CR11123A - Compuestos triciclicos que contienen nitrogeno como agentes antibacteriales - Google Patents

Compuestos triciclicos que contienen nitrogeno como agentes antibacteriales

Info

Publication number
CR11123A
CR11123A CR11123A CR11123A CR11123A CR 11123 A CR11123 A CR 11123A CR 11123 A CR11123 A CR 11123A CR 11123 A CR11123 A CR 11123A CR 11123 A CR11123 A CR 11123A
Authority
CR
Costa Rica
Prior art keywords
containing nitrogen
antibacterial agents
compounds containing
tricycle
tricycle compounds
Prior art date
Application number
CR11123A
Other languages
English (en)
Inventor
David Evan Davies
David Thomas Davies
Ilaria Giordano
Alan Joseph Hennessy
Neil David Pearson
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39580226&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CR11123(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB0707705A external-priority patent/GB0707705D0/en
Priority claimed from GB0720569A external-priority patent/GB0720569D0/en
Priority claimed from GB0805311A external-priority patent/GB0805311D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of CR11123A publication Critical patent/CR11123A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/16Peri-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • A61P31/06Antibacterial agents for tuberculosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/16Peri-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Virology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Compuesto triciclicos que contienen nitrogeno y su uso como agentes antibacterianos.
CR11123A 2007-04-20 2009-11-20 Compuestos triciclicos que contienen nitrogeno como agentes antibacteriales CR11123A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0707705A GB0707705D0 (en) 2007-04-20 2007-04-20 Compounds
GB0720569A GB0720569D0 (en) 2007-10-19 2007-10-19 Compounds
GB0805311A GB0805311D0 (en) 2008-03-20 2008-03-20 Compounds

Publications (1)

Publication Number Publication Date
CR11123A true CR11123A (es) 2010-03-08

Family

ID=39580226

Family Applications (2)

Application Number Title Priority Date Filing Date
CR11123A CR11123A (es) 2007-04-20 2009-11-20 Compuestos triciclicos que contienen nitrogeno como agentes antibacteriales
CR20150586A CR20150586A (es) 2007-04-20 2015-10-23 Compuestos triciclicos que contienen nitrogeno como agentes antibactercianos

Family Applications After (1)

Application Number Title Priority Date Filing Date
CR20150586A CR20150586A (es) 2007-04-20 2015-10-23 Compuestos triciclicos que contienen nitrogeno como agentes antibactercianos

Country Status (31)

Country Link
US (1) US8389524B2 (es)
EP (1) EP2137196B1 (es)
JP (1) JP5389013B2 (es)
KR (1) KR101567096B1 (es)
CN (1) CN101687887B (es)
AR (1) AR066111A1 (es)
AT (1) ATE483717T1 (es)
AU (1) AU2008240764C1 (es)
BR (1) BRPI0810064B8 (es)
CA (1) CA2684659C (es)
CL (1) CL2008001122A1 (es)
CO (1) CO6251368A2 (es)
CR (2) CR11123A (es)
CY (1) CY1111248T1 (es)
DE (1) DE602008002912D1 (es)
DK (1) DK2137196T3 (es)
DO (1) DOP2009000240A (es)
EA (1) EA015821B1 (es)
HR (1) HRP20100574T1 (es)
IL (1) IL201204A0 (es)
MA (1) MA31324B1 (es)
MX (1) MX2009011317A (es)
MY (1) MY149347A (es)
NZ (1) NZ579877A (es)
PE (1) PE20090274A1 (es)
PL (1) PL2137196T3 (es)
PT (1) PT2137196E (es)
SI (1) SI2137196T1 (es)
TW (1) TWI431006B (es)
UY (1) UY31038A1 (es)
WO (1) WO2008128942A1 (es)

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ATE537175T1 (de) 2007-10-19 2011-12-15 Boehringer Ingelheim Int Neue piperazino-dihydrothienopyrimidin-derivate
ES2524910T3 (es) * 2007-10-19 2014-12-15 Boehringer Ingelheim International Gmbh Piperidino-dihidrotienopirimidinas sustituidas
JP5341899B2 (ja) 2007-10-19 2013-11-13 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ヘテロ環置換ピペラジノ−ジヒドロチエノピリミジン
US8349828B2 (en) 2008-02-20 2013-01-08 Actelion Pharmaceuticals Ltd. Azatricyclic antibiotic compounds
US20110071155A1 (en) * 2008-05-23 2011-03-24 Carlos Alemparte-Gallardo Tricyclic Nitrogen Containing Compounds And Their Use As Antibacterials
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PT2344495E (pt) 2008-10-07 2015-04-01 Actelion Pharmaceuticals Ltd Compostos antibióticos de oxazolidinona tricíclica
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US9802954B2 (en) 2011-08-24 2017-10-31 Boehringer Ingelheim International Gmbh Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma
US20130059866A1 (en) 2011-08-24 2013-03-07 Boehringer Ingelheim International Gmbh Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthma
CN103113291B (zh) * 2013-02-04 2015-03-04 浙江大学 一种3位烯基吡啶衍生物的合成方法
JP6453216B2 (ja) * 2013-07-23 2019-01-16 エーザイ・アール・アンド・ディー・マネジメント株式会社 ヘテロ縮合環化合物
EP3639824A1 (en) * 2014-08-22 2020-04-22 GlaxoSmithKline Intellectual Property Development Limited Tricyclic nitrogen containing compounds for treating neisseria gonorrhoea infection
FI3474846T3 (fi) * 2016-06-22 2023-02-16 Univ Vanderbilt Muskariinisen asetyylikoliinireseptorin m4 positiiviset allosteeriset modulaattorit
EP3612513A4 (en) 2017-04-17 2020-09-30 Ohio State Innovation Foundation TYPE II TOPOISOMERASE INHIBITORS AND PROCESSES FOR THE PRODUCTION AND USE OF THE LATTER
JP2022528890A (ja) * 2019-04-03 2022-06-16 グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッド 細菌性尿路感染症の治療に使用するためのゲポチダシン
WO2021004910A1 (en) 2019-07-05 2021-01-14 Glaxosmithkline Intellectual Property Development Limited Combination for the treatment of infections caused by mycoplasma genitalium
EP4125905B1 (en) 2020-04-02 2024-12-25 GlaxoSmithKline Intellectual Property Development Limited Regimen for treating a neisseria gonorrhoeae infection with gepotidacin
EP4143188A1 (en) * 2020-04-29 2023-03-08 GlaxoSmithKline Intellectual Property Development Limited Crystalline forms of gepotidacin
CN111494241B (zh) * 2020-06-01 2023-03-24 湖北洁世达环保科技有限公司 一种纸巾柔润保湿液
WO2022167515A1 (en) 2021-02-05 2022-08-11 Glaxosmithkline Intellectual Property Development Limited Oral solid dose formulations
US20250099535A1 (en) 2022-01-21 2025-03-27 Glaxosmithkline Intellectual Property Development Limited Gepotidacin and vancomycin for use in the treatment of an infection caused by staphylococcus saprophyticus
EP4316463A1 (en) 2022-08-02 2024-02-07 GlaxoSmithKline Intellectual Property Development Limited Novel formulation
WO2024068524A1 (en) 2022-09-26 2024-04-04 Glaxosmithkline Intellectual Property Development Limited Gepotidacin for use in the treatment of bacterial prostatitis

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Also Published As

Publication number Publication date
CA2684659A1 (en) 2008-10-30
BRPI0810064B1 (pt) 2021-03-30
CY1111248T1 (el) 2015-06-11
CR20150586A (es) 2016-04-04
CN101687887A (zh) 2010-03-31
PT2137196E (pt) 2010-12-16
AU2008240764A1 (en) 2008-10-30
DE602008002912D1 (de) 2010-11-18
AU2008240764B2 (en) 2011-04-07
BRPI0810064B8 (pt) 2021-05-25
EA015821B1 (ru) 2011-12-30
TW200848420A (en) 2008-12-16
AR066111A1 (es) 2009-07-22
ATE483717T1 (de) 2010-10-15
EP2137196A1 (en) 2009-12-30
UY31038A1 (es) 2008-11-28
JP2010524884A (ja) 2010-07-22
CA2684659C (en) 2015-11-24
SI2137196T1 (sl) 2011-01-31
TWI431006B (zh) 2014-03-21
CO6251368A2 (es) 2011-02-21
DOP2009000240A (es) 2009-12-31
BRPI0810064A2 (pt) 2019-08-27
PL2137196T3 (pl) 2011-03-31
AU2008240764C1 (en) 2011-10-20
US20100137282A1 (en) 2010-06-03
MA31324B1 (fr) 2010-04-01
KR20100017133A (ko) 2010-02-16
EA200970987A1 (ru) 2010-04-30
DK2137196T3 (da) 2011-01-10
WO2008128942A1 (en) 2008-10-30
PE20090274A1 (es) 2009-04-03
KR101567096B1 (ko) 2015-11-06
EP2137196B1 (en) 2010-10-06
CN101687887B (zh) 2012-08-29
HRP20100574T1 (hr) 2010-12-31
IL201204A0 (en) 2010-05-17
NZ579877A (en) 2011-09-30
MY149347A (en) 2013-08-30
HK1138000A1 (en) 2010-08-13
JP5389013B2 (ja) 2014-01-15
MX2009011317A (es) 2009-11-05
CL2008001122A1 (es) 2008-10-24
US8389524B2 (en) 2013-03-05

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