DK0708105T3 - 5-HT4-receptoragonister - Google Patents
5-HT4-receptoragonisterInfo
- Publication number
- DK0708105T3 DK0708105T3 DK95307480T DK95307480T DK0708105T3 DK 0708105 T3 DK0708105 T3 DK 0708105T3 DK 95307480 T DK95307480 T DK 95307480T DK 95307480 T DK95307480 T DK 95307480T DK 0708105 T3 DK0708105 T3 DK 0708105T3
- Authority
- DK
- Denmark
- Prior art keywords
- receptor agonists
- agonists
- receptor
- Prior art date
Links
- 108091005482 5-HT4 receptors Proteins 0.000 title 1
- 239000000018 receptor agonist Substances 0.000 title 1
- 229940044601 receptor agonist Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/08—Bridged systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP25490794 | 1994-10-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK0708105T3 true DK0708105T3 (da) | 1999-08-23 |
Family
ID=17271511
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK95307480T DK0708105T3 (da) | 1994-10-20 | 1995-10-20 | 5-HT4-receptoragonister |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US5684003A (es) |
| EP (1) | EP0708105B1 (es) |
| KR (1) | KR960014128A (es) |
| CA (1) | CA2160420A1 (es) |
| DE (1) | DE69506826T2 (es) |
| DK (1) | DK0708105T3 (es) |
| ES (1) | ES2128668T3 (es) |
| TW (1) | TW403747B (es) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0829474B1 (en) * | 1995-05-31 | 2003-04-09 | Nisshin Seifun Group Inc. | Indazole derivatives having monocyclic amino group |
| US6069152A (en) * | 1997-10-07 | 2000-05-30 | Eli Lilly And Company | 5-HT4 agonists and antagonists |
| US5914405A (en) * | 1997-10-07 | 1999-06-22 | Eli Lilly And Company | Process for preparing 3-substituted indazoles |
| FR2792318B1 (fr) * | 1999-04-16 | 2001-06-15 | Synthelabo | Derives d'indazole, leur preparation et leur application en therapeutique |
| US7671097B2 (en) * | 2005-05-24 | 2010-03-02 | Georgia-Pacific Chemicals Llc | Stable phenolic resin polymer dispersions having low free aldehyde content |
| CA2464333C (en) | 2001-10-26 | 2011-07-26 | University Of Connecticut | Heteroindanes: a new class of potent cannabimimetic ligands |
| TW200533348A (en) * | 2004-02-18 | 2005-10-16 | Theravance Inc | Indazole-carboxamide compounds as 5-ht4 receptor agonists |
| TWI351282B (en) | 2004-04-07 | 2011-11-01 | Theravance Inc | Quinolinone-carboxamide compounds as 5-ht4 recepto |
| US7728006B2 (en) * | 2004-04-07 | 2010-06-01 | Theravance, Inc. | Quinolinone-carboxamide compounds as 5-HT4 receptor agonists |
| US8309575B2 (en) | 2004-04-07 | 2012-11-13 | Theravance, Inc. | Quinolinone-carboxamide compounds as 5-HT4 receptor agonists |
| WO2006052889A2 (en) * | 2004-11-05 | 2006-05-18 | Theravance, Inc. | Quinolinone-carboxamide compounds |
| US7399862B2 (en) * | 2004-11-05 | 2008-07-15 | Theravance, Inc. | 5-HT4 receptor agonist compounds |
| CA2588037A1 (en) * | 2004-12-22 | 2006-06-29 | Theravance, Inc. | Indazole-carboxamide compounds |
| CN101163701A (zh) * | 2005-03-02 | 2008-04-16 | 施万制药 | 作为5-ht4受体激动剂的喹啉酮化合物 |
| JOP20130213B1 (ar) | 2012-07-17 | 2021-08-17 | Takeda Pharmaceuticals Co | معارضات لمستقبلht3-5 |
| JP7055017B2 (ja) | 2014-09-29 | 2022-04-15 | 武田薬品工業株式会社 | 結晶形の1-(1-メチル-1h-ピラゾール-4-イル)-n-((1r,5s,7s)-9-メチル-3-オキサ-9-アザビシクロ[3.3.1]ノナン-7-イル)-1h-インドール-3-カルボキサミド |
| GB201511382D0 (en) | 2015-06-29 | 2015-08-12 | Imp Innovations Ltd | Novel compounds and their use in therapy |
| TW202412782A (zh) * | 2022-05-25 | 2024-04-01 | 天主教魯汶大學 | 用於治療trpm3介導之病症的吲唑衍生物 |
| JP2025530213A (ja) | 2022-09-09 | 2025-09-11 | ミリックス ファーマ リミテッド | Nmt阻害剤を含む抗体薬物コンジュゲート及びその使用 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8829079D0 (en) * | 1988-12-13 | 1989-01-25 | Beecham Group Plc | Novel compounds |
| GB9009389D0 (en) * | 1990-04-26 | 1990-06-20 | Smith Kline French Lab | Treatment |
| US5256656A (en) * | 1990-07-31 | 1993-10-26 | Nisshin Flour Milling Co., Ltd. | Azabicyclo derivatives |
| US5187166A (en) * | 1990-07-31 | 1993-02-16 | Nisshin Flour Milling Co., Ltd. | Azabicyclo derivatives and their use as antiemetics |
| TW251287B (es) * | 1993-04-30 | 1995-07-11 | Nissei Co Ltd |
-
1995
- 1995-10-12 CA CA002160420A patent/CA2160420A1/en not_active Abandoned
- 1995-10-12 US US08/543,853 patent/US5684003A/en not_active Expired - Lifetime
- 1995-10-20 DK DK95307480T patent/DK0708105T3/da active
- 1995-10-20 DE DE69506826T patent/DE69506826T2/de not_active Expired - Lifetime
- 1995-10-20 KR KR1019950036424A patent/KR960014128A/ko not_active Withdrawn
- 1995-10-20 TW TW084111089A patent/TW403747B/zh not_active IP Right Cessation
- 1995-10-20 EP EP95307480A patent/EP0708105B1/en not_active Expired - Lifetime
- 1995-10-20 ES ES95307480T patent/ES2128668T3/es not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| DE69506826T2 (de) | 1999-08-05 |
| DE69506826D1 (de) | 1999-02-04 |
| ES2128668T3 (es) | 1999-05-16 |
| CA2160420A1 (en) | 1996-04-21 |
| KR960014128A (ko) | 1996-05-22 |
| EP0708105A1 (en) | 1996-04-24 |
| EP0708105B1 (en) | 1998-12-23 |
| TW403747B (en) | 2000-09-01 |
| US5684003A (en) | 1997-11-04 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ATE214382T1 (de) | Östrogen-agonisten/antagonisten | |
| DK0708105T3 (da) | 5-HT4-receptoragonister | |
| FI964576A7 (fi) | Uusia agonistiyhdisteitä | |
| NO972016D0 (no) | Indolyl-Y-reseptorantagonister | |
| ID24836A (id) | Agonis prostaglandin | |
| DE69734833D1 (de) | Vitronektin rezeptor antagonisten | |
| EP0946164A4 (en) | INTEGRIN ANTAGONISTS | |
| NO961887D0 (no) | -adrenergiske agonister | |
| FI951249A7 (fi) | Serotiinireseptoriaineita | |
| EP0885205A4 (en) | Fibrinogen Receptor Antagonists | |
| DK0906294T3 (da) | Benzoxazinon-dopamin D4-receptor-antagonister | |
| ID17561A (id) | Komposisi untuk pemakaian luar | |
| TR199501389A2 (tr) | Adesyon reseptörü antagonistleri (karsitlari). | |
| FI974170A7 (fi) | B-adrenergisiä agonisteja | |
| NO985970L (no) | Indolinderivater anvendelige som 5_HT-2C-reseptor-antagonister | |
| BR9709521A (pt) | "3-Cianoaril-pirazóis" | |
| MA23795A1 (fr) | Derives d'indole substitues | |
| DE69431672D1 (de) | Adrenergischer rezeptor | |
| NO973624L (no) | Vasokonstriktive substituerte 2,3-dihydro-1,4-dioksinopiperidiner | |
| FR2758444B1 (fr) | Boucles d'oreille | |
| NO972771D0 (no) | Ny reseptor | |
| BR9708948A (pt) | 1,3 - Benzodioxois substituídos | |
| GB9715018D0 (en) | 3-Fluoro-4-aminopiperidine derivatives as 5-HT receptor agonists | |
| KR960012039U (ko) | 모니터용 서류고정대 | |
| NO303314B1 (no) | Uthaler for fiskeliner |