CN1030388C - 1,5-苯并硫杂吖庚因衍生物的制造方法 - Google Patents

1,5-苯并硫杂吖庚因衍生物的制造方法 Download PDF

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Publication number
CN1030388C
CN1030388C CN87100139A CN87100139A CN1030388C CN 1030388 C CN1030388 C CN 1030388C CN 87100139 A CN87100139 A CN 87100139A CN 87100139 A CN87100139 A CN 87100139A CN 1030388 C CN1030388 C CN 1030388C
Authority
CN
China
Prior art keywords
cis
methanol
ethyl
benzothiazepine
chloro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
CN87100139A
Other languages
English (en)
Chinese (zh)
Other versions
CN87100139A (zh
Inventor
井上博纯
大塚久男
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Tanabe Pharma Corp
Original Assignee
Tanabe Seiyaku Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tanabe Seiyaku Co Ltd filed Critical Tanabe Seiyaku Co Ltd
Publication of CN87100139A publication Critical patent/CN87100139A/zh
Application granted granted Critical
Publication of CN1030388C publication Critical patent/CN1030388C/zh
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CN87100139A 1986-01-07 1987-01-07 1,5-苯并硫杂吖庚因衍生物的制造方法 Expired - Fee Related CN1030388C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP61001845A JPS62161776A (ja) 1986-01-07 1986-01-07 １，５−ベンゾチアゼピン誘導体の製法
JP1845/86 1986-01-07

Publications (2)

Publication Number Publication Date
CN87100139A CN87100139A (zh) 1987-08-12
CN1030388C true CN1030388C (zh) 1995-11-29

Family

ID=11512884

Family Applications (1)

Application Number Title Priority Date Filing Date
CN87100139A Expired - Fee Related CN1030388C (zh) 1986-01-07 1987-01-07 1,5-苯并硫杂吖庚因衍生物的制造方法

Country Status (14)

Country Link
JP (1) JPS62161776A (fr)
KR (1) KR910002879B1 (fr)
CN (1) CN1030388C (fr)
AT (1) AT394367B (fr)
BG (1) BG46747A3 (fr)
CA (1) CA1291134C (fr)
DD (1) DD257426A5 (fr)
ES (1) ES2003642A6 (fr)
FI (1) FI865343L (fr)
HU (1) HU198031B (fr)
IE (1) IE59359B1 (fr)
IL (1) IL81039A (fr)
PT (1) PT84036B (fr)
SU (1) SU1544187A3 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5580867A (en) * 1994-09-09 1996-12-03 Universite De Montreal Myocardial protection during ischemia and reperfusion

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57169476A (en) * 1981-04-13 1982-10-19 Hamari Yakuhin Kogyo Kk Novel preparation of benzothiazepine derivative
JPS57175182A (en) * 1981-04-22 1982-10-28 Hamari Yakuhin Kogyo Kk Novel preparation of benzothiazepin derivative
JPS58113186A (ja) * 1981-12-28 1983-07-05 Hamari Yakuhin Kogyo Kk ベンゾチアゼピン誘導体の新規な製造法
JPS58116476A (ja) * 1981-12-29 1983-07-11 Hamari Yakuhin Kogyo Kk ベンゾチアゼピン誘導体の新規製造法
US4567175A (en) * 1983-06-03 1986-01-28 Tanabe Seiyaku Co., Ltd. 8-Chloro-1,5-benzothiazepine derivatives
US4585768A (en) * 1984-04-10 1986-04-29 Tanabe Seiyaku Co., Ltd. 1,5-benzothiazepine derivatives and processes for preparing the same

Also Published As

Publication number Publication date
ATA1687A (de) 1991-09-15
IE59359B1 (en) 1994-02-09
ES2003642A6 (es) 1988-11-01
HUT45242A (en) 1988-06-28
DD257426A5 (de) 1988-06-15
IL81039A0 (en) 1987-03-31
CN87100139A (zh) 1987-08-12
AT394367B (de) 1992-03-25
IE863269L (en) 1987-07-07
FI865343A0 (fi) 1986-12-30
KR910002879B1 (ko) 1991-05-09
PT84036B (pt) 1989-01-17
CA1291134C (fr) 1991-10-22
FI865343A7 (fi) 1987-07-08
KR870007147A (ko) 1987-08-17
PT84036A (en) 1987-01-01
JPS62161776A (ja) 1987-07-17
SU1544187A3 (ru) 1990-02-15
IL81039A (en) 1991-07-18
FI865343L (fi) 1987-07-08
HU198031B (en) 1989-07-28
JPH0573749B2 (fr) 1993-10-15
BG46747A3 (bg) 1990-02-15

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C19 Lapse of patent right due to non-payment of the annual fee
CF01 Termination of patent right due to non-payment of annual fee