DK0929525T3 - Heteroaryloxyethylaminer som ligander af 5-HT1A-receptor - Google Patents
Heteroaryloxyethylaminer som ligander af 5-HT1A-receptorInfo
- Publication number
- DK0929525T3 DK0929525T3 DK97943000T DK97943000T DK0929525T3 DK 0929525 T3 DK0929525 T3 DK 0929525T3 DK 97943000 T DK97943000 T DK 97943000T DK 97943000 T DK97943000 T DK 97943000T DK 0929525 T3 DK0929525 T3 DK 0929525T3
- Authority
- DK
- Denmark
- Prior art keywords
- heteroberloxyethylamines
- ligands
- ht1a receptor
- ht1a
- receptor
- Prior art date
Links
- 102100022738 5-hydroxytryptamine receptor 1A Human genes 0.000 title 1
- 101710138638 5-hydroxytryptamine receptor 1A Proteins 0.000 title 1
- 239000003446 ligand Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C07D215/24—Oxygen atoms attached in position 8
- C07D215/26—Alcohols; Ethers thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C07D215/24—Oxygen atoms attached in position 8
- C07D215/26—Alcohols; Ethers thereof
- C07D215/28—Alcohols; Ethers thereof with halogen atoms or nitro radicals in positions 5, 6 or 7
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Otolaryngology (AREA)
- Hospice & Palliative Care (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Quinoline Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9611798A FR2753968B1 (fr) | 1996-09-27 | 1996-09-27 | Nouvelles heteroaryloxyethylamines, leur procede de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant |
| PCT/FR1997/001691 WO1998013349A2 (fr) | 1996-09-27 | 1997-09-26 | Heteroaryloxyethylamines en tant que ligands 5-ht¿1a? |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK0929525T3 true DK0929525T3 (da) | 2002-12-02 |
Family
ID=9496126
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK97943000T DK0929525T3 (da) | 1996-09-27 | 1997-09-26 | Heteroaryloxyethylaminer som ligander af 5-HT1A-receptor |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US6063784A (de) |
| EP (1) | EP0929525B1 (de) |
| JP (1) | JP2001503393A (de) |
| AR (1) | AR008486A1 (de) |
| AT (1) | ATE223380T1 (de) |
| AU (1) | AU731459B2 (de) |
| BR (1) | BR9711560A (de) |
| CA (1) | CA2267247C (de) |
| DE (1) | DE69715223T2 (de) |
| DK (1) | DK0929525T3 (de) |
| ES (1) | ES2182120T3 (de) |
| FR (1) | FR2753968B1 (de) |
| HU (1) | HUP0001189A3 (de) |
| IL (1) | IL128917A (de) |
| MY (1) | MY118992A (de) |
| NO (1) | NO311935B1 (de) |
| NZ (1) | NZ334623A (de) |
| PL (1) | PL190221B1 (de) |
| RU (1) | RU2176639C2 (de) |
| TW (1) | TW425390B (de) |
| WO (1) | WO1998013349A2 (de) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4507398B2 (ja) * | 1999-12-06 | 2010-07-21 | 宇部興産株式会社 | 3−ハロメチルオキセタン化合物の合成方法 |
| US20040147581A1 (en) * | 2002-11-18 | 2004-07-29 | Pharmacia Corporation | Method of using a Cox-2 inhibitor and a 5-HT1A receptor modulator as a combination therapy |
| RU2234315C1 (ru) * | 2003-06-30 | 2004-08-20 | Государственный научный центр - Институт биофизики | Фармацевтическая композиция, содержащая ондансетрон, метацин и бензамид |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1989003681A1 (en) * | 1987-10-19 | 1989-05-05 | Pfizer Inc. | Substituted tetralins, chromans and related compounds in the treatment of asthma |
| DK203990D0 (da) * | 1990-08-24 | 1990-08-24 | Novo Nordisk As | Piperazinylderivater |
| MX9201991A (es) * | 1991-05-02 | 1992-11-01 | Jonh Wyeth & Brother Limited | Derivados de piperazina y procedimiento para su preparacion. |
| US5240800A (en) * | 1991-07-29 | 1993-08-31 | Eastman Kodak Company | Near-infrared radiation sensitive photoelectrographic master and imaging method |
| EP0643045B1 (de) * | 1993-09-10 | 2000-03-08 | Novartis AG | Chinolin-Verbindungen als Leukotriene Antagonisten |
| GB9507288D0 (en) * | 1995-04-07 | 1995-05-31 | Sod Conseils Rech Applic | Phenoxyethylamine derivatives with high affinity for 5-HT1A receptors |
-
1996
- 1996-09-27 FR FR9611798A patent/FR2753968B1/fr not_active Expired - Fee Related
-
1997
- 1997-09-24 AR ARP970104385A patent/AR008486A1/es unknown
- 1997-09-25 MY MYPI97004469A patent/MY118992A/en unknown
- 1997-09-26 CA CA002267247A patent/CA2267247C/fr not_active Expired - Fee Related
- 1997-09-26 US US09/254,787 patent/US6063784A/en not_active Expired - Fee Related
- 1997-09-26 DK DK97943000T patent/DK0929525T3/da active
- 1997-09-26 NZ NZ334623A patent/NZ334623A/en unknown
- 1997-09-26 DE DE69715223T patent/DE69715223T2/de not_active Expired - Lifetime
- 1997-09-26 TW TW086114116A patent/TW425390B/zh not_active IP Right Cessation
- 1997-09-26 ES ES97943000T patent/ES2182120T3/es not_active Expired - Lifetime
- 1997-09-26 EP EP97943000A patent/EP0929525B1/de not_active Expired - Lifetime
- 1997-09-26 RU RU99108674/04A patent/RU2176639C2/ru not_active IP Right Cessation
- 1997-09-26 JP JP51535198A patent/JP2001503393A/ja not_active Withdrawn
- 1997-09-26 WO PCT/FR1997/001691 patent/WO1998013349A2/fr not_active Ceased
- 1997-09-26 BR BR9711560A patent/BR9711560A/pt active Search and Examination
- 1997-09-26 PL PL97332480A patent/PL190221B1/pl not_active IP Right Cessation
- 1997-09-26 HU HU0001189A patent/HUP0001189A3/hu unknown
- 1997-09-26 AT AT97943000T patent/ATE223380T1/de not_active IP Right Cessation
- 1997-09-26 IL IL12891797A patent/IL128917A/xx not_active IP Right Cessation
- 1997-09-26 AU AU44637/97A patent/AU731459B2/en not_active Ceased
-
1999
- 1999-03-26 NO NO19991481A patent/NO311935B1/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES2182120T3 (es) | 2003-03-01 |
| FR2753968A1 (fr) | 1998-04-03 |
| PL190221B1 (pl) | 2005-11-30 |
| WO1998013349A3 (fr) | 1998-11-05 |
| CA2267247A1 (fr) | 1998-04-02 |
| AU731459B2 (en) | 2001-03-29 |
| EP0929525A2 (de) | 1999-07-21 |
| IL128917A (en) | 2003-10-31 |
| NO991481D0 (no) | 1999-03-26 |
| RU2176639C2 (ru) | 2001-12-10 |
| AU4463797A (en) | 1998-04-17 |
| IL128917A0 (en) | 2000-02-17 |
| NO991481L (no) | 1999-03-26 |
| DE69715223T2 (de) | 2003-04-30 |
| ATE223380T1 (de) | 2002-09-15 |
| EP0929525B1 (de) | 2002-09-04 |
| TW425390B (en) | 2001-03-11 |
| FR2753968B1 (fr) | 1998-11-27 |
| JP2001503393A (ja) | 2001-03-13 |
| PL332480A1 (en) | 1999-09-13 |
| AR008486A1 (es) | 2000-01-19 |
| WO1998013349A2 (fr) | 1998-04-02 |
| CA2267247C (fr) | 2009-05-05 |
| MY118992A (en) | 2005-02-28 |
| BR9711560A (pt) | 1999-08-24 |
| DE69715223D1 (de) | 2002-10-10 |
| HUP0001189A3 (en) | 2001-12-28 |
| US6063784A (en) | 2000-05-16 |
| NZ334623A (en) | 1999-09-29 |
| NO311935B1 (no) | 2002-02-18 |
| HUP0001189A2 (hu) | 2000-10-28 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK0908449T3 (da) | Fremstilling af carotenoider | |
| IS5354A (is) | Ný efnasambönd | |
| DK1032566T3 (da) | Fremgangsmåde til fremstilling af citalopram | |
| IS5430A (is) | Ný samsetning | |
| DK0937055T3 (da) | Fremgangsmåde til fremstilling af d,I-alfa-tocopherol | |
| DK1073416T3 (da) | Anvendelse af NO som anti-inflammatorisk middel | |
| DK0975623T3 (da) | Indazolamidforbindelser som sertoninerge midler | |
| EE9800430A (et) | Uued ühendid | |
| DK0911311T3 (da) | Fremstilling af lycopenmetabolitter | |
| DK0996642T3 (da) | Fremgangsmåde til fremstilling af heparin | |
| DK0970939T3 (da) | Fremgangsmåde til fremstilling af methanol | |
| NO994106D0 (no) | Oksazolidiner som 5-HT2A-antagonister | |
| DK0864564T3 (da) | Særlig fremgangsmåde til fremstillingen af alfa-bromlactamderivater | |
| FI970727A0 (fi) | Foerfarande och anordning foer torkning av objekt som innehaoller vatten | |
| DK0929525T3 (da) | Heteroaryloxyethylaminer som ligander af 5-HT1A-receptor | |
| DK0810216T3 (da) | Derivater af 10,11-dihydro-10-oxo-5H-dibenz/b/,f/azepin-5-carboxamid | |
| DK1012152T3 (da) | Fremgangsmåde til fremstilling af oxazaphosphorin-2-aminer | |
| NO983656D0 (no) | Heterocyklyl-ergolinderivater som 5-HT1A reseptorligander | |
| DK0915076T3 (da) | Fremgangsmåde til fremstilling af trans-(R,R)-actinol | |
| DK0927163T3 (da) | Fremstilling af 1-butyl-4-piperidinylmethylamin | |
| FI980053A0 (fi) | Anordning foer utformande av fiberbollar av laongstraeckta fibrer som foeljer med enluftstroem | |
| DK0921111T3 (da) | Fremgangsmåde til fremstilling af substituerede anthraquinoner | |
| DK1051401T3 (da) | Fremgangsmåde til fremstilling af formylimidazoler | |
| DE69827603D1 (de) | Synchrondemodulator | |
| DK0857720T3 (da) | Fremgangsmåde til syntese af desoxypyridinolin |