CS253746B2 - Process for preparing new derivatives of pyrrolo /1,2-e//azepinone - Google Patents

Process for preparing new derivatives of pyrrolo /1,2-e//azepinone Download PDF

Info

Publication number: CS253746B2
Authority: CS; Czechoslovakia
Prior art keywords: solution; piperazinyl; washed; column; mixture
Prior art date: 1985-03-15

Application number

CS861697A

Other languages

Czech (cs)

English (en)

Inventor

Michel Barreau

Marie-Therese Comte

Daniel Farge

Jean-Luc Malleron

Gerard Ponsinet

Gerard Roussel

Original Assignee

Rhone Poulenc Sante

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-03-15

Filing date

1986-03-12

Publication date

1987-12-17

1986-03-12 Application filed by Rhone Poulenc Sante filed Critical Rhone Poulenc Sante

1986-07-08 Priority to CS865164A priority Critical patent/CS253750B2/cs

1987-12-17 Publication of CS253746B2 publication Critical patent/CS253746B2/cs

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Psychiatry (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Plural Heterocyclic Compounds (AREA)

CS861697A 1985-03-15 1986-03-12 Process for preparing new derivatives of pyrrolo /1,2-e//azepinone CS253746B2 (en)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
CS865164A CS253750B2 (cs)	1985-03-15	1986-07-08	Způsob výroby nových derivátů pyrrolo[1,2-a]azepinonu

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR8503840A FR2578842B1 (fr)	1985-03-15	1985-03-15	Nouveaux derives de la pyrrolo(1,2-a) azepinone, leur preparation et les compositions pharmaceutiques qui les contiennent

Publications (1)

Publication Number	Publication Date
CS253746B2 true CS253746B2 (en)	1987-12-17

Family

ID=9317228

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
CS861697A CS253746B2 (en)	1985-03-15	1986-03-12	Process for preparing new derivatives of pyrrolo /1,2-e//azepinone
CS865164A CS253750B2 (cs)	1985-03-15	1986-07-08	Způsob výroby nových derivátů pyrrolo[1,2-a]azepinonu

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
CS865164A CS253750B2 (cs)	1985-03-15	1986-07-08	Způsob výroby nových derivátů pyrrolo[1,2-a]azepinonu

Country Status (23)

Country	Link
US (2)	US4769366A (fi)
EP (1)	EP0196955B1 (fi)
JP (1)	JPS61215392A (fi)
KR (1)	KR860007262A (fi)
AT (1)	ATE44032T1 (fi)
AU (1)	AU576064B2 (fi)
CA (1)	CA1261323A (fi)
CS (2)	CS253746B2 (fi)
DD (1)	DD251351A5 (fi)
DE (1)	DE3663948D1 (fi)
DK (1)	DK118886A (fi)
ES (2)	ES8801275A1 (fi)
FI (2)	FI861071A7 (fi)
FR (1)	FR2578842B1 (fi)
GR (1)	GR860672B (fi)
HU (1)	HU195510B (fi)
IL (1)	IL78135A (fi)
MA (1)	MA20638A1 (fi)
NZ (1)	NZ215471A (fi)
PT (1)	PT82182B (fi)
SU (2)	SU1447285A3 (fi)
TN (1)	TNSN86037A1 (fi)
ZA (1)	ZA861881B (fi)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL121432A (en)	1995-12-01	2000-09-28	Suntory Ltd	Pyrrolo [3,2-C]azepine-4-one derivatives and pyrrolo [3,4-C]azepine-4-one derivatives their preparation and pharmaceutical compositions containing them

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1189553B (de) *	1962-08-09	1965-03-25	Degussa	Verfahren zur Herstellung von racemischen und optisch aktiven Piperazinderivaten
DE2557341A1 (de) *	1975-12-19	1977-06-30	Hoechst Ag	Basisch substituierte indolderivate und verfahren zu ihrer herstellung

1985
- 1985-03-15 FR FR8503840A patent/FR2578842B1/fr not_active Expired
1986
- 1986-03-06 MA MA20863A patent/MA20638A1/fr unknown
- 1986-03-12 GR GR860672A patent/GR860672B/el unknown
- 1986-03-12 CS CS861697A patent/CS253746B2/cs unknown
- 1986-03-12 PT PT82182A patent/PT82182B/pt unknown
- 1986-03-13 AU AU54701/86A patent/AU576064B2/en not_active Ceased
- 1986-03-13 IL IL78135A patent/IL78135A/xx unknown
- 1986-03-13 ZA ZA861881A patent/ZA861881B/xx unknown
- 1986-03-13 US US06/839,101 patent/US4769366A/en not_active Expired - Fee Related
- 1986-03-13 NZ NZ215471A patent/NZ215471A/xx unknown
- 1986-03-14 EP EP86400548A patent/EP0196955B1/fr not_active Expired
- 1986-03-14 AT AT86400548T patent/ATE44032T1/de not_active IP Right Cessation
- 1986-03-14 TN TNTNSN86037A patent/TNSN86037A1/fr unknown
- 1986-03-14 FI FI861071A patent/FI861071A7/fi not_active Application Discontinuation
- 1986-03-14 DK DK118886A patent/DK118886A/da not_active Application Discontinuation
- 1986-03-14 SU SU864027174A patent/SU1447285A3/ru active
- 1986-03-14 HU HU861083A patent/HU195510B/hu not_active IP Right Cessation
- 1986-03-14 CA CA000504176A patent/CA1261323A/fr not_active Expired
- 1986-03-14 ES ES553028A patent/ES8801275A1/es not_active Expired
- 1986-03-14 KR KR1019860001870A patent/KR860007262A/ko not_active Withdrawn
- 1986-03-14 JP JP61055136A patent/JPS61215392A/ja active Pending
- 1986-03-14 FI FI892181A patent/FI892181A0/fi not_active Application Discontinuation
- 1986-03-14 DD DD86287910A patent/DD251351A5/de unknown
- 1986-03-14 DE DE8686400548T patent/DE3663948D1/de not_active Expired
- 1986-06-25 ES ES556722A patent/ES8800947A1/es not_active Expired
- 1986-07-08 CS CS865164A patent/CS253750B2/cs unknown
- 1986-12-23 SU SU864028690A patent/SU1537139A3/ru active
1987
- 1987-11-04 US US07/116,725 patent/US4826974A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
US4769366A (en)	1988-09-06
DK118886A (da)	1986-09-16
DK118886D0 (da)	1986-03-14
TNSN86037A1 (fr)	1990-01-01
ES556722A0 (es)	1987-12-01
FI892181L (fi)	1989-05-05
FI892181A7 (fi)	1989-05-05
FR2578842B1 (fr)	1987-04-10
ES8800947A1 (es)	1987-12-01
CA1261323A (fr)	1989-09-26
DE3663948D1 (en)	1989-07-20
US4826974A (en)	1989-05-02
ATE44032T1 (de)	1989-06-15
MA20638A1 (fr)	1986-10-01
FR2578842A1 (fr)	1986-09-19
ZA861881B (en)	1986-12-30
FI861071A7 (fi)	1986-09-16
ES553028A0 (es)	1987-12-16
KR860007262A (ko)	1986-10-10
SU1447285A3 (ru)	1988-12-23
ES8801275A1 (es)	1987-12-16
HU195510B (en)	1988-05-30
AU5470186A (en)	1986-09-18
GR860672B (en)	1986-05-27
EP0196955A1 (fr)	1986-10-08
SU1537139A3 (ru)	1990-01-15
DD251351A5 (de)	1987-11-11
HUT42773A (en)	1987-08-28
PT82182A (fr)	1986-04-01
PT82182B (fr)	1988-01-07
IL78135A (en)	1989-02-28
AU576064B2 (en)	1988-08-11
IL78135A0 (en)	1986-07-31
NZ215471A (en)	1988-08-30
EP0196955B1 (fr)	1989-06-14
JPS61215392A (ja)	1986-09-25
FI861071A0 (fi)	1986-03-14
CS253750B2 (cs)	1987-12-17
FI892181A0 (fi)	1989-05-05

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