CR9292A - Comprimidos con dispersion mejorada de la sustancia farmacologica - Google Patents

Comprimidos con dispersion mejorada de la sustancia farmacologica

Info

Publication number
CR9292A
CR9292A CR9292A CR9292A CR9292A CR 9292 A CR9292 A CR 9292A CR 9292 A CR9292 A CR 9292A CR 9292 A CR9292 A CR 9292A CR 9292 A CR9292 A CR 9292A
Authority
CR
Costa Rica
Prior art keywords
dispersion
conveyor
compressed
improved dispersion
pharmacological substance
Prior art date
Application number
CR9292A
Other languages
English (en)
Inventor
Nathalie Bernigal
Eric Garcia
Susanne Page
Joseph Tardio
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36406213&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CR9292(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of CR9292A publication Critical patent/CR9292A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682—Processes
    • A61K9/1694—Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Inorganic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invencion se refiere a un metodo para la preparacion de composiciones farmaceuticas en forma de comprimidos con dispersion mejorada de la sustancia farmacologica, caracterizandose dicho metodo en que comprende los pasos de: a)preparacion de una dispersion en un liquido de al menos una sustancia farmacologica activa a nivel farmaceutico y al menos un surfactante y/o enlazante; b)preparacion de un transportador mediante mezcla seca de uno o mas excipientes incluyendo al menos un transportador poroso; c) granulado por pulverizacion de la dispersion preparada en a) en un transportador preparado en b) para obtener un producto granulado por pulverizacion.
CR9292A 2005-02-25 2007-08-07 Comprimidos con dispersion mejorada de la sustancia farmacologica CR9292A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP05101458 2005-02-25

Publications (1)

Publication Number Publication Date
CR9292A true CR9292A (es) 2010-04-21

Family

ID=36406213

Family Applications (1)

Application Number Title Priority Date Filing Date
CR9292A CR9292A (es) 2005-02-25 2007-08-07 Comprimidos con dispersion mejorada de la sustancia farmacologica

Country Status (20)

Country Link
US (2) US20060193910A1 (es)
EP (2) EP1855655A2 (es)
JP (1) JP2008531509A (es)
KR (1) KR20070094666A (es)
CN (1) CN101128189A (es)
AR (1) AR055561A1 (es)
AU (1) AU2006218193A1 (es)
BR (1) BRPI0606187A2 (es)
CA (1) CA2598762A1 (es)
CR (1) CR9292A (es)
IL (1) IL185011A0 (es)
MA (1) MA29268B1 (es)
MX (1) MX2007009571A (es)
NO (1) NO20074092L (es)
NZ (1) NZ560232A (es)
RU (1) RU2007129642A (es)
TW (1) TW200640502A (es)
UA (1) UA90708C2 (es)
WO (1) WO2006089674A2 (es)
ZA (1) ZA200706495B (es)

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SG185257A1 (en) * 2007-10-10 2012-11-29 Avantor Performance Mat Inc Directly compressible high functionality granular microcrystalline cellulose based excipient, manufacturing process and use thereof
DE102008047910A1 (de) 2008-09-19 2010-03-25 Molkerei Meggle Wasserburg Gmbh & Co. Kg Tablettierhilfsstoff auf Laktose- und Cellulosebasis
RU2537224C2 (ru) * 2009-01-23 2014-12-27 Ф.Хоффманн-Ля Рош Аг Фармацевтическая композиция, содержащая алеглитазар
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KR20170003414A (ko) * 2015-06-30 2017-01-09 (주)아모레퍼시픽 속붕해형 과립환 모발 세정용 조성물
WO2017003137A1 (ko) * 2015-06-30 2017-01-05 (주)아모레퍼시픽 속붕해형 과립환 모발 세정용 조성물
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CN109701441B (zh) * 2018-12-16 2021-04-09 桂林理工大学 一种卵磷脂选择性改性高岭石的制备方法及其应用
TWI728709B (zh) * 2020-02-19 2021-05-21 台灣森本生物科技開發股份有限公司 含有得自於藤黃樹脂的丙酮萃取產物的藥學組成物以及由該組成物所製得的配方
CN111548218A (zh) * 2020-04-27 2020-08-18 上海应用技术大学 一种通用型花肥速释片及其制备方法和应用
CN116602928A (zh) * 2023-06-30 2023-08-18 康普药业股份有限公司 一种甲苯磺酸艾多沙班组合物和制备方法
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Also Published As

Publication number Publication date
NO20074092L (no) 2007-09-04
IL185011A0 (en) 2007-12-03
WO2006089674A2 (en) 2006-08-31
EP1855655A2 (en) 2007-11-21
NZ560232A (en) 2010-11-26
US20060193910A1 (en) 2006-08-31
AU2006218193A1 (en) 2006-08-31
MA29268B1 (fr) 2008-02-01
UA90708C2 (ru) 2010-05-25
JP2008531509A (ja) 2008-08-14
EP2281556A1 (en) 2011-02-09
RU2007129642A (ru) 2009-03-27
WO2006089674A3 (en) 2007-02-08
CN101128189A (zh) 2008-02-20
TW200640502A (en) 2006-12-01
ZA200706495B (en) 2008-10-29
KR20070094666A (ko) 2007-09-20
AR055561A1 (es) 2007-08-22
US20090304795A1 (en) 2009-12-10
BRPI0606187A2 (pt) 2009-06-09
MX2007009571A (es) 2007-09-21
CA2598762A1 (en) 2006-08-31

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