CY1604A - Pharmaceutical 9,10-dihydro ergot alkaloid containing compositions - Google Patents

Pharmaceutical 9,10-dihydro ergot alkaloid containing compositions Download PDF

Info

Publication number: CY1604A
Authority: CY; Cyprus
Prior art keywords: dergocrine; aformulation; dihydroergotamine; formulation; formulation according
Prior art date: 1985-02-05

Application number

CY1604A

Other languages

English (en)

Original Assignee

Sandoz Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-02-05

Filing date

1992-04-03

Publication date

1992-04-03

1985-02-05 Priority claimed from GB858502889A external-priority patent/GB8502889D0/en

1985-07-12 Priority claimed from GB858517604A external-priority patent/GB8517604D0/en

1992-04-03 Application filed by Sandoz Ltd filed Critical Sandoz Ltd

1992-04-03 Publication of CY1604A publication Critical patent/CY1604A/en

Links

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229960003133 ergot alkaloid Drugs 0.000 title claims description 24
238000009472 formulation Methods 0.000 claims description 29
229960004704 dihydroergotamine Drugs 0.000 claims description 25
239000000463 material Substances 0.000 claims description 23
HESHRHUZIWVEAJ-JGRZULCMSA-N dihydroergotamine Chemical compound C([C@H]1C(=O)N2CCC[C@H]2[C@]2(O)O[C@@](C(N21)=O)(C)NC(=O)[C@H]1CN([C@H]2[C@@H](C3=CC=CC4=NC=C([C]34)C2)C1)C)C1=CC=CC=C1 HESHRHUZIWVEAJ-JGRZULCMSA-N 0.000 claims description 21
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SBFXHXZNBNFPHV-PXXBSISHSA-N epicriptine Chemical compound C1=CC([C@H]2C[C@H](CN(C)[C@@H]2C2)C(=O)N[C@]3(C(=O)N4[C@H](C(N5CCC[C@H]5[C@]4(O)O3)=O)[C@H](C)CC)C(C)C)=C3C2=CNC3=C1 SBFXHXZNBNFPHV-PXXBSISHSA-N 0.000 claims description 11
FLPJVCMIKUWSDR-UHFFFAOYSA-N 2-(4-formylphenoxy)acetamide Chemical compound NC(=O)COC1=CC=C(C=O)C=C1 FLPJVCMIKUWSDR-UHFFFAOYSA-N 0.000 claims description 10
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230000001225 therapeutic effect Effects 0.000 description 1
230000002792 vascular Effects 0.000 description 1
XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 description 1
XOOUIPVCVHRTMJ-UHFFFAOYSA-L zinc stearate Chemical class [Zn+2].CCCCCCCCCCCCCCCCCC([O-])=O.CCCCCCCCCCCCCCCCCC([O-])=O XOOUIPVCVHRTMJ-UHFFFAOYSA-L 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/48—Ergoline derivatives, e.g. lysergic acid, ergotamine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4866—Organic macromolecular compounds

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

CY1604A 1985-02-05 1992-04-03 Pharmaceutical 9,10-dihydro ergot alkaloid containing compositions CY1604A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB858502889A GB8502889D0 (en)	1985-02-05	1985-02-05	Co-dergocrine compositions
GB858517604A GB8517604D0 (en)	1985-07-12	1985-07-12	Dihydroergotamine compositions

Publications (1)

Publication Number	Publication Date
CY1604A true CY1604A (en)	1992-04-03

Family

ID=26288767

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CY1604A CY1604A (en)	1985-02-05	1992-04-03	Pharmaceutical 9,10-dihydro ergot alkaloid containing compositions

Country Status (24)

Country	Link
JP (1)	JPS61183225A (fr)
KR (1)	KR920010388B1 (fr)
AU (1)	AU597570B2 (fr)
BE (1)	BE904152A (fr)
CA (1)	CA1263087A (fr)
CH (1)	CH667592A5 (fr)
CY (1)	CY1604A (fr)
DE (1)	DE3602577A1 (fr)
DK (1)	DK167138B1 (fr)
ES (1)	ES8800040A1 (fr)
FR (1)	FR2576787B1 (fr)
GB (1)	GB2170407B (fr)
GR (1)	GR860310B (fr)
HK (1)	HK57191A (fr)
HU (1)	HU195729B (fr)
IE (1)	IE59293B1 (fr)
IT (1)	IT1191255B (fr)
LU (1)	LU86289A1 (fr)
NL (1)	NL8600161A (fr)
NZ (1)	NZ215020A (fr)
PH (1)	PH23384A (fr)
PT (1)	PT81954B (fr)
SE (1)	SE8600496L (fr)
SG (1)	SG56191G (fr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2610827B1 (fr) *	1987-02-18	1991-09-13	Pf Medicament	Comprime de dihydroergotamine (d.h.e.) du type a matrice hydrophile et son procede de fabrication
SI8710406B (sl) *	1987-03-11	1998-08-31	Lek	Tablete s podaljšanim delovanjem na osnovi hidroksipropilmetilceluloze z veliko molsko maso in postopek za njihovo pripravo
US7771746B2 (en)	1999-12-03	2010-08-10	Polichem Sa	Methods for making sustained-release pharmaceutical compositions of ergot alkaloids having improved bioavailability and compositions thereof
EP1512403A1 (fr) *	1999-12-03	2005-03-09	Polichem S.A.	Pocédés permettant la préparation de compositions pharmaceutiques à libération prolongée d'alcaloides d'ergot presentant une biodisponibilité ameliorée et compositions ainsi obtenues
US6696491B2 (en)	2000-05-12	2004-02-24	Meracol Corporation Limited	Treating irritable bowel syndrome or disease
NZ504526A (en) *	2000-05-12	2003-05-30	Meracol Corp Ltd	Treating herpes simplex symptoms using a mixture of cetyl myristate and cetyl palmitate
CA2408541C (fr) *	2000-05-12	2009-07-28	Meracol Corporation Limited	Traitement contre l'eczema et/ou le psoriasis
US20030153620A1 (en)	2000-05-12	2003-08-14	Meakin Timothy David	Treating eczema and/or psoriasis
WO2003026640A1 (fr) *	2001-09-28	2003-04-03	Meracol Corporation Limited	Traitement d'allergies alimentaires et/ou d'intolerances alimentaires
CN111297815B (zh) *	2020-04-29	2022-04-15	宝利化（南京）制药有限公司	一种甲磺酸二氢麦角碱缓释片及其制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3147187A (en) *	1962-09-10	1964-09-01	Don Hall Lab	Sustained release pharmaceutical
CH630257A5 (en) *	1975-03-17	1982-06-15	Hoffmann La Roche	Sustained release formulation
DE3124983A1 (de) *	1981-06-25	1983-01-20	Meditest Inst Fuer Medizinisch	Arzneiformen zur oralen verabreichung
CH649300A5 (de) *	1981-08-07	1985-05-15	Sandoz Ag	Ergopeptinderivate, ihre herstellung und verwendung.
US4369172A (en) *	1981-12-18	1983-01-18	Forest Laboratories Inc.	Prolonged release therapeutic compositions based on hydroxypropylmethylcellulose
DE3303616A1 (de) *	1982-02-12	1983-08-25	Sandoz-Patent-GmbH, 7850 Lörrach	Mutterkornalkaloide, verfahren zu deren herstellung sowie diese verbindungen enthaltende pharmazeutische zubereitungen
US4421736A (en) *	1982-05-20	1983-12-20	Merrel Dow Pharmaceuticals Inc.	Sustained release diethylpropion compositions
JPS604120A (ja) *	1983-06-22	1985-01-10	Shionogi & Co Ltd	作用持続型ピナシジル製剤
GB2154874B (en) *	1984-02-29	1987-11-04	Sandoz Ltd	Bromoscriptine compositions
GB8413795D0 (en) *	1984-05-30	1984-07-04	Sandoz Ltd	Organic compounds

1986
- 1986-01-24 HU HU86361A patent/HU195729B/hu not_active IP Right Cessation
- 1986-01-24 NL NL8600161A patent/NL8600161A/nl not_active Application Discontinuation
- 1986-01-27 CH CH296/86A patent/CH667592A5/de not_active IP Right Cessation
- 1986-01-29 DE DE19863602577 patent/DE3602577A1/de not_active Ceased
- 1986-01-31 FR FR868601477A patent/FR2576787B1/fr not_active Expired - Lifetime
- 1986-02-03 BE BE1/011431A patent/BE904152A/fr not_active IP Right Cessation
- 1986-02-03 GR GR860310A patent/GR860310B/el unknown
- 1986-02-03 AU AU52942/86A patent/AU597570B2/en not_active Ceased
- 1986-02-03 IE IE29186A patent/IE59293B1/en not_active IP Right Cessation
- 1986-02-03 GB GB08602602A patent/GB2170407B/en not_active Expired
- 1986-02-03 CA CA000501011A patent/CA1263087A/fr not_active Expired
- 1986-02-03 DK DK052086A patent/DK167138B1/da not_active IP Right Cessation
- 1986-02-03 PT PT81954A patent/PT81954B/pt not_active IP Right Cessation
- 1986-02-03 NZ NZ215020A patent/NZ215020A/xx unknown
- 1986-02-03 KR KR1019860000698A patent/KR920010388B1/ko not_active Expired
- 1986-02-04 PH PH33379A patent/PH23384A/en unknown
- 1986-02-04 ES ES551635A patent/ES8800040A1/es not_active Expired
- 1986-02-04 LU LU86289A patent/LU86289A1/fr unknown
- 1986-02-04 JP JP61023666A patent/JPS61183225A/ja active Pending
- 1986-02-04 SE SE8600496A patent/SE8600496L/ not_active Application Discontinuation
- 1986-02-05 IT IT47620/86A patent/IT1191255B/it active
1991
- 1991-07-16 SG SG561/91A patent/SG56191G/en unknown
- 1991-07-25 HK HK571/91A patent/HK57191A/xx unknown
1992
- 1992-04-03 CY CY1604A patent/CY1604A/en unknown

Also Published As

Publication number	Publication date
GB2170407A (en)	1986-08-06
FR2576787A1 (fr)	1986-08-08
CA1263087A (fr)	1989-11-21
PT81954A (en)	1986-03-01
DK167138B1 (da)	1993-09-06
IT8647620A0 (it)	1986-02-05
JPS61183225A (ja)	1986-08-15
DK52086D0 (da)	1986-02-03
GR860310B (en)	1986-05-27
IE860291L (en)	1986-08-05
ES551635A0 (es)	1987-10-16
NL8600161A (nl)	1986-09-01
SE8600496L (sv)	1986-08-06
IT1191255B (it)	1988-02-24
HU195729B (en)	1988-07-28
BE904152A (fr)	1986-08-04
PH23384A (en)	1989-07-26
IE59293B1 (en)	1994-02-09
PT81954B (pt)	1988-07-01
ES8800040A1 (es)	1987-10-16
KR860006265A (ko)	1986-09-09
HK57191A (en)	1991-08-02
AU5294286A (en)	1986-08-14
DK52086A (da)	1986-08-06
KR920010388B1 (ko)	1992-11-27
HUT41984A (en)	1987-06-29
SG56191G (en)	1991-08-23
FR2576787B1 (fr)	1990-01-12
DE3602577A1 (de)	1986-08-28
LU86289A1 (fr)	1986-09-02
NZ215020A (en)	1989-07-27
CH667592A5 (de)	1988-10-31
GB2170407B (en)	1988-10-26
AU597570B2 (en)	1990-06-07
SE8600496D0 (sv)	1986-02-04
GB8602602D0 (en)	1986-03-12

Publication	Publication Date	Title
JPH08504201A (ja)	1996-05-07	抗うつ作用を有する医薬組成物としての２‐アミノ‐６‐ｎ‐プロピル‐アミノ‐４，５，６，７‐テトラヒドロベンゾチアゾールの使用
NZ220769A (en)	1990-12-21	Compositions of ketotifen (4-(1-methyl-4-piperidylidene)- 4h-benzo(4,5)cyclohepta(1,2-b)thiophen-10-9(h)-one)
CY1604A (en)	1992-04-03	Pharmaceutical 9,10-dihydro ergot alkaloid containing compositions
CY1564A (en)	1991-05-17	Bromocriptine compositions
US5069911A (en)	1991-12-03	Pharmaceutical 9,10-dihydrogenated ergot alkaloid containing compositions
UA65652C2 (uk)	2004-04-15	Таблетка з регульованим вивільненням бетагістину та спосіб її виготовлення
CY1622A (en)	1992-07-10	Pharmaceutical formulations with controlled release of the active substance
AU756338B2 (en)	2003-01-09	Stabile compositions comprising levosimendan and alginic acid
CA1256374A (fr)	1989-06-27	Composes de bromocriptine
DK170016B1 (da)	1995-05-01	Præparat med kontrolleret afgivelse af det aktive stof
US4105796A (en)	1978-08-08	Pharmaceutical compositions containing racemic or optically active 1-(2,6-dimethyl-phenoxy)-2-methylamino-propane and method of use
AU598751B2 (en)	1990-07-05	Pharmaceutical formulations with controlled release of the active substance
US4152435A (en)	1979-05-01	Compositions and methods to treat hypertension comprising a pyridazine and N-amidino-2-(2,6-dichlorophenyl) acetamide
KR20160025946A (ko)	2016-03-09	N-desalkylquetiapine을 활성성분으로 포함하는 서방성 약제학적 조성물
AT388101B (de)	1989-05-10	Verfahren zur herstellung einer pharmazeutischen zusammensetzung zur oralen verabreichung mit kontrollierter wirkstofffreisetzung
JPH0827000A (ja)	1996-01-30	悪阻による諸症状の予防または治療薬
JPH0827001A (ja)	1996-01-30	術後嘔吐の予防または治療薬
HK1031998B (en)	2003-07-11	Stable compositions comprising levosimendan and alginic acid