DK1017384T3 - Azabenzimidazolbaserede forbindelser til modulation af serin/threoninproteinkinasefunktion - Google Patents

Azabenzimidazolbaserede forbindelser til modulation af serin/threoninproteinkinasefunktion

Info

Publication number
DK1017384T3
DK1017384T3 DK98949464T DK98949464T DK1017384T3 DK 1017384 T3 DK1017384 T3 DK 1017384T3 DK 98949464 T DK98949464 T DK 98949464T DK 98949464 T DK98949464 T DK 98949464T DK 1017384 T3 DK1017384 T3 DK 1017384T3
Authority
DK
Denmark
Prior art keywords
azabenzimidazole
protein kinase
based compounds
threonine protein
kinase function
Prior art date
Application number
DK98949464T
Other languages
Danish (da)
English (en)
Inventor
Gerald Mcmahon
Bernhard Kutscher
Heinz Weinberger
Harald App
Original Assignee
Zentaris Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zentaris Gmbh filed Critical Zentaris Gmbh
Application granted granted Critical
Publication of DK1017384T3 publication Critical patent/DK1017384T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK98949464T 1997-09-26 1998-09-23 Azabenzimidazolbaserede forbindelser til modulation af serin/threoninproteinkinasefunktion DK1017384T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US6014597P 1997-09-26 1997-09-26
EP98949464A EP1017384B1 (fr) 1997-09-26 1998-09-23 Composes a base d'azabenzimidazole destines a la modulation d'une fonction de proteine kinase de serine/threonine
PCT/US1998/019973 WO1999016438A1 (fr) 1997-09-26 1998-09-23 Composes a base d'azabenzimidazole destines a la modulation d'une fonction de proteine kinase de serine/threonine

Publications (1)

Publication Number Publication Date
DK1017384T3 true DK1017384T3 (da) 2005-01-31

Family

ID=22027657

Family Applications (1)

Application Number Title Priority Date Filing Date
DK98949464T DK1017384T3 (da) 1997-09-26 1998-09-23 Azabenzimidazolbaserede forbindelser til modulation af serin/threoninproteinkinasefunktion

Country Status (27)

Country Link
US (2) US6093728A (fr)
EP (1) EP1017384B1 (fr)
JP (1) JP2001517699A (fr)
KR (1) KR100547929B1 (fr)
CN (1) CN1167420C (fr)
AR (1) AR017266A1 (fr)
AT (1) ATE281834T1 (fr)
AU (1) AU748849B2 (fr)
BG (1) BG64784B1 (fr)
BR (1) BR9812682A (fr)
CA (1) CA2305370C (fr)
DE (1) DE69827516T2 (fr)
DK (1) DK1017384T3 (fr)
ES (1) ES2230719T3 (fr)
HU (1) HUP0004024A3 (fr)
IL (4) IL158649A0 (fr)
NO (1) NO325663B1 (fr)
NZ (2) NZ503432A (fr)
PL (1) PL191618B1 (fr)
PT (1) PT1017384E (fr)
RU (1) RU2230553C2 (fr)
SK (1) SK285357B6 (fr)
TR (1) TR200001546T2 (fr)
TW (1) TW581815B (fr)
UA (1) UA72448C2 (fr)
WO (1) WO1999016438A1 (fr)
ZA (1) ZA988797B (fr)

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Also Published As

Publication number Publication date
IL158649A (en) 2006-12-10
HUP0004024A3 (en) 2001-10-29
ZA988797B (en) 1999-12-02
TW581815B (en) 2004-04-01
NZ517808A (en) 2003-07-25
KR20010015623A (ko) 2001-02-26
IL158649A0 (en) 2004-05-12
ATE281834T1 (de) 2004-11-15
JP2001517699A (ja) 2001-10-09
PL339744A1 (en) 2001-01-02
UA72448C2 (en) 2005-03-15
BG104356A (en) 2000-12-29
US6093728A (en) 2000-07-25
EP1017384B1 (fr) 2004-11-10
HK1032206A1 (en) 2001-07-13
SK285357B6 (sk) 2006-11-03
IL135109A (en) 2007-07-04
NZ503432A (en) 2002-11-26
CA2305370C (fr) 2006-11-28
US20030181480A1 (en) 2003-09-25
ES2230719T3 (es) 2005-05-01
PT1017384E (pt) 2005-03-31
CA2305370A1 (fr) 1999-04-08
PL191618B1 (pl) 2006-06-30
TR200001546T2 (tr) 2000-10-23
AR017266A1 (es) 2001-09-05
IL135109A0 (en) 2001-05-20
AU748849B2 (en) 2002-06-13
DE69827516D1 (de) 2004-12-16
SK4152000A3 (en) 2002-02-05
RU2230553C2 (ru) 2004-06-20
CN1278172A (zh) 2000-12-27
NO325663B1 (no) 2008-07-07
US6855723B2 (en) 2005-02-15
KR100547929B1 (ko) 2006-02-02
BR9812682A (pt) 2000-08-22
HUP0004024A2 (hu) 2001-04-28
NO20001555D0 (no) 2000-03-24
DE69827516T2 (de) 2005-12-01
NO20001555L (no) 2000-03-24
BG64784B1 (bg) 2006-04-28
AU9578198A (en) 1999-04-23
EP1017384A1 (fr) 2000-07-12
CN1167420C (zh) 2004-09-22
WO1999016438A1 (fr) 1999-04-08

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