CR7039A - Modificacion cristalina de un depsipeptido ciclico con actividad mejorada - Google Patents

Modificacion cristalina de un depsipeptido ciclico con actividad mejorada

Info

Publication number
CR7039A
CR7039A CR7039A CR7039A CR7039A CR 7039 A CR7039 A CR 7039A CR 7039 A CR7039 A CR 7039A CR 7039 A CR7039 A CR 7039A CR 7039 A CR7039 A CR 7039A
Authority
CR
Costa Rica
Prior art keywords
cyclic depsipeptide
improved activity
crystal modification
depsipeptide
cyclic
Prior art date
Application number
CR7039A
Other languages
English (en)
Inventor
Kalbe Jochen
Traebuel Michael
Harder Achim
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of CR7039A publication Critical patent/CR7039A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K11/00—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K11/02—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15—Depsipeptides; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Engineering & Computer Science (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

La invencion se refiere al empleo de la modificacion cristalina (I) del depsipeptido ciclico de la formula (I) para la obtencion de medicamentos, especialmente para la lucha contra endoparasitos.
CR7039A 2001-02-01 2003-07-30 Modificacion cristalina de un depsipeptido ciclico con actividad mejorada CR7039A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10104362A DE10104362A1 (de) 2001-02-01 2001-02-01 Kristallmodifikation eines cyclischen Depsipeptids mit besserer Wirksamkeit

Publications (1)

Publication Number Publication Date
CR7039A true CR7039A (es) 2004-06-08

Family

ID=7672376

Family Applications (1)

Application Number Title Priority Date Filing Date
CR7039A CR7039A (es) 2001-02-01 2003-07-30 Modificacion cristalina de un depsipeptido ciclico con actividad mejorada

Country Status (27)

Country Link
US (1) US20040115483A1 (es)
EP (1) EP1357932B1 (es)
JP (1) JP2004525111A (es)
KR (2) KR20030081378A (es)
CN (1) CN1278735C (es)
AT (1) ATE284703T1 (es)
AU (1) AU2002226415B2 (es)
BR (1) BRPI0206841B8 (es)
CA (1) CA2436832C (es)
CR (1) CR7039A (es)
CZ (1) CZ299564B6 (es)
DE (2) DE10104362A1 (es)
EE (1) EE05490B1 (es)
ES (1) ES2233805T3 (es)
HR (1) HRP20030635A2 (es)
HU (1) HU229229B1 (es)
IL (2) IL157026A0 (es)
MX (1) MXPA03006866A (es)
NO (1) NO331289B1 (es)
NZ (1) NZ527230A (es)
PL (1) PL213106B1 (es)
PT (1) PT1357932E (es)
RU (1) RU2300390C2 (es)
SK (1) SK286280B6 (es)
UA (1) UA74623C2 (es)
WO (1) WO2002066048A1 (es)
ZA (1) ZA200305864B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20080003546A1 (en) * 2006-06-29 2008-01-03 Dunbar Kimberly L Animated digital charted yarncraft instruction
CN107835818B (zh) 2015-05-20 2022-04-29 勃林格殷格翰动物保健美国公司 驱虫缩酚酸肽化合物
KR20220003663A (ko) 2015-12-28 2022-01-10 뵈링거 잉겔하임 애니멀 헬스 유에스에이 인코포레이티드 구충성 뎁시펩티드 화합물
EP3541789A1 (en) 2016-11-16 2019-09-25 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic depsipeptide compounds
CN114195732A (zh) * 2022-01-04 2022-03-18 丽珠集团福州福兴医药有限公司 一种艾默德斯的单晶型iii及其制备方法
CN114262303A (zh) * 2022-01-04 2022-04-01 丽珠集团福州福兴医药有限公司 一种艾默德斯的单晶型ii及其制备方法
CN114989110A (zh) * 2022-07-13 2022-09-02 丽珠集团福州福兴医药有限公司 单晶型ⅳ的艾默德斯及其制备方法
CN115010680A (zh) * 2022-07-13 2022-09-06 丽珠集团福州福兴医药有限公司 单晶型i的艾默德斯及其制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2096907A (en) * 1981-04-22 1982-10-27 Exxon Research Engineering Co Distillation column with steam stripping
CA2132199C (en) * 1992-03-17 2000-01-18 Hitoshi Nishiyama Depsipeptide derivative, production thereof and use thereof
DE4317458A1 (de) * 1992-06-11 1993-12-16 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
DE4400464A1 (de) * 1994-01-11 1995-07-13 Bayer Ag Endoparasitizide Mittel
CN1071323C (zh) * 1995-06-30 2001-09-19 藤泽药品工业株式会社 缩肽衍生物或其盐的制造方法
NZ318515A (en) * 1995-09-22 2000-05-26 Bayer Ag Cyclodepsipeptide PF1022 derivatives and compositions thereof
ATE221055T1 (de) * 1997-11-10 2002-08-15 Fujisawa Pharmaceutical Co Kristall eines depsipeptid-derivates und verfahren zu seiner herstellung
DE10008128A1 (de) * 2000-02-22 2001-08-23 Bayer Ag Endoparasitizide Mittel
DE10031044A1 (de) * 2000-06-26 2002-01-03 Bayer Ag Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere

Also Published As

Publication number Publication date
DE10104362A1 (de) 2002-08-08
US20040115483A1 (en) 2004-06-17
EP1357932B1 (de) 2004-12-15
BRPI0206841B8 (pt) 2021-05-25
IL157026A (en) 2010-11-30
RU2003126589A (ru) 2005-02-27
CN1592631A (zh) 2005-03-09
MXPA03006866A (es) 2004-05-31
PT1357932E (pt) 2005-04-29
EE05490B1 (et) 2011-12-15
HU229229B1 (en) 2013-09-30
CZ20032063A3 (cs) 2003-11-12
HUP0302880A2 (hu) 2003-12-29
ATE284703T1 (de) 2005-01-15
NO20033413L (no) 2003-09-26
CA2436832C (en) 2013-06-11
CN1278735C (zh) 2006-10-11
EE200300365A (et) 2003-10-15
WO2002066048A1 (de) 2002-08-29
NO331289B1 (no) 2011-11-21
WO2002066048A8 (de) 2003-11-20
PL213106B1 (pl) 2013-01-31
DE50201777D1 (de) 2005-01-20
EP1357932A1 (de) 2003-11-05
KR20030081378A (ko) 2003-10-17
HUP0302880A3 (en) 2005-05-30
NZ527230A (en) 2005-04-29
UA74623C2 (en) 2006-01-16
HRP20030635A2 (en) 2005-10-31
SK9882003A3 (en) 2003-12-02
KR20090041451A (ko) 2009-04-28
CA2436832A1 (en) 2002-08-29
SK286280B6 (sk) 2008-06-06
JP2004525111A (ja) 2004-08-19
ES2233805T3 (es) 2005-06-16
HK1075013A1 (en) 2005-12-02
BRPI0206841B1 (pt) 2018-02-14
NO20033413D0 (no) 2003-07-30
AU2002226415B2 (en) 2007-03-22
PL362389A1 (en) 2004-11-02
CZ299564B6 (cs) 2008-09-03
BR0206841A (pt) 2004-02-25
ZA200305864B (en) 2004-08-27
IL157026A0 (en) 2004-02-08
RU2300390C2 (ru) 2007-06-10

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