CR7678A - Heterociclilpyrimidinos sustituidos - Google Patents

Heterociclilpyrimidinos sustituidos

Info

Publication number
CR7678A
CR7678A CR7678A CR7678A CR7678A CR 7678 A CR7678 A CR 7678A CR 7678 A CR7678 A CR 7678A CR 7678 A CR7678 A CR 7678A CR 7678 A CR7678 A CR 7678A
Authority
CR
Costa Rica
Prior art keywords
heterociclilpyrimidinos
replaced
heterocyclypyrimidines
fluorine
procedures
Prior art date
Application number
CR7678A
Other languages
English (en)
Inventor
Rudiger Fischer
Thomas Bretschneider
Fritz Maurer
Christoph Erdelen
Jorg Konze
Peter Losel
Yukiyoshi Watanabe
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of CR7678A publication Critical patent/CR7678A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Se refiere a heterociclipirimidinas susbtituidas de la formula que se presenta. En la que n significa los numero 0, 1 o 2. R significa hidrogeno o fluor y X, Y y Z tienen los significados indicados en la descripcion. a procedimientos para su obtencion y a su empleo como agentes para la lucha contra las pestes.
CR7678A 2002-08-23 2005-02-09 Heterociclilpyrimidinos sustituidos CR7678A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10238725A DE10238725A1 (de) 2002-08-23 2002-08-23 Substituierte Heterocyclypyrimidine

Publications (1)

Publication Number Publication Date
CR7678A true CR7678A (es) 2005-09-02

Family

ID=31197289

Family Applications (1)

Application Number Title Priority Date Filing Date
CR7678A CR7678A (es) 2002-08-23 2005-02-09 Heterociclilpyrimidinos sustituidos

Country Status (18)

Country Link
US (1) US20060106042A1 (es)
EP (1) EP1534701A1 (es)
JP (1) JP2006508059A (es)
KR (1) KR20050032586A (es)
CN (1) CN1688571A (es)
AU (1) AU2003271560A1 (es)
BR (1) BR0313751A (es)
CA (1) CA2496306A1 (es)
CR (1) CR7678A (es)
DE (1) DE10238725A1 (es)
HR (1) HRP20050270A2 (es)
IL (1) IL166740A0 (es)
MX (1) MXPA05001962A (es)
NO (1) NO20051500D0 (es)
PL (1) PL375550A1 (es)
RU (1) RU2005108352A (es)
WO (1) WO2004026858A1 (es)
ZA (1) ZA200501457B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2217602B1 (en) 2007-11-30 2018-08-29 Boehringer Ingelheim International GmbH 1,5-dihydro-pyrazolo[3,4-d]pyrimidin-4-one derivatives and their use as pde9a modulators for the treatment of cns disorders
UA105362C2 (en) 2008-04-02 2014-05-12 Бьорингер Ингельхайм Интернациональ Гмбх 1-heterocyclyl-1, 5-dihydro-pyrazolo [3, 4-d] pyrimidin-4-one derivatives and their use as pde9a modulators
PE20110383A1 (es) 2008-09-08 2011-07-15 Boehringer Ingelheim Int Pirazolopirimidinonas como inhibidores de la fosfodiesterasa 9a (pde9a)
MX2011008379A (es) 2009-03-04 2011-09-06 Basf Se Compuestos de 3-arilquinazolin-4-ona para combatir plagas de invertebrados.
CA2757231A1 (en) 2009-03-31 2010-10-07 Boehringer Ingelheim International Gmbh 1-heterocyclyl-1,5-dihydro-pyrazolo [3,4-d] pyrimidin-4-one derivatives and their use as pde9a modulators
KR101123178B1 (ko) * 2009-04-09 2012-06-13 (주)에스메디 2-아릴벤조싸이오펜 유도체 또는 이의 약학적으로 허용가능한 염, 이의 제조방법 및 이를 유효성분으로 함유하는 퇴행성 뇌질환의 진단 또는 치료용 약학적 조성물
CA2807687C (en) 2010-08-12 2019-01-08 Boehringer Ingelheim International Gmbh 6-cycloalkyl-1, 5-dihydro-pyrazolo [3,4-d] pyrimidin-4-one derivatives and their use as pde9a inhibitors
US8809345B2 (en) 2011-02-15 2014-08-19 Boehringer Ingelheim International Gmbh 6-cycloalkyl-pyrazolopyrimidinones for the treatment of CNS disorders
EP3363786A1 (en) * 2017-02-15 2018-08-22 Merck Patent GmbH Compounds for optically active devices
CN120379982A (zh) 2022-12-02 2025-07-25 纽摩拉治疗公司 治疗神经障碍的方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE58904307D1 (de) * 1988-03-19 1993-06-17 Hoechst Ag Verfahren zur herstellung von ungesaettigten halogenierten kohlenwasserstoffen.
GB9205484D0 (en) * 1991-03-28 1992-04-29 Ici Plc Heterocyclic compounds
GB9219635D0 (en) * 1992-09-16 1992-10-28 Ici Plc Heterocyclic compounds
KR100234555B1 (ko) * 1993-08-05 1999-12-15 돈 리사 로얄 플루오로아테닐티오 복소환식 유도체의 제조방법
IL112721A0 (en) * 1994-03-10 1995-05-26 Zeneca Ltd Azole derivatives
GB9510459D0 (en) * 1995-05-24 1995-07-19 Zeneca Ltd Bicyclic amines
US6080772A (en) * 1995-06-07 2000-06-27 Sugen, Inc. Thiazole compounds and methods of modulating signal transduction
DE19605585A1 (de) * 1996-02-15 1997-08-21 Bayer Ag Verfahren zur Herstellung eines Gemisches aus Cyclohexylamin und Dicyclohexylamin
GB9624611D0 (en) * 1996-11-26 1997-01-15 Zeneca Ltd Bicyclic amine compounds
TR199901704T2 (xx) * 1996-11-26 1999-12-21 Zeneca Limited 8-Azabisiklo$3.2.1]oktan-, 8-azabisiklo$3.2.1]okt-6-en-,9-azabisiklo$3.3.1] nonan-,9-aza-3-oksabisiklo$3.3.1]nonan-ve 9-aza-3-tiabisiklo$3.3.1]nonan t�revleri, bunlar�n haz�rlanmas� ve insektisidler olarak kullan�mlar�.

Also Published As

Publication number Publication date
NO20051500L (no) 2005-03-21
AU2003271560A1 (en) 2004-04-08
EP1534701A1 (de) 2005-06-01
IL166740A0 (en) 2006-01-15
US20060106042A1 (en) 2006-05-18
HRP20050270A2 (hr) 2006-07-31
PL375550A1 (en) 2005-11-28
KR20050032586A (ko) 2005-04-07
BR0313751A (pt) 2005-06-21
WO2004026858A1 (de) 2004-04-01
MXPA05001962A (es) 2005-04-28
JP2006508059A (ja) 2006-03-09
NO20051500D0 (no) 2005-03-21
CN1688571A (zh) 2005-10-26
RU2005108352A (ru) 2005-08-27
ZA200501457B (en) 2006-04-26
DE10238725A1 (de) 2004-03-04
CA2496306A1 (en) 2004-04-01

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal (granting procedure)