DD263775A5 - Verfahren zur herstellung ungesaettigter aminosaeuren - Google Patents

Verfahren zur herstellung ungesaettigter aminosaeuren Download PDF

Info

Publication number: DD263775A5
Authority: DD; German Democratic Republic
Prior art keywords: amino; hydroxy; hydrogen; formula; alkyl
Prior art date: 1986-02-13

Application number

DD87299843A

Other languages

German (de)

English (en)

Inventor

Christof Angst

Derek E Brundish

John G Dingwall

Graham E Fagg

Original Assignee

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Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-02-13

Filing date

1987-02-11

Publication date

1989-01-11

1987-02-11 Application filed by ��@��@��k�� filed Critical ��@��@��k��

1989-01-11 Publication of DD263775A5 publication Critical patent/DD263775A5/de

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
- C07F9/3826—Acyclic unsaturated acids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
- C07F9/302—Acyclic unsaturated acids
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
- C07F9/32—Esters thereof
- C07F9/3205—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
- C07F9/3217—Esters of acyclic unsaturated acids
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/40—Esters thereof
- C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
- C07F9/4015—Esters of acyclic unsaturated acids

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Molecular Biology (AREA)
Biochemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Neurology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Neurosurgery (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Biomedical Technology (AREA)
Cardiology (AREA)
Urology & Nephrology (AREA)
Heart & Thoracic Surgery (AREA)
Psychiatry (AREA)
Anesthesiology (AREA)
Pain & Pain Management (AREA)
Vascular Medicine (AREA)
Hospice & Palliative Care (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Saccharide Compounds (AREA)
Pyrrole Compounds (AREA)
Compounds Of Unknown Constitution (AREA)
Medicines Containing Material From Animals Or Micro-Organisms (AREA)

DD87299843A 1986-02-13 1987-02-11 Verfahren zur herstellung ungesaettigter aminosaeuren DD263775A5 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
CH57886		1986-02-13

Publications (1)

Publication Number	Publication Date
DD263775A5 true DD263775A5 (de)	1989-01-11

Family

ID=4190244

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DD87299843A DD263775A5 (de)	1986-02-13	1987-02-11	Verfahren zur herstellung ungesaettigter aminosaeuren

Country Status (23)

Country	Link
EP (1)	EP0233154B1 (da)
JP (2)	JPH0717665B2 (da)
KR (1)	KR900003533B1 (da)
AT (1)	ATE70535T1 (da)
AU (1)	AU610493B2 (da)
CA (1)	CA1331625C (da)
CY (1)	CY1821A (da)
DD (1)	DD263775A5 (da)
DE (1)	DE3775229D1 (da)
DK (1)	DK169341B1 (da)
ES (1)	ES2038690T3 (da)
FI (1)	FI85144C (da)
GR (1)	GR3003526T3 (da)
HK (1)	HK95594A (da)
HU (1)	HU204532B (da)
IE (1)	IE59417B1 (da)
IL (1)	IL81543A0 (da)
NO (1)	NO170938C (da)
NZ (1)	NZ219255A (da)
PH (1)	PH23762A (da)
PT (1)	PT84270B (da)
SG (1)	SG92294G (da)
ZA (1)	ZA871022B (da)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5175344A (en) *	1986-02-13	1992-12-29	Ciba-Geigy Corporation	Unsaturated amino acids
PT85874B (pt) *	1986-10-09	1990-07-31	Ciba Geigy Ag	Processo para a preparacao de oligo-peptidos com accao antibiotica
PH27591A (en) *	1987-08-04	1993-08-31	Ciba Geigy Ag	A process for the manufacture of novel unsaturated amino acid compound
US5175153A (en) *	1987-11-30	1992-12-29	Warner-Lambert Company	Substituted alpha-amino acids having pharmaceutical activity
US5179085A (en) *	1989-03-15	1993-01-12	Warner-Lambert Company	N-substituted α-amino acids and derivatives thereof having pharmaceutical activity
ATE112282T1 (de) *	1989-04-07	1994-10-15	Ciba Geigy Ag	Ungesättigte aminodicarbonsäurederivate.
US5500419A (en) *	1989-09-19	1996-03-19	Merrell Dow Pharmaceuticals Inc.	NMDA antagonists
DK0420806T3 (da) *	1989-09-26	1995-10-16	Ciba Geigy Ag	Phosphonsyrer, fremgangsmåde til deres fremstilling og deres anvendelse som lægemiddel
US5294734A (en) *	1989-09-26	1994-03-15	Ciba-Geigy Corp.	4-substituted 2-aminoalk-3-enoic acids
US5488140A (en) *	1989-09-26	1996-01-30	Ciba-Geigy Corporation	4-substituted 2-aminoalk-3-enoic
US5238958A (en) *	1990-02-26	1993-08-24	Warner-Lambert Company	Substituted α-amino acids having selected acidic moieties for use as excitatory amino acid antagonists in pharmaceuticals
JPH07505908A (ja) *	1992-09-28	1995-06-29	マックセチーニ、マリア　ルイザ	Ｎｍｄａ受容体のアロステリックモジュレーター
US20090170813A1 (en) *	2005-10-18	2009-07-02	Francine Acher	Hypophosphorous Acid Derivatives and their Therapeutical Applications
DE102007032669A1 (de) *	2007-07-13	2009-01-15	Clariant International Limited	Alkylphosphonigsäuren, -salze und -ester, Verfahren zu deren Herstellung und ihre Verwendung

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4477391A (en) *	1981-08-14	1984-10-16	Collins James F	Amino acid isomers, their production and their medicinal use
GB2104079B (en) *	1981-08-14	1985-08-21	London Polytech	New aminoacid isomers, their production and their medicinal use

1987
- 1987-02-10 AT AT87810080T patent/ATE70535T1/de not_active IP Right Cessation
- 1987-02-10 ES ES198787810080T patent/ES2038690T3/es not_active Expired - Lifetime
- 1987-02-10 DE DE8787810080T patent/DE3775229D1/de not_active Expired - Lifetime
- 1987-02-10 EP EP87810080A patent/EP0233154B1/de not_active Expired - Lifetime
- 1987-02-11 PT PT84270A patent/PT84270B/pt not_active IP Right Cessation
- 1987-02-11 KR KR1019870001107A patent/KR900003533B1/ko not_active Expired
- 1987-02-11 DD DD87299843A patent/DD263775A5/de not_active IP Right Cessation
- 1987-02-11 FI FI870558A patent/FI85144C/fi not_active IP Right Cessation
- 1987-02-11 CA CA000529448A patent/CA1331625C/en not_active Expired - Fee Related
- 1987-02-11 IL IL81543A patent/IL81543A0/xx not_active IP Right Cessation
- 1987-02-12 IE IE36587A patent/IE59417B1/en not_active IP Right Cessation
- 1987-02-12 ZA ZA871022A patent/ZA871022B/xx unknown
- 1987-02-12 JP JP62028375A patent/JPH0717665B2/ja not_active Expired - Lifetime
- 1987-02-12 DK DK070787A patent/DK169341B1/da not_active IP Right Cessation
- 1987-02-12 HU HU87554A patent/HU204532B/hu not_active IP Right Cessation
- 1987-02-12 NZ NZ219255A patent/NZ219255A/xx unknown
- 1987-02-12 AU AU68726/87A patent/AU610493B2/en not_active Ceased
- 1987-02-13 PH PH34860A patent/PH23762A/en unknown
- 1987-02-13 NO NO870577A patent/NO170938C/no unknown
1992
- 1992-01-08 GR GR910402040T patent/GR3003526T3/el unknown
1994
- 1994-07-11 SG SG92294A patent/SG92294G/en unknown
- 1994-09-01 JP JP6208837A patent/JP2509465B2/ja not_active Expired - Lifetime
- 1994-09-08 HK HK95594A patent/HK95594A/xx not_active IP Right Cessation
1995
- 1995-10-20 CY CY182195A patent/CY1821A/xx unknown

Also Published As

Publication number	Publication date
JPS62246586A (ja)	1987-10-27
EP0233154B1 (de)	1991-12-18
AU610493B2 (en)	1991-05-23
ZA871022B (en)	1987-09-30
HK95594A (en)	1994-09-16
FI85144B (fi)	1991-11-29
NO170938C (no)	1992-12-30
DK169341B1 (da)	1994-10-10
ES2038690T3 (es)	1993-08-01
KR870007942A (ko)	1987-09-23
KR900003533B1 (ko)	1990-05-21
DE3775229D1 (de)	1992-01-30
HU204532B (en)	1992-01-28
NO870577L (no)	1987-08-14
EP0233154A3 (en)	1989-06-14
PH23762A (en)	1989-11-03
IL81543A0 (en)	1987-09-16
DK70787D0 (da)	1987-02-12
CY1821A (en)	1995-10-20
NO170938B (no)	1992-09-21
FI85144C (fi)	1992-03-10
PT84270B (pt)	1989-09-14
ATE70535T1 (de)	1992-01-15
HUT43863A (en)	1987-12-28
DK70787A (da)	1987-08-14
NZ219255A (en)	1989-08-29
PT84270A (en)	1987-03-01
IE59417B1 (en)	1994-02-23
JP2509465B2 (ja)	1996-06-19
FI870558A0 (fi)	1987-02-11
GR3003526T3 (da)	1993-03-16
CA1331625C (en)	1994-08-23
JPH07206683A (ja)	1995-08-08
AU6872687A (en)	1987-08-20
NO870577D0 (no)	1987-02-13
JPH0717665B2 (ja)	1995-03-01
SG92294G (en)	1995-04-28
FI870558A7 (fi)	1987-08-14
EP0233154A2 (de)	1987-08-19
IE870365L (en)	1987-08-13

Legal Events

Date	Code	Title	Description
1996-05-09	ENJ	Ceased due to non-payment of renewal fee

Publication	Publication Date	Title
DE3889638T2 (de)	1994-09-15	Substituierte Propanphosphinsäure-Verbindungen.
EP0463560B1 (de)	1995-10-25	Neuartige Antiepileptika
DD263775A5 (de)	1989-01-11	Verfahren zur herstellung ungesaettigter aminosaeuren
DE2942781A1 (de)	1980-04-30	Phosphinylalkanoylproline, verfahren zu ihrer herstellung und ihre verwendung als hypotensive wirkstoffe
CH637952A5 (de)	1983-08-31	Verfahren zur herstellung von allylcarbonsaeuren.
DE69018514T2 (de)	1995-09-21	Substituierte Aminoalkylphosphinsäure.
EP0371921B1 (de)	1994-06-08	Phenylaliphatylaminoalkandi-phosphonsäuren
DD282016A5 (de)	1990-08-29	Verfahren zur herstellung neuer ungesaettigter aminosaeureverbindungen
US5051413A (en)	1991-09-24	Unsaturated amino acids
EP0391850B1 (de)	1994-09-28	Ungesättigte Aminodicarbonsäurederivate
US5489717A (en)	1996-02-06	Glutamate (NMDA) receptor antagonists
EP0420806B1 (de)	1995-07-05	Phosphonsäure, Verfahren zur Herstellung und Verwendung als Arzneimittelwirkstoff
DD294945A5 (de)	1991-10-17	Verfahren zur herstellung von p-substituierten propanphosphinsaeureverbindungen
DE69310524T2 (de)	1997-12-04	Phosphono substituierte tetrazol-derivate
US5175344A (en)	1992-12-29	Unsaturated amino acids
EP0703919B1 (de)	1998-09-02	Phosphonobernsteinsäurederivate und ihre verwendung als arzneimittel
EP0213080A2 (de)	1987-03-04	Hydropyridin-Derivate
DE4211536A1 (de)	1993-10-07	Verfahren zur Herstellung von Derivaten der Bis(aminomethyl)phosphinsäure
DE2918160B2 (de)	1981-05-27	Verfahren zur Herstellung von 1.2-Diphosphonobernsteinsäureestern
WO1998022481A1 (de)	1998-05-28	Arylsubstituierte aminoacylierte phosphonsäuren und deren halbester
SI8811501A (sl)	1996-10-31	Postopek za pripravo novih nenasičenih spojin amino kislin
DE4329533A1 (de)	1995-03-09	Dibenzyl-N,N-dialkylphosphorigsäureamide als Phosphorylierungsreagenzien sowie ein Verfahren zu ihrer Herstellung
DE2011092A1 (de)	1970-09-17	Herstellung von Phosphonsäuren
EP0538689A1 (de)	1993-04-28	Neue substituierte 2,3-Dihydropyrane, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel