DE10351663A1 - Pulverförmige Arzneimittel enthaltend ein Tiotropiumsalz und Salmeterolxinafoat - Google Patents

Pulverförmige Arzneimittel enthaltend ein Tiotropiumsalz und Salmeterolxinafoat Download PDF

Info

Publication number: DE10351663A1
Authority: DE; Germany
Prior art keywords: inhalation; powder; tiotropium; salmeterol; salmeterol xinafoate
Prior art date: 2002-12-20
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Withdrawn

Application number

DE10351663A

Other languages

German (de)

English (en)

Inventor

Hagen Graebner

Mareke Hartig

Peter Sieger

Rainer Soyka

Michael Trunk

Michael Walz

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Boehringer Ingelheim Pharma GmbH and Co KG

Boehringer Ingelheim Pharmaceuticals Inc

Original Assignee

Boehringer Ingelheim Pharma GmbH and Co KG

Boehringer Ingelheim Pharmaceuticals Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-12-20

Filing date

2003-11-05

Publication date

2004-07-01

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32404034&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE10351663(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2003-11-05 Application filed by Boehringer Ingelheim Pharma GmbH and Co KG, Boehringer Ingelheim Pharmaceuticals Inc filed Critical Boehringer Ingelheim Pharma GmbH and Co KG

2003-11-05 Priority to DE10351663A priority Critical patent/DE10351663A1/de

2004-07-01 Publication of DE10351663A1 publication Critical patent/DE10351663A1/de

Status Withdrawn legal-status Critical Current

Links

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Classifications

- A—HUMAN NECESSITIES
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- A61K9/00—Medicinal preparations characterised by special physical form
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/205—Amine addition salts of organic acids; Inner quaternary ammonium salts, e.g. betaine, carnitine
- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics

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Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Pulmonology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Emergency Medicine (AREA)
General Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Otolaryngology (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

DE10351663A 2002-12-20 2003-11-05 Pulverförmige Arzneimittel enthaltend ein Tiotropiumsalz und Salmeterolxinafoat Withdrawn DE10351663A1 (de)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
DE10351663A DE10351663A1 (de)	2002-12-20	2003-11-05	Pulverförmige Arzneimittel enthaltend ein Tiotropiumsalz und Salmeterolxinafoat

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
DE10259912.2		2002-12-20
DE10259912		2002-12-20
DE10351663A DE10351663A1 (de)	2002-12-20	2003-11-05	Pulverförmige Arzneimittel enthaltend ein Tiotropiumsalz und Salmeterolxinafoat

Publications (1)

Publication Number	Publication Date
DE10351663A1 true DE10351663A1 (de)	2004-07-01

Family

ID=32404034

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DE10351663A Withdrawn DE10351663A1 (de)	2002-12-20	2003-11-05	Pulverförmige Arzneimittel enthaltend ein Tiotropiumsalz und Salmeterolxinafoat

Country Status (21)

Country	Link
EP (1)	EP1581198A1 (es)
JP (1)	JP2006516135A (es)
KR (1)	KR20050086930A (es)
CN (1)	CN1728988B (es)
AU (1)	AU2003288226B2 (es)
BR (1)	BR0317443A (es)
CA (1)	CA2510779A1 (es)
DE (1)	DE10351663A1 (es)
EA (1)	EA010588B1 (es)
EC (1)	ECSP055855A (es)
FR (1)	FR2848849B1 (es)
HR (1)	HRP20050570A2 (es)
IT (1)	ITMI20032473A1 (es)
MX (1)	MXPA05006519A (es)
NO (1)	NO20053548L (es)
NZ (1)	NZ541303A (es)
PL (1)	PL376231A1 (es)
RS (1)	RS20050484A (es)
UA (1)	UA83813C2 (es)
WO (1)	WO2004058233A1 (es)
ZA (1)	ZA200503692B (es)

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PE20091730A1 (es)	2008-04-03	2009-12-10	Boehringer Ingelheim Int	Formulaciones que comprenden un inhibidor de dpp4
BRPI0916997A2 (pt)	2008-08-06	2020-12-15	Boehringer Ingelheim International Gmbh	Inibidor de dpp-4 e seu uso
UY32030A (es)	2008-08-06	2010-03-26	Boehringer Ingelheim Int	"tratamiento para diabetes en pacientes inapropiados para terapia con metformina"
US20200155558A1 (en)	2018-11-20	2020-05-21	Boehringer Ingelheim International Gmbh	Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug
CN102256976A (zh)	2008-12-23	2011-11-23	贝林格尔.英格海姆国际有限公司	有机化合物的盐形式
AR074990A1 (es)	2009-01-07	2011-03-02	Boehringer Ingelheim Int	Tratamiento de diabetes en pacientes con un control glucemico inadecuado a pesar de la terapia con metformina
KR20240090632A (ko)	2009-11-27	2024-06-21	베링거 인겔하임 인터내셔날 게엠베하	리나글립틴과 같은 ｄｐｐ－ｉｖ 억제제를 사용한 유전자형 검사된 당뇨병 환자의 치료
CN102946875A (zh)	2010-05-05	2013-02-27	贝林格尔.英格海姆国际有限公司	组合疗法
WO2011161161A1 (en)	2010-06-24	2011-12-29	Boehringer Ingelheim International Gmbh	Diabetes therapy
AR083878A1 (es)	2010-11-15	2013-03-27	Boehringer Ingelheim Int	Terapia antidiabetica vasoprotectora y cardioprotectora, linagliptina, metodo de tratamiento
US8883800B2 (en)	2011-07-15	2014-11-11	Boehringer Ingelheim International Gmbh	Substituted quinazolines, the preparation thereof and the use thereof in pharmaceutical compositions
US9555001B2 (en)	2012-03-07	2017-01-31	Boehringer Ingelheim International Gmbh	Pharmaceutical composition and uses thereof
JP6218811B2 (ja)	2012-05-14	2017-10-25	ベーリンガーインゲルハイムインターナショナルゲゼルシャフトミットベシュレンクテルハフツング	Ｓｉｒｓ及び／又は敗血症の治療に用いるｄｐｐ−４阻害薬としてのキサンチン誘導体
JP6224084B2 (ja)	2012-05-14	2017-11-01	ベーリンガーインゲルハイムインターナショナルゲゼルシャフトミットベシュレンクテルハフツング	糸球体上皮細胞関連障害及び／又はネフローゼ症候群の治療に用いるｄｐｐ−４阻害薬としてのキサンチン誘導体
WO2013174767A1 (en)	2012-05-24	2013-11-28	Boehringer Ingelheim International Gmbh	A xanthine derivative as dpp -4 inhibitor for use in modifying food intake and regulating food preference
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KR101748796B1 (ko) *	2015-09-30	2017-06-19	한미약품 주식회사	활성성분의 전달량이 향상된 흡입용 캡슐제
CN109310697A (zh)	2016-06-10	2019-02-05	勃林格殷格翰国际有限公司	利格列汀和二甲双胍的组合
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2003
- 2003-04-12 UA UAA200507088A patent/UA83813C2/ru unknown
- 2003-11-05 DE DE10351663A patent/DE10351663A1/de not_active Withdrawn
- 2003-12-04 RS YUP-2005/0484A patent/RS20050484A/sr unknown
- 2003-12-04 CN CN2003801069216A patent/CN1728988B/zh not_active Expired - Fee Related
- 2003-12-04 KR KR1020057011668A patent/KR20050086930A/ko not_active Ceased
- 2003-12-04 BR BR0317443-3A patent/BR0317443A/pt not_active IP Right Cessation
- 2003-12-04 HR HR20050570A patent/HRP20050570A2/xx not_active Application Discontinuation
- 2003-12-04 WO PCT/EP2003/013691 patent/WO2004058233A1/de not_active Ceased
- 2003-12-04 JP JP2004562686A patent/JP2006516135A/ja active Pending
- 2003-12-04 PL PL03376231A patent/PL376231A1/xx not_active Application Discontinuation
- 2003-12-04 EA EA200500902A patent/EA010588B1/ru not_active IP Right Cessation
- 2003-12-04 NZ NZ541303A patent/NZ541303A/en unknown
- 2003-12-04 EP EP03780120A patent/EP1581198A1/de not_active Withdrawn
- 2003-12-04 CA CA002510779A patent/CA2510779A1/en not_active Abandoned
- 2003-12-04 AU AU2003288226A patent/AU2003288226B2/en not_active Ceased
- 2003-12-04 MX MXPA05006519A patent/MXPA05006519A/es unknown
- 2003-12-16 IT IT002473A patent/ITMI20032473A1/it unknown
- 2003-12-19 FR FR0315082A patent/FR2848849B1/fr not_active Expired - Fee Related
2005
- 2005-05-09 ZA ZA200503692A patent/ZA200503692B/en unknown
- 2005-06-15 EC EC2005005855A patent/ECSP055855A/es unknown
- 2005-07-19 NO NO20053548A patent/NO20053548L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
AU2003288226A1 (en)	2004-07-22
AU2003288226B2 (en)	2010-01-07
KR20050086930A (ko)	2005-08-30
CN1728988A (zh)	2006-02-01
ECSP055855A (es)	2005-11-22
PL376231A1 (en)	2005-12-27
CA2510779A1 (en)	2004-07-15
BR0317443A (pt)	2005-11-16
ITMI20032473A1 (it)	2004-06-21
UA83813C2 (ru)	2008-08-26
HRP20050570A2 (en)	2006-07-31
MXPA05006519A (es)	2005-08-26
EP1581198A1 (de)	2005-10-05
EA010588B1 (ru)	2008-10-30
NZ541303A (en)	2008-11-28
WO2004058233A1 (de)	2004-07-15
JP2006516135A (ja)	2006-06-22
CN1728988B (zh)	2010-04-28
EA200500902A1 (ru)	2006-02-24
ZA200503692B (en)	2006-10-25
FR2848849A1 (fr)	2004-06-25
NO20053548L (no)	2005-09-02
RS20050484A (sr)	2007-11-15
FR2848849B1 (fr)	2007-01-05

Legal Events

Date	Code	Title	Description
2011-02-03	8141	Disposal/no request for examination

Publication	Publication Date	Title
DE10351663A1 (de)	2004-07-01	Pulverförmige Arzneimittel enthaltend ein Tiotropiumsalz und Salmeterolxinafoat
EP1379220B1 (de)	2004-12-29	Inhalationskapseln
WO2002030389A1 (de)	2002-04-18	Neue tiotropium-haltige inhalationspulver
EP2182933B1 (de)	2016-09-07	Neue pulverförmige arzneimittel enthaltend tiotropium und salmeterol sowie laktose als hilfsstoff
EP1785422B1 (de)	2016-11-16	Kristallines Mikronisat des Tiotropiumbromids
EP1326585B1 (de)	2006-03-08	Verfahren zur herstellung von pulverformulierungen
EP1283036B1 (de)	2008-01-02	Multidosis-Trockenpulverinhalator mit Pulverreservoir
DE10141377A1 (de)	2003-03-13	Aufstreuverfahren zur Herstellung von Pulverformulierungen
EP1424996B1 (de)	2005-04-27	Verfahren zur herstellung von inhalationspulvern
EP1567135B1 (de)	2008-07-23	Tiotropiumhaltige pulverformulierung für die inhalation
DE60308497T2 (de)	2007-02-22	Pulverzubereitungen zur inhalation
EP2298415B1 (de)	2013-06-12	Tiotropiumbromid-Mikronisat
EP1646365B1 (de)	2009-01-14	Pulverformulierungen für die inhalation enthaltend ein neues anticholinergikum
DE10338407A1 (de)	2005-03-17	Neue Inhalationspulver enthaltend den CGRP-Antagonisten 1-[N2-[3,5-Dibrom-N-[[4-(3,4-dihydro-2(1H)-oxochinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)-piperazin
DE10138022A1 (de)	2003-02-20	Verfahren zur Herstellung von Pulverformulierungen