CR5959A - Tratamiento para la disfuncion sexual femenina - Google Patents
Tratamiento para la disfuncion sexual femeninaInfo
- Publication number
- CR5959A CR5959A CR5959A CR5959A CR5959A CR 5959 A CR5959 A CR 5959A CR 5959 A CR5959 A CR 5959A CR 5959 A CR5959 A CR 5959A CR 5959 A CR5959 A CR 5959A
- Authority
- CR
- Costa Rica
- Prior art keywords
- apomorphine
- treatment
- sexual dysfunction
- female sexual
- clitoris
- Prior art date
Links
- 206010057671 Female sexual dysfunction Diseases 0.000 title 1
- VMWNQDUVQKEIOC-CYBMUJFWSA-N apomorphine Chemical compound C([C@H]1N(C)CC2)C3=CC=C(O)C(O)=C3C3=C1C2=CC=C3 VMWNQDUVQKEIOC-CYBMUJFWSA-N 0.000 abstract 3
- 229960004046 apomorphine Drugs 0.000 abstract 3
- 239000008280 blood Substances 0.000 abstract 2
- 210000004369 blood Anatomy 0.000 abstract 2
- 210000003029 clitoris Anatomy 0.000 abstract 2
- 230000000694 effects Effects 0.000 abstract 1
- 230000001568 sexual effect Effects 0.000 abstract 1
- 230000000638 stimulation Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/02—Drugs for genital or sexual disorders; Contraceptives for disorders of the vagina
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Emergency Medicine (AREA)
- Epidemiology (AREA)
- Gynecology & Obstetrics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Compounds Of Unknown Constitution (AREA)
- Medicines Containing Plant Substances (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Abstract
LA DISFUNSION SEXUAL EN LA MUJER PUEDE SER AMINORADA, SIN EFECTOS SECUNDARIOS SUBSTANCIALES INDESEABLES POR LA ADMINISTRACION SUBLINGUAL DE DOSIS DE APOMORFINA. LA ADMINISTRACION DE APOMORFINA INCREMENTA LA ESTIMULACION DEL CLITORIS MEDIANTE EL FLUJO DE LA SANGRE INTRACAVERNOSAL Y EL FLUJO DE SANGRE EN LAS PAREDES DE LA VAGINA PARA OBTENER LA ERECCION DEL CLITORIS Y EL CONGESTIONAMIENTO VAGINAL DE LA MUJER. LA CONCENTRACION DE PLASMA DE APOMORFINA DE NO MAS DE 5.5 MANOGRAMOS POR MILILITRO ES PREFERIBLEMENTE MANTENIDA.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/016,252 US5945117A (en) | 1998-01-30 | 1998-01-30 | Treatment of female sexual dysfunction |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CR5959A true CR5959A (es) | 1999-07-28 |
Family
ID=21776169
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CR5959A CR5959A (es) | 1998-01-30 | 1999-01-28 | Tratamiento para la disfuncion sexual femenina |
Country Status (34)
| Country | Link |
|---|---|
| US (2) | US5945117A (es) |
| EP (1) | EP1056419A4 (es) |
| JP (1) | JP2002501875A (es) |
| KR (1) | KR20010040477A (es) |
| CN (1) | CN1250221C (es) |
| AR (1) | AR017976A1 (es) |
| AU (1) | AU752928B2 (es) |
| BG (1) | BG64667B1 (es) |
| BR (1) | BR9908038A (es) |
| CA (1) | CA2322289A1 (es) |
| CO (1) | CO4970819A1 (es) |
| CR (1) | CR5959A (es) |
| DZ (1) | DZ2714A1 (es) |
| GC (1) | GC0000096A (es) |
| GT (1) | GT199900013A (es) |
| HK (1) | HK1040901B (es) |
| HN (1) | HN1999000015A (es) |
| HU (1) | HUP0101268A3 (es) |
| IL (2) | IL137569A0 (es) |
| JO (1) | JO2085B1 (es) |
| MA (1) | MA26600A1 (es) |
| MX (1) | MXPA00007447A (es) |
| NO (1) | NO319821B1 (es) |
| NZ (1) | NZ506597A (es) |
| PA (1) | PA8467801A1 (es) |
| PE (1) | PE20000240A1 (es) |
| PL (1) | PL194350B1 (es) |
| SK (1) | SK11362000A3 (es) |
| TN (1) | TNSN99008A1 (es) |
| TR (1) | TR200002220T2 (es) |
| TW (1) | TW550069B (es) |
| UY (1) | UY25374A1 (es) |
| WO (1) | WO1999038467A1 (es) |
| ZA (1) | ZA99686B (es) |
Families Citing this family (47)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20020165122A1 (en) * | 1994-04-22 | 2002-11-07 | Heaton Jeremy P. W. | Method and compositions for the treatment or amelioration of female sexual dysfunction |
| US6395744B1 (en) * | 1994-04-22 | 2002-05-28 | Queen's University At Kingston | Method and compositions for the treatment or amelioration of female sexual dysfunction |
| US20050065161A1 (en) * | 1996-02-02 | 2005-03-24 | Nitromed, Inc. | Nitrosated and nitrosylated alpha-adrenergic receptor antagonist compounds, compositions and their uses |
| US6472425B1 (en) | 1997-10-31 | 2002-10-29 | Nitromed, Inc. | Methods for treating female sexual dysfunctions |
| US5945117A (en) * | 1998-01-30 | 1999-08-31 | Pentech Pharmaceuticals, Inc. | Treatment of female sexual dysfunction |
| AU2003204720B2 (en) * | 1998-05-29 | 2006-06-29 | Tap Pharmaceutical Products Inc. | Methods for the normalization of sexual response and amelioration of long term genital tissue degradation |
| EP1089736A2 (en) * | 1998-06-22 | 2001-04-11 | Queen's University At Kingston | Method and compositions for the treatment or amelioration of female sexual dysfunction |
| US20050245494A1 (en) * | 1999-07-01 | 2005-11-03 | 40 J's Llc | Methods to treat one or all of the defined etiologies of female sexual dysfunction |
| US20040254153A1 (en) * | 1999-11-08 | 2004-12-16 | Pfizer Inc | Compounds for the treatment of female sexual dysfunction |
| BR0005797A (pt) * | 2000-03-20 | 2001-10-16 | Abbott Lab | Métodos para o tratamento de disfunção sexual com apomorfina em nìveis de concentração plasmática especificados |
| CN1471395A (zh) * | 2000-04-07 | 2004-01-28 | ����ҽҩƷ����˾ | 阿扑吗啡衍生物及其使用方法 |
| CA2408399A1 (en) | 2000-05-09 | 2001-11-15 | Nitromed, Inc. | Infrared thermography and methods of use |
| ES2291333T3 (es) * | 2000-06-27 | 2008-03-01 | Qualilife Pharmaceuticals Inc. | Composiciones y metodos para el tratamiento de la respuesta sexual de las mujeres. |
| EP1365794A2 (en) * | 2000-07-21 | 2003-12-03 | Lue, Tom | Prevention and treatment of sexual arousal disorders |
| US7223406B2 (en) | 2000-07-21 | 2007-05-29 | The Regents Of The University Of California | Methods and compositions for preventing and treating male erectile dysfunction and female sexual arousal disorder |
| US20020065286A1 (en) * | 2000-08-21 | 2002-05-30 | Davies Michael John | Treatment of wounds |
| CN1486183A (zh) | 2000-11-15 | 2004-03-31 | ����ҽҩƷ����˾ | 使用阿朴吗啡治疗抗抑郁药引发的性功能障碍 |
| WO2002041894A2 (en) * | 2000-11-22 | 2002-05-30 | Abbott Laboratories | Selective dopamine d4 receptor agonists for treating sexual dysfunction |
| MXPA03007081A (es) * | 2001-02-08 | 2004-10-15 | Pharmacia Corp | Medicamento de accion rapida para el tratamiento de disfuncion sexual. |
| KR20050008658A (ko) * | 2002-03-19 | 2005-01-21 | 마이클 홀릭 | 아포모르핀의 글리코시드 및 오르토에스테르 글리코시드유도체들, 유사체들 및 그것의 용도 |
| US20030219696A1 (en) * | 2002-05-23 | 2003-11-27 | Moreland Gerald W. | Method and apparatus for preventing backflow in dental saliva evacuators |
| GB0219961D0 (en) | 2002-08-28 | 2002-10-02 | Pfizer Ltd | Oxytocin inhibitors |
| GB0221711D0 (en) * | 2002-09-19 | 2002-10-30 | Ardana Bioscience Ltd | Methods |
| CA2445212A1 (en) * | 2002-10-10 | 2004-04-10 | Queen's University At Kingston | Treatment of sexual dysfunction |
| CA2451267A1 (en) * | 2002-12-13 | 2004-06-13 | Warner-Lambert Company Llc | Pharmaceutical uses for alpha2delta ligands |
| US20040204439A1 (en) * | 2003-04-14 | 2004-10-14 | Staniforth John Nicholas | Composition, device, and method for treating sexual dysfunction via inhalation |
| JP2006522785A (ja) * | 2003-04-14 | 2006-10-05 | ベクトゥラ・リミテッド | アポモルヒネを含む肺吸入用医薬組成物 |
| US7306812B2 (en) | 2003-05-09 | 2007-12-11 | Cephalon, Inc. | Dissolvable backing layer for use with a transmucosal delivery device |
| US7276246B2 (en) * | 2003-05-09 | 2007-10-02 | Cephalon, Inc. | Dissolvable backing layer for use with a transmucosal delivery device |
| GB0314054D0 (en) * | 2003-06-17 | 2003-07-23 | Pfizer Ltd | Amide derivatives as selective serotonin re-uptake inhibitors |
| US20050054688A1 (en) * | 2003-08-08 | 2005-03-10 | Pfizer Inc | Selective serotonin reuptake inhibitors in the treatment of disease |
| DE10338174A1 (de) * | 2003-08-20 | 2005-03-24 | Lts Lohmann Therapie-Systeme Ag | Transdermale Arzneimittelzubereitungen mit Wirkstoffkombinationen zur Behandlung der Parkinson-Krankheit |
| US7291640B2 (en) * | 2003-09-22 | 2007-11-06 | Pfizer Inc. | Substituted triazole derivatives as oxytocin antagonists |
| GB0409744D0 (en) * | 2004-04-30 | 2004-06-09 | Pfizer Ltd | Novel compounds |
| AP2006003771A0 (en) * | 2004-04-30 | 2006-10-31 | Warner Lambert Co | Substituted morpholine compounds for the treatmentof central nervous system disorders |
| JP2008533193A (ja) * | 2005-03-21 | 2008-08-21 | ファイザー・リミテッド | オキシトシン拮抗薬としての置換トリアゾール誘導体 |
| WO2006100557A1 (en) * | 2005-03-21 | 2006-09-28 | Pfizer Limited | Substituted triazole derivatives as oxytocin antagonists |
| RU2406480C2 (ru) * | 2005-04-08 | 2010-12-20 | Озфарма Пти Лтд | Трансбуккальная система доставки |
| CA2618103A1 (en) * | 2005-08-10 | 2007-02-15 | Pfizer Limited | Substituted triazole derivatives as oxytocin antagonists |
| EP2233472B1 (en) | 2006-03-28 | 2014-01-15 | Atir Holding S.A. | Heterocyclic compounds and uses thereof in the treatment of sexual disorders |
| US7800094B2 (en) * | 2007-06-11 | 2010-09-21 | Macronix International Co., Ltd. | Resistance memory with tungsten compound and manufacturing |
| PL2952191T3 (pl) | 2009-06-12 | 2019-02-28 | Sunovion Pharmaceuticals Inc. | Apomorfina w postaci do podawania podjęzykowego |
| US20130210867A1 (en) * | 2010-04-15 | 2013-08-15 | Life Science Enhancement Corporation | Methods and compositions for enhancing female sexual arousal and treating female sexual dysfunction |
| EA031156B1 (ru) * | 2010-12-16 | 2018-11-30 | Суновион Фармасьютикалз Инк. | Сублингвальные пленки |
| WO2012140642A1 (en) | 2011-04-10 | 2012-10-18 | Atir Holding S.A. | Heterocyclic compounds and uses thereof in the treatment of sexual disorders |
| EP2545905A1 (en) | 2011-07-11 | 2013-01-16 | Britannia Pharmaceuticals Limited | A new therapeutical composition containing apomorphine as active ingredient |
| EP3285771B1 (en) | 2015-04-21 | 2025-02-12 | Sunovion Pharmaceuticals Inc. | Methods of treating parkinson's disease by administration of apomorphine to an oral mucosa |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4521421A (en) * | 1983-09-26 | 1985-06-04 | Eli Lilly And Company | Treatment of sexual dysfunction |
| JPH07506823A (ja) * | 1992-05-18 | 1995-07-27 | スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー | 記憶障害,性的機能不全およびパーキンソン氏病の治療のためのインドロン誘導体の使用 |
| US5565466A (en) * | 1993-08-13 | 1996-10-15 | Zonagen, Inc. | Methods for modulating the human sexual response |
| ES2143049T3 (es) * | 1994-04-22 | 2000-05-01 | Pentech Pharmaceuticals Inc | Formas sublinguales de dosificacion que contienen apomorfina y su uso para el tratamiento de la disfuncion erectil. |
| US5562917A (en) * | 1994-12-23 | 1996-10-08 | Pentech Pharmaceuticals, Inc. | Transdermal administration of apomorphine |
| US5624677A (en) * | 1995-06-13 | 1997-04-29 | Pentech Pharmaceuticals, Inc. | Controlled release of drugs delivered by sublingual or buccal administration |
| US5945117A (en) * | 1998-01-30 | 1999-08-31 | Pentech Pharmaceuticals, Inc. | Treatment of female sexual dysfunction |
-
1998
- 1998-01-30 US US09/016,252 patent/US5945117A/en not_active Expired - Fee Related
-
1999
- 1999-01-21 TN TNTNSN99008A patent/TNSN99008A1/fr unknown
- 1999-01-28 PL PL99342062A patent/PL194350B1/pl unknown
- 1999-01-28 NZ NZ506597A patent/NZ506597A/en unknown
- 1999-01-28 ZA ZA9900686A patent/ZA99686B/xx unknown
- 1999-01-28 JP JP2000529203A patent/JP2002501875A/ja not_active Withdrawn
- 1999-01-28 KR KR1020007008333A patent/KR20010040477A/ko not_active Ceased
- 1999-01-28 HN HN1999000015A patent/HN1999000015A/es unknown
- 1999-01-28 JO JO19992085A patent/JO2085B1/en active
- 1999-01-28 AU AU25644/99A patent/AU752928B2/en not_active Ceased
- 1999-01-28 BR BR9908038-9A patent/BR9908038A/pt not_active Application Discontinuation
- 1999-01-28 HU HU0101268A patent/HUP0101268A3/hu unknown
- 1999-01-28 MX MXPA00007447A patent/MXPA00007447A/es not_active IP Right Cessation
- 1999-01-28 CN CNB998044423A patent/CN1250221C/zh not_active Expired - Fee Related
- 1999-01-28 CR CR5959A patent/CR5959A/es not_active Application Discontinuation
- 1999-01-28 HK HK02101988.0A patent/HK1040901B/zh not_active IP Right Cessation
- 1999-01-28 SK SK1136-2000A patent/SK11362000A3/sk unknown
- 1999-01-28 EP EP99905497A patent/EP1056419A4/en not_active Withdrawn
- 1999-01-28 WO PCT/US1999/001776 patent/WO1999038467A1/en not_active Ceased
- 1999-01-28 CA CA002322289A patent/CA2322289A1/en not_active Abandoned
- 1999-01-28 TR TR2000/02220T patent/TR200002220T2/xx unknown
- 1999-01-28 IL IL13756999A patent/IL137569A0/xx active IP Right Grant
- 1999-01-29 TW TW088101384A patent/TW550069B/zh not_active IP Right Cessation
- 1999-01-29 PA PA19998467801A patent/PA8467801A1/es unknown
- 1999-01-29 CO CO99005067A patent/CO4970819A1/es unknown
- 1999-01-29 PE PE1999000067A patent/PE20000240A1/es not_active Application Discontinuation
- 1999-01-29 UY UY25374A patent/UY25374A1/es not_active Application Discontinuation
- 1999-01-29 AR ARP990100389A patent/AR017976A1/es not_active Application Discontinuation
- 1999-01-29 MA MA25442A patent/MA26600A1/fr unknown
- 1999-01-30 DZ DZ990015A patent/DZ2714A1/xx active
- 1999-01-31 GC GCP199973 patent/GC0000096A/xx active
- 1999-07-02 US US09/345,009 patent/US6193992B1/en not_active Expired - Fee Related
-
2000
- 2000-07-27 NO NO20003845A patent/NO319821B1/no unknown
- 2000-07-27 IL IL137569A patent/IL137569A/en unknown
- 2000-08-28 BG BG104715A patent/BG64667B1/bg unknown
-
2001
- 2001-07-20 GT GT199900013A patent/GT199900013A/es unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal (granting procedure) |