DK0572425T3 - Imidazopyridin-PAF/H1-antagonister - Google Patents

Imidazopyridin-PAF/H1-antagonister

Info

Publication number
DK0572425T3
DK0572425T3 DK92902889.2T DK92902889T DK0572425T3 DK 0572425 T3 DK0572425 T3 DK 0572425T3 DK 92902889 T DK92902889 T DK 92902889T DK 0572425 T3 DK0572425 T3 DK 0572425T3
Authority
DK
Denmark
Prior art keywords
pct
paf
antagonists
sec
imidazopyridine
Prior art date
Application number
DK92902889.2T
Other languages
English (en)
Inventor
David Alker
Robert John Bass
Kelvin Cooper
Original Assignee
Pfizer
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer, Pfizer Ltd filed Critical Pfizer
Application granted granted Critical
Publication of DK0572425T3 publication Critical patent/DK0572425T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cosmetics (AREA)
  • Prostheses (AREA)
  • Steroid Compounds (AREA)
DK92902889.2T 1991-02-13 1992-01-24 Imidazopyridin-PAF/H1-antagonister DK0572425T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB919102997A GB9102997D0 (en) 1991-02-13 1991-02-13 Therapeutic agents

Publications (1)

Publication Number Publication Date
DK0572425T3 true DK0572425T3 (da) 1994-09-12

Family

ID=10689943

Family Applications (1)

Application Number Title Priority Date Filing Date
DK92902889.2T DK0572425T3 (da) 1991-02-13 1992-01-24 Imidazopyridin-PAF/H1-antagonister

Country Status (29)

Country Link
US (1) US5358953A (da)
EP (1) EP0572425B1 (da)
JP (1) JP2506541B2 (da)
KR (1) KR970005302B1 (da)
CN (1) CN1040326C (da)
AT (1) ATE109482T1 (da)
AU (1) AU650322B2 (da)
BR (1) BR9205615A (da)
CA (1) CA2099381C (da)
CZ (1) CZ280504B6 (da)
DE (1) DE69200304T2 (da)
DK (1) DK0572425T3 (da)
EG (1) EG20085A (da)
ES (1) ES2059212T3 (da)
FI (1) FI933531A7 (da)
GB (1) GB9102997D0 (da)
HU (2) HUT65947A (da)
IE (1) IE65125B1 (da)
IL (1) IL100887A (da)
MX (1) MX9200589A (da)
MY (1) MY108437A (da)
NO (1) NO300592B1 (da)
NZ (1) NZ241597A (da)
PL (1) PL169304B1 (da)
RU (1) RU2114845C1 (da)
TW (1) TW227000B (da)
WO (1) WO1992014734A1 (da)
YU (1) YU48238B (da)
ZA (1) ZA921005B (da)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2042421B1 (es) * 1992-05-22 1994-08-01 Uriach & Cia Sa J Procedimiento para la obtencion de la 8-cloro-11-*1-*(5-metil-3-piridil)metil*-4-piperidiliden*-6,11-dihidro-5h-benzo*5,6*ciclohepta*1,2-b*piridina.
US5753671A (en) * 1994-08-10 1998-05-19 British Biotech Pharmaceuticals Limited Imidazopyridine derivatives as dual histamine (H1) and platelet activating factor (PAF) antagonists
ES2087038B1 (es) * 1994-11-07 1997-03-16 Uriach & Cia Sa J Nuevas piperidinas con actividad antagonista del paf.
US5567711A (en) * 1995-04-19 1996-10-22 Abbott Laboratories Indole-3-carbonyl and indole-3-sulfonyl derivatives as platelet activating factor antagonists
GB9508748D0 (en) * 1995-04-28 1995-06-14 British Biotech Pharm Benzimidazole derivatives
AU698487B2 (en) * 1995-08-05 1998-10-29 British Biotech Pharmaceuticals Limited Imidazopyridine derivatives
SE9801526D0 (sv) * 1998-04-29 1998-04-29 Astra Ab New compounds
CA2774959C (en) 2000-08-04 2016-05-31 Dmi Biosciences, Inc. Method of using diketopiperazines and composition containing them
CN103191409A (zh) 2003-05-15 2013-07-10 Dmi生物科学公司 T-细胞介导的疾病的治疗
US7687515B2 (en) * 2006-01-17 2010-03-30 N.V. Organon 6-phenyl-1H-imidazo[4,5-c]pyridine-4-carbonitrile derivatives
AU2008349239B2 (en) 2008-01-30 2012-12-06 Nippon Zoki Pharmaceutical Co., Ltd. Piperidine derivative
US8217047B2 (en) 2008-05-27 2012-07-10 Dmi Acquisition Corp. Therapeutic methods and compounds
EP2727919B1 (en) * 2011-06-28 2019-05-08 Fujian Mindong Rejuvenation Pharmaceutical Co., Ltd. Benzocycloheptanethiophene derivatives for anti-allergic reactions
EP2765968A4 (en) 2011-10-10 2015-01-21 Ampio Pharmaceuticals Inc IMPLANTABLE MEDICINE PRODUCTS WITH INCREASED IMMUNO TOLERANCE AND PROCESSING AND IMPLANTATION METHODS
CA2846598C (en) 2011-10-10 2019-12-10 Ampio Pharmaceuticals, Inc. Treatment of degenerative joint disease
HK1198812A1 (en) * 2011-10-28 2015-06-12 Ampio Pharmaceuticals, Inc. Treatment of rhinitis
EA201500943A1 (ru) 2013-03-15 2016-08-31 Ампио Фармасьютикалс, Инк. Составы для мобилизации, хоуминга, размножения и дифференцировки стволовых клеток и способы применения составов
CA2958080A1 (en) 2014-08-18 2016-02-25 Ampio Pharmaceuticals, Inc. Treatment of joint conditions
US11389512B2 (en) 2015-06-22 2022-07-19 Ampio Pharmaceuticals, Inc. Use of low molecular weight fractions of human serum albumin in treating diseases
CN113880801A (zh) * 2020-07-03 2022-01-04 合肥医工医药股份有限公司 一类三环化合物、其制备方法及其医药用途

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL132137C (da) * 1963-04-24
EP0404797B1 (en) * 1988-03-15 1995-02-01 G.D. Searle & Co. 1H/3H-[4-(N,N-CYCLOALKYL AND/OR BRANCHED-ALKYLCARBOXAMIDO) -BENZYL]IMIDAZO[4,5-c]PYRIDINES AS PAF ANTAGONISTS
NZ228889A (en) * 1988-04-28 1991-09-25 Schering Corp Fused tri- or tetracyclic heterocyclic compounds and pharmaceutical compositions
US5250681A (en) * 1988-06-02 1993-10-05 Ajinomoto Co., Inc. Piperidine derivatives and hypotensives containing the same
US5114919A (en) * 1990-02-26 1992-05-19 Merck & Co., Inc. Adjuncts in cancer chemotherapy
BR9106433A (pt) * 1990-05-09 1993-05-04 Pfizer Imidazo (4,5-c) piridinas com atividade antagonista ao paf

Also Published As

Publication number Publication date
ZA921005B (en) 1993-08-12
ATE109482T1 (de) 1994-08-15
TW227000B (da) 1994-07-21
FI933531L (fi) 1993-08-10
HU211202A9 (en) 1995-11-28
DE69200304T2 (de) 1994-12-08
CN1064275A (zh) 1992-09-09
AU650322B2 (en) 1994-06-16
NO932889L (no) 1993-08-13
AU1168392A (en) 1992-09-15
YU14392A (sh) 1994-11-15
CS42592A3 (en) 1992-09-16
FI933531A0 (fi) 1993-08-10
HUT65947A (en) 1994-08-29
YU48238B (sh) 1997-08-22
HU9302327D0 (en) 1993-10-28
FI933531A7 (fi) 1993-08-10
JP2506541B2 (ja) 1996-06-12
EP0572425A1 (en) 1993-12-08
WO1992014734A1 (en) 1992-09-03
GB9102997D0 (en) 1991-03-27
IE920449A1 (en) 1992-08-12
NO300592B1 (no) 1997-06-23
NO932889D0 (no) 1993-08-13
NZ241597A (en) 1993-04-28
CN1040326C (zh) 1998-10-21
BR9205615A (pt) 1994-05-17
EP0572425B1 (en) 1994-08-03
IL100887A0 (en) 1992-11-15
CA2099381C (en) 1996-07-09
CA2099381A1 (en) 1992-08-14
RU2114845C1 (ru) 1998-07-10
EG20085A (en) 1997-05-31
PL169304B1 (pl) 1996-06-28
DE69200304D1 (de) 1994-09-08
IL100887A (en) 1996-01-19
MY108437A (en) 1996-09-30
US5358953A (en) 1994-10-25
JPH06504992A (ja) 1994-06-09
KR970005302B1 (ko) 1997-04-15
MX9200589A (es) 1992-10-01
CZ280504B6 (cs) 1996-02-14
IE65125B1 (en) 1995-10-04
ES2059212T3 (es) 1994-11-01

Similar Documents

Publication Publication Date Title
DK0572425T3 (da) Imidazopyridin-PAF/H1-antagonister
YU48426B (sh) Novi supstituisani pirazolilpirazoli, postupak njihovog dobijanja, medjuproizvodi za njihovo dobijanje i primena kao sredstava sa herbicidnim delovanjem
ES2162061T3 (es) Derivados de piperidina como antagonistas de la neuroquinina.
YU84791A (sh) Biciklicni 1-aza-cikloalkalni
UA26427A (uk) Похідhі ксаhтиhу у вигляді суміші ізомерів або іhдивідуальhих ізомерів, що мають властивість аhтагоhіста адеhозиhу
HRP941000B9 (hr) Morfolin i tiomorfolin antagonisti receptora tahikinina
RU93054165A (ru) Производные имидазопиридина, способ их получения, фармацевтическая композиция, способ лечения
CO4410319A1 (es) Derivados de fenetanolamina
FI922341A0 (fi) Piperidin- och pyrrolidinderivat.
MX9300312A (es) Antagonistas benzopiranicos y relacionado de ltb.
SG164268A1 (en) Quinolin-4-yl derivatives i
ATE64373T1 (de) Muscarin-rezeptor-antagonisten.
YU4393A (sr) Supstituisani heksahidroazepinoni i tetrahidrobenzazepinoni
ES2095995T3 (es) Procedimiento para la obtencion de 2,2-difluorbenzo(1,3)dioxol-carbaldehidos y nuevos productos intermedios.
MX9606654A (es) Derivados de alaquildiamina substituida y su uso como antagonistas de taquicinina.
DE69014903D1 (de) Disubstituierte piperidine und pyrrolidine als anticholinergische mittel.
FI973558L (fi) Menetelmä terapeuttisesti käytt¦kelpoisten 2-metyyli-imidatsoÄ4,5-cÜpyrid-1-yylijohdannaisten valmistamiseksi
DE3484375D1 (de) Pharmazeutische zusammenstellung fuer die prophylaxe oder behandlung von tierhaltungsketose.
PT100223A (pt) Processo para a preparacao de imidazopiridinas antagonistas de paf/h1
NO900646L (no) Fremgangsmaate for fremstilling av calsiumantagonister.
ES2084547B1 (es) Antagonistas benzopiranicos y relacionados de leucotrieno b4.
DE69001794D1 (de) Phenothiazinderivate, ihre herstellung und sie enthaltende pharmazeutische zusammensetzungen.
SE8301039D0 (sv) Heterocykliska derivat
ECSP003687A (es) Derivados 1 de quinolin-4- il
DK71084A (da) Nitromethylenderivat med pesticid virkning