ARTRITIS REUMATOIDE, LUPUS, ENFERMEDAD INFLAMATORIA DEL INTESTINO, ENTRE OTRAS.
CL2015002706A 2013-03-14 2015-09-14 Inhibidores tripeptídicos de la epoxicetona proteasa. CL2015002706A1 (es)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
US201361786086P 2013-03-14 2013-03-14
US201361785608P 2013-03-14 2013-03-14
US201361847780P 2013-07-18 2013-07-18
US201361856847P 2013-07-22 2013-07-22
US201361883843P 2013-09-27 2013-09-27
US201361883798P 2013-09-27 2013-09-27
US201461941798P 2014-02-19 2014-02-19
ARP140100970A AR095426A1 (es) 2013-03-14 2014-03-13 Inhibidores tripeptídicos de la epoxicetona proteasa

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US10947224B2 (en) 2014-03-13 2021-03-16 Indiana University Research And Technology Corporation Hepatitis B core protein allosteric modulators
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US10987360B2 (en) 2016-09-15 2021-04-27 Assembly Biosciences, Inc. Hepatitis B core protein modulators
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