CR7749A - NEW IMIDAZOL COMPOUNDS AS INHIBITORS OF THE TRANSFORMING GROWTH FACTOR (TGF) - Google Patents
NEW IMIDAZOL COMPOUNDS AS INHIBITORS OF THE TRANSFORMING GROWTH FACTOR (TGF)Info
- Publication number
- CR7749A CR7749A CR7749A CR7749A CR7749A CR 7749 A CR7749 A CR 7749A CR 7749 A CR7749 A CR 7749A CR 7749 A CR7749 A CR 7749A CR 7749 A CR7749 A CR 7749A
- Authority
- CR
- Costa Rica
- Prior art keywords
- tgf
- growth factor
- inhibitors
- transforming growth
- new
- Prior art date
Links
- 201000010099 disease Diseases 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 230000003176 fibrotic effect Effects 0.000 abstract 1
- 239000003102 growth factor Substances 0.000 abstract 1
- 150000002460 imidazoles Chemical class 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 230000003389 potentiating effect Effects 0.000 abstract 1
- 230000019491 signal transduction Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Se describen nuevos compuestos de imidazol, incluyendo sus derivados, intermedios para su preparacion, composiciones farmaceuticas que los contienen y su uso medicinal. Los componentes de la presente invencion son inhibidores potentes de la ruta de senalizacion del factor de crecimiento transformante ("TGF"). Son de utilidad en el tratamiento de diversos estados de enfermedad relacionados con TGF icluyendo por ejemplo, cancer, y enfermedades fibroticas.New imidazole compounds are described, including their derivatives, intermediates for their preparation, pharmaceutical compositions containing them and their medicinal use. The components of the present invention are potent inhibitors of the transformative growth factor signaling pathway ("TGF"). They are useful in the treatment of various disease states related to TGF including, for example, cancer, and fibrotic diseases.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US41189402P | 2002-09-18 | 2002-09-18 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CR7749A true CR7749A (en) | 2005-06-15 |
Family
ID=44839285
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CR7749A CR7749A (en) | 2002-09-18 | 2005-03-16 | NEW IMIDAZOL COMPOUNDS AS INHIBITORS OF THE TRANSFORMING GROWTH FACTOR (TGF) |
Country Status (3)
| Country | Link |
|---|---|
| CR (1) | CR7749A (en) |
| GT (1) | GT200300196A (en) |
| TN (1) | TNSN05083A1 (en) |
-
2003
- 2003-09-16 GT GT200300196A patent/GT200300196A/en unknown
-
2005
- 2005-03-16 CR CR7749A patent/CR7749A/en not_active Application Discontinuation
- 2005-03-18 TN TNP2005000083A patent/TNSN05083A1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| TNSN05083A1 (en) | 2007-05-14 |
| GT200300196A (en) | 2004-04-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal (granting procedure) |