DK0781282T3 - [1,2]triazolo[4,3-a]quinoxalinonderivater, deres fremstilling og anvendelse - Google Patents

[1,2]triazolo[4,3-a]quinoxalinonderivater, deres fremstilling og anvendelse

Info

Publication number
DK0781282T3
DK0781282T3 DK95930410T DK95930410T DK0781282T3 DK 0781282 T3 DK0781282 T3 DK 0781282T3 DK 95930410 T DK95930410 T DK 95930410T DK 95930410 T DK95930410 T DK 95930410T DK 0781282 T3 DK0781282 T3 DK 0781282T3
Authority
DK
Denmark
Prior art keywords
alkyl
triazolo
independently
preparation
pox
Prior art date
Application number
DK95930410T
Other languages
English (en)
Inventor
Flemming Elmelund Nielsen
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Application granted granted Critical
Publication of DK0781282T3 publication Critical patent/DK0781282T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Hospice & Palliative Care (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Otolaryngology (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK95930410T 1994-09-16 1995-09-12 [1,2]triazolo[4,3-a]quinoxalinonderivater, deres fremstilling og anvendelse DK0781282T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK106694 1994-09-16
PCT/DK1995/000365 WO1996008493A1 (en) 1994-09-16 1995-09-12 [1,2,4]TRIAZOLO[4,3-a]QUINOXALINONE DERIVATIVES, THEIR PREPARATION AND USE

Publications (1)

Publication Number Publication Date
DK0781282T3 true DK0781282T3 (da) 2000-02-28

Family

ID=8100607

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95930410T DK0781282T3 (da) 1994-09-16 1995-09-12 [1,2]triazolo[4,3-a]quinoxalinonderivater, deres fremstilling og anvendelse

Country Status (22)

Country Link
EP (1) EP0781282B1 (da)
JP (1) JPH10506620A (da)
KR (1) KR970706285A (da)
CN (1) CN1193973A (da)
AT (1) ATE183186T1 (da)
AU (1) AU694554B2 (da)
CA (1) CA2200056A1 (da)
CZ (1) CZ284930B6 (da)
DE (1) DE69511420T2 (da)
DK (1) DK0781282T3 (da)
ES (1) ES2138233T3 (da)
FI (1) FI971076A7 (da)
GR (1) GR3031788T3 (da)
HU (1) HUT76802A (da)
IL (1) IL115299A0 (da)
NO (1) NO308797B1 (da)
NZ (1) NZ292108A (da)
PL (1) PL319175A1 (da)
SK (1) SK282457B6 (da)
TW (1) TW397835B (da)
WO (1) WO1996008493A1 (da)
ZA (1) ZA957794B (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL125950A0 (en) * 1997-09-05 1999-04-11 Pfizer Prod Inc Methods of administering ampa receptor antagonists to treat dyskinesias associated with dopamine agonist therapy
CN1285834A (zh) 1997-11-11 2001-02-28 小野药品工业株式会社 稠合吡嗪化合物
WO2010101230A1 (ja) 2009-03-05 2010-09-10 アステラス製薬株式会社 キノキサリン化合物
BR112013005439A2 (pt) 2010-09-07 2017-09-19 Astellas Pharma Inc compostos de quinoxalina

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4354027A (en) * 1980-05-19 1982-10-12 Usv Pharmaceutical Corporation Triazoloquinoxalin-4-ones
US5153196A (en) * 1991-06-05 1992-10-06 Eli Lilly And Company Excitatory amino acid receptor antagonists and methods for the use thereof
DK162491D0 (da) * 1991-09-20 1991-09-20 Novo Nordisk As Heterocycliske forbindelser, deres fremstilling og farmaceutiske praeparater indeholdende forbindelserne
AU3767793A (en) * 1992-04-03 1993-11-08 Yamanouchi Pharmaceutical Co., Ltd. Fused quinoxalinone derivative and pharmaceutical composition containing the same
DK31093D0 (da) * 1993-03-19 1993-03-19 Novo Nordisk As
WO1994026746A1 (en) * 1993-05-06 1994-11-24 Novo Nordisk A/S [1,2,4]TRIAZOLO[4,3-a]QUINOXALINE COMPOUNDS, THEIR PREPARATION AND USE

Also Published As

Publication number Publication date
CA2200056A1 (en) 1996-03-21
KR970706285A (ko) 1997-11-03
CN1193973A (zh) 1998-09-23
FI971076L (fi) 1997-05-13
DE69511420T2 (de) 2000-03-30
NO308797B1 (no) 2000-10-30
FI971076A0 (fi) 1997-03-14
CZ75397A3 (en) 1997-08-13
GR3031788T3 (en) 2000-02-29
ZA957794B (en) 1996-05-14
SK33497A3 (en) 1998-02-04
TW397835B (en) 2000-07-11
NZ292108A (en) 1999-02-25
AU694554B2 (en) 1998-07-23
EP0781282A1 (en) 1997-07-02
NO971187L (no) 1997-05-15
ES2138233T3 (es) 2000-01-01
IL115299A0 (en) 1995-12-31
CZ284930B6 (cs) 1999-04-14
AU3380895A (en) 1996-03-29
JPH10506620A (ja) 1998-06-30
PL319175A1 (en) 1997-08-04
HUT76802A (en) 1997-11-28
ATE183186T1 (de) 1999-08-15
NO971187D0 (no) 1997-03-14
DE69511420D1 (de) 1999-09-16
EP0781282B1 (en) 1999-08-11
SK282457B6 (sk) 2002-02-05
FI971076A7 (fi) 1997-05-13
WO1996008493A1 (en) 1996-03-21

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