DK0739344T3 - Antiparasitiske pyrrolobenzoxazinforbindelser - Google Patents

Antiparasitiske pyrrolobenzoxazinforbindelser

Info

Publication number
DK0739344T3
DK0739344T3 DK95905762T DK95905762T DK0739344T3 DK 0739344 T3 DK0739344 T3 DK 0739344T3 DK 95905762 T DK95905762 T DK 95905762T DK 95905762 T DK95905762 T DK 95905762T DK 0739344 T3 DK0739344 T3 DK 0739344T3
Authority
DK
Denmark
Prior art keywords
pct
formula
antiparasitic
compounds
sec
Prior art date
Application number
DK95905762T
Other languages
Danish (da)
English (en)
Inventor
Yasuhiro Kojima
Yuji Yamauchi
Nakao Kojima
Bernard F Bishop
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of DK0739344T3 publication Critical patent/DK0739344T3/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12NMICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
    • C12N1/00Microorganisms; Compositions thereof; Processes of propagating, maintaining or preserving microorganisms or compositions thereof; Processes of preparing or isolating a composition containing a microorganism; Culture media therefor
    • C12N1/14Fungi; Culture media therefor
    • C12N1/145Fungi isolates
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P17/00Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms
    • C12P17/18Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms containing at least two hetero rings condensed among themselves or condensed with a common carbocyclic ring system, e.g. rifamycin
    • C12P17/188Heterocyclic compound containing in the condensed system at least one hetero ring having nitrogen atoms and oxygen atoms as the only ring heteroatoms
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12RINDEXING SCHEME ASSOCIATED WITH SUBCLASSES C12C - C12Q, RELATING TO MICROORGANISMS
    • C12R2001/00Microorganisms ; Processes using microorganisms
    • C12R2001/645Fungi ; Processes using fungi
    • C12R2001/66Aspergillus

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Genetics & Genomics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Engineering & Computer Science (AREA)
  • Microbiology (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Botany (AREA)
  • Mycology (AREA)
  • Virology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
DK95905762T 1994-01-14 1995-01-11 Antiparasitiske pyrrolobenzoxazinforbindelser DK0739344T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP1582594 1994-01-14
PCT/JP1995/000025 WO1995019363A1 (fr) 1994-01-14 1995-01-11 COMPOSéS ANTIPARASITAIRES A BASE DE PYRROLOBENZOXAZINE

Publications (1)

Publication Number Publication Date
DK0739344T3 true DK0739344T3 (da) 1999-07-26

Family

ID=11899636

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95905762T DK0739344T3 (da) 1994-01-14 1995-01-11 Antiparasitiske pyrrolobenzoxazinforbindelser

Country Status (11)

Country Link
US (1) US5801023A (fr)
EP (1) EP0739344B1 (fr)
JP (1) JP2767161B2 (fr)
AT (1) ATE173264T1 (fr)
AU (1) AU684334B2 (fr)
CA (1) CA2181168C (fr)
DE (1) DE69505946T2 (fr)
DK (1) DK0739344T3 (fr)
ES (1) ES2123948T3 (fr)
NZ (1) NZ278143A (fr)
WO (1) WO1995019363A1 (fr)

Families Citing this family (162)

* Cited by examiner, † Cited by third party
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GB0303439D0 (en) * 2003-02-14 2003-03-19 Pfizer Ltd Antiparasitic terpene alkaloids
TWI487486B (zh) 2009-12-01 2015-06-11 Syngenta Participations Ag 以異唑啉衍生物為主之殺蟲化合物
BR112012020521B1 (pt) 2010-02-17 2017-12-26 Syngenta Participations Ag Derivative compounds of isoxazoline, its intermediaries and method for controlling insects, mites, nematodes, or molluscs
EA201201171A1 (ru) 2010-02-22 2013-03-29 Зингента Партисипейшнс Аг Дигидрофурановые производные в качестве инсектицидных соединений
AU2011220041A1 (en) 2010-02-25 2012-08-23 Syngenta Limited Process for the preparation of isoxazoline derivatives
CN103153949A (zh) 2010-10-05 2013-06-12 先正达参股股份有限公司 杀虫的吡咯烷-基-芳基-甲酰胺
WO2012049327A2 (fr) 2010-10-15 2012-04-19 Syngenta Participations Ag Mélanges pesticides
EP2643302A1 (fr) 2010-11-23 2013-10-02 Syngenta Participations AG Composés insecticides
CN103261188A (zh) 2010-12-17 2013-08-21 先正达参股股份有限公司 杀虫化合物
BR112013020213A2 (pt) 2011-02-09 2016-08-02 Syngenta Participations Ag compostos inseticidas
EP2688864A1 (fr) 2011-03-22 2014-01-29 Syngenta Participations AG Composés insecticides
WO2012156400A1 (fr) 2011-05-18 2012-11-22 Syngenta Participations Ag Composés insecticides à base de dérivés d'arylthiacétamide
WO2012163948A1 (fr) 2011-05-31 2012-12-06 Syngenta Participations Ag Mélanges pesticides comprenant des dérivés d'isoxazoline
TW201311677A (zh) 2011-05-31 2013-03-16 Syngenta Participations Ag 殺蟲化合物
WO2012175474A1 (fr) 2011-06-20 2012-12-27 Syngenta Participations Ag Pesticides à base de 1,2,3-triazole
US20140343049A1 (en) 2011-08-22 2014-11-20 Syngenta Participations Ag Dihydrofuran derivatives as insecticidal compounds
EP2748137A1 (fr) 2011-08-22 2014-07-02 Syngenta Participations AG Dérivés de dihydrofurane en tant que composés insecticides
WO2013026695A1 (fr) 2011-08-25 2013-02-28 Syngenta Participations Ag Dérivés d'isoxazoline en tant que composés insecticides
US9204648B2 (en) 2011-08-25 2015-12-08 Syngenta Participations Ag Process for the preparation of thietane derivatives
KR20140054302A (ko) 2011-08-25 2014-05-08 신젠타 파티서페이션즈 아게 살곤충 화합물로서의 이속사졸린 유도체
WO2013026929A1 (fr) 2011-08-25 2013-02-28 Syngenta Participations Ag Dérivés de dihydropyrrole en tant que composés insecticides
US9307766B2 (en) 2011-08-25 2016-04-12 Syngenta Participations Ag Isoxazoline derivatives as insecticidal compounds
EP2755969B1 (fr) 2011-09-13 2017-01-18 Syngenta Participations AG Dérivés d'isothiazoline en tant que composés insecticides
WO2013050261A1 (fr) 2011-10-03 2013-04-11 Syngenta Participations Ag Dérivés de 2-méthoxybenzamide insecticides
JP2014534182A (ja) 2011-10-03 2014-12-18 シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト 殺虫化合物としてのイソオキサゾリン誘導体
WO2013135674A1 (fr) 2012-03-12 2013-09-19 Syngenta Participations Ag Composés de 2-aryl-acétamide insecticides
WO2014001120A1 (fr) 2012-06-25 2014-01-03 Syngenta Participations Ag Dérivés d'isothiazole en tant que composés insecticides
WO2014001121A1 (fr) 2012-06-25 2014-01-03 Syngenta Participations Ag Dérivés d'isothiazole en tant que composés insecticides
CA2888041A1 (fr) 2012-10-31 2014-05-08 Syngenta Participations Ag Composes insecticides
WO2014079935A1 (fr) 2012-11-21 2014-05-30 Syngenta Participations Ag Composés insecticides à base de dérivés d'arylthioacétamide
BR112015025028B1 (pt) 2013-04-02 2020-10-13 Syngenta Participations Ag compostos, processo para a produção de compostos, métodos para controle de insetos, ácaros, nematódeos ou moluscos e para proteção de plantas úteis e composição
CN113336699A (zh) 2013-04-02 2021-09-03 先正达参股股份有限公司 杀虫化合物
WO2015007451A1 (fr) 2013-07-15 2015-01-22 Syngenta Participations Ag Dérivés hétérobicycliques microbiocides
EP3556744B1 (fr) 2013-12-23 2022-06-01 Syngenta Participations AG Composés insecticides
WO2016087593A1 (fr) 2014-12-05 2016-06-09 Syngenta Participations Ag Nouvelles quinolinylamidines fongicides
JP6662901B2 (ja) 2015-03-27 2020-03-11 シンジェンタ パーティシペーションズ アーゲー 殺微生物性二環式複素環式誘導体
WO2016155831A1 (fr) 2015-04-02 2016-10-06 Syngenta Participations Ag Dérivés d'isoxazoline-styrène utilisés comme composés insecticides
SI3356358T1 (sl) 2015-10-02 2020-09-30 Syngenta Participations Ag Mikrobiocidni derivati oksadiazola
US20180319753A1 (en) 2015-10-28 2018-11-08 Syngenta Participations Ag Microbiocidal oxadiazole derivatives
JP2018538362A (ja) 2015-11-04 2018-12-27 シンジェンタ パーティシペーションズ アーゲー 殺微生物アニリド誘導体
MX2018006474A (es) 2015-12-02 2018-08-01 Syngenta Participations Ag Derivados de oxadiazol microbicidas.
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US20190292174A1 (en) 2016-03-15 2019-09-26 Syngenta Participations Ag Microbiocidal oxadiazole derivatives
WO2017162868A1 (fr) 2016-03-24 2017-09-28 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
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BR112018070785B1 (pt) 2016-04-12 2023-01-10 Syngenta Participations Ag Compostos derivados de oxadiazol microbiocidas, composição agroquímica, método de controle ou prevenção de infestação de plantas úteis por microrganismos fitopatogênicos e uso dos referidos compostos
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BR112019000942B1 (pt) 2016-07-22 2022-11-08 Syngenta Participations Ag Composto compreendendo derivados de oxadiazol e seu uso, composição agroquímica e método para controlar ou prevenir a infestação de plantas úteis por micro-organismos fitopatogênicos
BR112019001229B1 (pt) 2016-07-22 2022-11-16 Syngenta Participations Ag Composto derivado de oxadiazol, composição agroquímica compreendendo o mesmo, método para controlar ou impedir infestação de plantas úteis por microrganismos fitopatogênicos e uso do referido composto como fungicida
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WO2018029242A1 (fr) 2016-08-11 2018-02-15 Syngenta Participations Ag Dérivés d'oxadiazole microbicides
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WO2018184988A1 (fr) 2017-04-05 2018-10-11 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
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JP2026502124A (ja) 2022-12-19 2026-01-21 シンジェンタ クロップ プロテクション アクチェンゲゼルシャフト 殺微生物性ピリダジンジヒドロオキサジアジン誘導体
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WO2025078263A1 (fr) 2023-10-11 2025-04-17 Syngenta Crop Protection Ag Dérivés de pyridyl pyrazole microbiocides
WO2025104152A1 (fr) 2023-11-15 2025-05-22 Syngenta Crop Protection Ag Dérivés de tétrahydroisoquinoléine microbiocides
WO2025114167A1 (fr) 2023-11-28 2025-06-05 Syngenta Crop Protection Ag Dérivés de pyrazole microbiocides
PY24108853A (es) 2023-12-08 2025-10-06 Syngenta Crop Protection Ag Polimorfos
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* Cited by examiner, † Cited by third party
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GB8917064D0 (en) * 1989-07-26 1989-09-13 Pfizer Ltd Antiparasitic agent
GB2240100A (en) * 1990-01-17 1991-07-24 Pfizer Ltd Anti-parasitic compound

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EP0739344A1 (fr) 1996-10-30
CA2181168C (fr) 2000-05-09
JPH09500909A (ja) 1997-01-28
ATE173264T1 (de) 1998-11-15
JP2767161B2 (ja) 1998-06-18
EP0739344B1 (fr) 1998-11-11
ES2123948T3 (es) 1999-01-16
WO1995019363A1 (fr) 1995-07-20
NZ278143A (en) 1997-11-24
CA2181168A1 (fr) 1995-07-20
AU1424895A (en) 1995-08-01
DE69505946T2 (de) 1999-04-15
US5801023A (en) 1998-09-01
DE69505946D1 (de) 1998-12-17
AU684334B2 (en) 1997-12-11

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