CR9660A - Nuevo derivado de heterocicliden acetamida - Google Patents

Nuevo derivado de heterocicliden acetamida

Info

Publication number
CR9660A
CR9660A CR9660A CR9660A CR9660A CR 9660 A CR9660 A CR 9660A CR 9660 A CR9660 A CR 9660A CR 9660 A CR9660 A CR 9660A CR 9660 A CR9660 A CR 9660A
Authority
CR
Costa Rica
Prior art keywords
group
heterocicliden
acetamida
new derivative
hydrocarbon
Prior art date
Application number
CR9660A
Other languages
English (en)
Inventor
Hideharu Uchida
Naoto Kosuga
Tsutomu Satoh
Daido Hotta
Tomoyuki Kamino
Yoshitaka Maeda
Ken-Ichi Amano
Yasushige Akada
Original Assignee
Mochida Pharm Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mochida Pharm Co Ltd filed Critical Mochida Pharm Co Ltd
Publication of CR9660A publication Critical patent/CR9660A/es

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    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
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    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
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    • C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pulmonology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Oncology (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Communicable Diseases (AREA)
  • Child & Adolescent Psychology (AREA)
  • Otolaryngology (AREA)
  • Vascular Medicine (AREA)

Abstract

La presente invencion se refiere a un compuesto, representado por la formula(I): en donde m, n, y p cada uno representa 0 hasta 2; q representa 0 o 1; R1 representa halogeno, un grupo hidrocarburo, un grupo heterociclico, un grupo alcoxi, un grupo alcoxicarbonilo, un grupo sulfamoilo, un grupo CN, o un grupo NO2 o similares; R2 representa halogeno, amino, un grupo hidrocarburo, un grupo heterociclico aromatico, o un grupo oxo; X1 representa O, -NR3- o -S(O)r-; Q representa un grupo heteroarilo, un grupo heteroarilalquilo, un grupo arilo sustituido.
CR9660A 2005-07-22 2008-01-14 Nuevo derivado de heterocicliden acetamida CR9660A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2005213534 2005-07-22
JP2005330890 2005-11-15
JP2006045985 2006-02-22

Publications (1)

Publication Number Publication Date
CR9660A true CR9660A (es) 2008-05-22

Family

ID=37668470

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Application Number Title Priority Date Filing Date
CR9660A CR9660A (es) 2005-07-22 2008-01-14 Nuevo derivado de heterocicliden acetamida

Country Status (14)

Country Link
US (2) US7910751B2 (es)
EP (1) EP1908753B1 (es)
JP (2) JP4754566B2 (es)
KR (2) KR101136183B1 (es)
AU (1) AU2006271297C1 (es)
BR (1) BRPI0613771B1 (es)
CA (1) CA2616079C (es)
CR (1) CR9660A (es)
EC (1) ECSP088129A (es)
ES (1) ES2531621T3 (es)
NO (1) NO341962B1 (es)
NZ (1) NZ565080A (es)
PT (1) PT1908753E (es)
WO (1) WO2007010383A1 (es)

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US20100016285A1 (en) * 2007-01-24 2010-01-21 Mochida Pharmaceutical Co., Ltd. Heterocyclidene-n-(aryl) acetamide derivative
PE20081692A1 (es) * 2007-01-24 2008-12-18 Mochida Pharm Co Ltd Nuevo derivado de heterocicliden acetamida
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US8765815B2 (en) 2007-09-20 2014-07-01 Ramot At Tel-Aviv University Ltd. N-phenyl anthranilic acid derivatives and uses thereof
CA2728405A1 (en) * 2008-06-17 2010-01-14 Glenmark Pharmaceuticals, S.A. Chromane derivatives as trpv3 modulators
JP2011201777A (ja) * 2008-07-23 2011-10-13 Mochida Pharmaceut Co Ltd 光学活性なヘテロシクリデン−ｎ−アリールアセトアミド誘導体
JP2011201778A (ja) * 2008-07-23 2011-10-13 Mochida Pharmaceut Co Ltd ｐ−置換アリールアセトアミドを有するヘテロシクリデン誘導体
UY33966A (es) 2011-03-25 2012-10-31 Abbott Lab Antagonistas del receptor transitorio potencial de vanilloides 1 (trpv1)
US8969325B2 (en) 2011-12-19 2015-03-03 Abbvie Inc. TRPV1 antagonists
US8859584B2 (en) 2011-12-19 2014-10-14 Abbvie, Inc. TRPV1 antagonists
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US9643947B2 (en) 2013-08-28 2017-05-09 Northwestern University 7-membered fused heterocycles and methods of their synthesis
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