DK0708105T3 - 5-HT4-receptoragonister - Google Patents

5-HT4-receptoragonister

Info

Publication number
DK0708105T3
DK0708105T3 DK95307480T DK95307480T DK0708105T3 DK 0708105 T3 DK0708105 T3 DK 0708105T3 DK 95307480 T DK95307480 T DK 95307480T DK 95307480 T DK95307480 T DK 95307480T DK 0708105 T3 DK0708105 T3 DK 0708105T3
Authority
DK
Denmark
Prior art keywords
receptor agonists
agonists
receptor
Prior art date
Application number
DK95307480T
Other languages
English (en)
Inventor
Hiroaki Satoh
Masashi Suzuki
Ruta Fukutomi
Masahiro Ueno
Koichiro Hagihara
Takeo Arai
Setsuko Mino
Yumiko Noguchi
Haruhiko Kikuchi
Original Assignee
Nisshin Flour Milling Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nisshin Flour Milling Co filed Critical Nisshin Flour Milling Co
Application granted granted Critical
Publication of DK0708105T3 publication Critical patent/DK0708105T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK95307480T 1994-10-20 1995-10-20 5-HT4-receptoragonister DK0708105T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP25490794 1994-10-20

Publications (1)

Publication Number Publication Date
DK0708105T3 true DK0708105T3 (da) 1999-08-23

Family

ID=17271511

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95307480T DK0708105T3 (da) 1994-10-20 1995-10-20 5-HT4-receptoragonister

Country Status (8)

Country Link
US (1) US5684003A (da)
EP (1) EP0708105B1 (da)
KR (1) KR960014128A (da)
CA (1) CA2160420A1 (da)
DE (1) DE69506826T2 (da)
DK (1) DK0708105T3 (da)
ES (1) ES2128668T3 (da)
TW (1) TW403747B (da)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69627323T2 (de) * 1995-05-31 2004-01-15 Nisshin Seifun Group Inc Indazolderivate mit einer cyclischen aminogruppe
US5914405A (en) * 1997-10-07 1999-06-22 Eli Lilly And Company Process for preparing 3-substituted indazoles
US6069152A (en) * 1997-10-07 2000-05-30 Eli Lilly And Company 5-HT4 agonists and antagonists
FR2792318B1 (fr) * 1999-04-16 2001-06-15 Synthelabo Derives d'indazole, leur preparation et leur application en therapeutique
US7671097B2 (en) * 2005-05-24 2010-03-02 Georgia-Pacific Chemicals Llc Stable phenolic resin polymer dispersions having low free aldehyde content
US7666867B2 (en) 2001-10-26 2010-02-23 University Of Connecticut Heteroindanes: a new class of potent cannabimimetic ligands
TW200533348A (en) * 2004-02-18 2005-10-16 Theravance Inc Indazole-carboxamide compounds as 5-ht4 receptor agonists
US7728006B2 (en) * 2004-04-07 2010-06-01 Theravance, Inc. Quinolinone-carboxamide compounds as 5-HT4 receptor agonists
TWI351282B (en) * 2004-04-07 2011-11-01 Theravance Inc Quinolinone-carboxamide compounds as 5-ht4 recepto
US8309575B2 (en) 2004-04-07 2012-11-13 Theravance, Inc. Quinolinone-carboxamide compounds as 5-HT4 receptor agonists
ATE441646T1 (de) * 2004-11-05 2009-09-15 Theravance Inc 5-ht4-rezeptoragonistenverbindungen
EP1807423B1 (en) * 2004-11-05 2009-05-20 Theravance, Inc. Quinolinone-carboxamide compounds
ATE469897T1 (de) * 2004-12-22 2010-06-15 Theravance Inc Indazolcarbonsäureamidverbindungen
NZ560828A (en) * 2005-03-02 2011-01-28 Theravance Inc Quinolinone compounds as 5-HT4 receptor agonists
JOP20130213B1 (ar) * 2012-07-17 2021-08-17 Takeda Pharmaceuticals Co معارضات لمستقبلht3-5
CA2962429C (en) 2014-09-29 2023-01-03 Takeda Pharmaceutical Company Limited Crystalline form of 1-(1-methyl-1h-pyrazol-4-yl)-n-((1r,5s,7s)-9-methyl-3-oxa-9-azabicyclo[3.3.1]nonan-7-yl)-1h-indole-3-carboxamide
GB201511382D0 (en) 2015-06-29 2015-08-12 Imp Innovations Ltd Novel compounds and their use in therapy
TW202412782A (zh) * 2022-05-25 2024-04-01 天主教魯汶大學 用於治療trpm3介導之病症的吲唑衍生物
WO2024052685A1 (en) 2022-09-09 2024-03-14 MyricX Pharma Limited Cytotoxic imidazo[1,2-a]pyridine compounds and their use in therapy

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8829079D0 (en) * 1988-12-13 1989-01-25 Beecham Group Plc Novel compounds
GB9009389D0 (en) * 1990-04-26 1990-06-20 Smith Kline French Lab Treatment
US5187166A (en) * 1990-07-31 1993-02-16 Nisshin Flour Milling Co., Ltd. Azabicyclo derivatives and their use as antiemetics
US5256656A (en) * 1990-07-31 1993-10-26 Nisshin Flour Milling Co., Ltd. Azabicyclo derivatives
TW251287B (da) * 1993-04-30 1995-07-11 Nissei Co Ltd

Also Published As

Publication number Publication date
DE69506826T2 (de) 1999-08-05
US5684003A (en) 1997-11-04
EP0708105B1 (en) 1998-12-23
KR960014128A (ko) 1996-05-22
TW403747B (en) 2000-09-01
EP0708105A1 (en) 1996-04-24
CA2160420A1 (en) 1996-04-21
ES2128668T3 (es) 1999-05-16
DE69506826D1 (de) 1999-02-04

Similar Documents

Publication Publication Date Title
DK0802910T3 (da) Estrogenagonister/antagonister
DK0708105T3 (da) 5-HT4-receptoragonister
EP0934305A4 (en) INTEGRINANTAGONISTS
FI964576A7 (fi) Uusia agonistiyhdisteitä
NO972016D0 (no) Indolyl-Y-reseptorantagonister
ID24836A (id) Agonis prostaglandin
DE69734833D1 (de) Vitronektin rezeptor antagonisten
EP0946164A4 (en) INTEGRIN ANTAGONISTS
NO961887D0 (no) -adrenergiske agonister
FI951249L (fi) Serotiinireseptoriaineita
EP0885205A4 (en) Fibrinogen Receptor Antagonists
DK0906294T3 (da) Benzoxazinon-dopamin D4-receptor-antagonister
ID17561A (id) Komposisi untuk pemakaian luar
TR199501389A2 (tr) Adesyon reseptörü antagonistleri (karsitlari).
FI974170L (fi) B-adrenergisiä agonisteja
NO985970L (no) Indolinderivater anvendelige som 5_HT-2C-reseptor-antagonister
BR9709521A (pt) "3-Cianoaril-pirazóis"
FI971492L (fi) Indolijohdannaiset 5-HT1-tyyppisinä agonisteina
MA23795A1 (fr) Derives d'indole substitues
DE69431672D1 (de) Adrenergischer rezeptor
NO973624L (no) Vasokonstriktive substituerte 2,3-dihydro-1,4-dioksinopiperidiner
FR2758444B1 (fr) Boucles d'oreille
BR9708948A (pt) 1,3 - Benzodioxois substituídos
FI972558A0 (fi) Uusi reseptori
GB9715018D0 (en) 3-Fluoro-4-aminopiperidine derivatives as 5-HT receptor agonists