DK1077703T3 - Orale lægemiddelformer med reproducerbar frisættelse af gatifloxacin eller farmaceutisk anvendelige salte eller hydrater deraf - Google Patents

Orale lægemiddelformer med reproducerbar frisættelse af gatifloxacin eller farmaceutisk anvendelige salte eller hydrater deraf

Info

Publication number
DK1077703T3
DK1077703T3 DK99923491T DK99923491T DK1077703T3 DK 1077703 T3 DK1077703 T3 DK 1077703T3 DK 99923491 T DK99923491 T DK 99923491T DK 99923491 T DK99923491 T DK 99923491T DK 1077703 T3 DK1077703 T3 DK 1077703T3
Authority
DK
Denmark
Prior art keywords
gatifloxacin
hydrates
oral pharmaceutical
pharmaceutical forms
pharmaceutically usable
Prior art date
Application number
DK99923491T
Other languages
English (en)
Inventor
Johannes Bartholomaeus
Juergen Betzing
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Application granted granted Critical
Publication of DK1077703T3 publication Critical patent/DK1077703T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK99923491T 1998-05-09 1999-04-29 Orale lægemiddelformer med reproducerbar frisættelse af gatifloxacin eller farmaceutisk anvendelige salte eller hydrater deraf DK1077703T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19820801A DE19820801A1 (de) 1998-05-09 1998-05-09 Orale Arzneiformen mit reproduzierbarer Wirkstofffreisetzung von Gatifloxacin oder pharmazeutisch verwendbaren Salzen oder Hydraten
PCT/EP1999/002893 WO1999058129A1 (de) 1998-05-09 1999-04-29 Orale arzneiformen mit reproduzierbarer wirkstofffreisetzung von gatifloxacin oder pharmazeutisch verwendbaren salzen oder hydraten

Publications (1)

Publication Number Publication Date
DK1077703T3 true DK1077703T3 (da) 2003-06-23

Family

ID=7867223

Family Applications (1)

Application Number Title Priority Date Filing Date
DK99923491T DK1077703T3 (da) 1998-05-09 1999-04-29 Orale lægemiddelformer med reproducerbar frisættelse af gatifloxacin eller farmaceutisk anvendelige salte eller hydrater deraf

Country Status (27)

Country Link
US (1) US6291462B1 (da)
EP (1) EP1077703B1 (da)
JP (1) JP2002514600A (da)
KR (1) KR100587210B1 (da)
CN (1) CN1198615C (da)
AR (1) AR019279A1 (da)
AT (1) ATE235242T1 (da)
AU (1) AU753482B2 (da)
BR (1) BR9910350A (da)
CA (1) CA2325636A1 (da)
CO (1) CO5050341A1 (da)
DE (2) DE19820801A1 (da)
DK (1) DK1077703T3 (da)
ES (1) ES2195573T3 (da)
HU (1) HUP0101597A3 (da)
IL (1) IL139512A0 (da)
MY (1) MY118569A (da)
NO (1) NO20005385D0 (da)
NZ (1) NZ507968A (da)
PE (1) PE20000480A1 (da)
PL (1) PL343936A1 (da)
PT (1) PT1077703E (da)
RU (1) RU2226394C2 (da)
SK (1) SK16772000A3 (da)
UA (1) UA60364C2 (da)
WO (1) WO1999058129A1 (da)
ZA (1) ZA200006440B (da)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU230030B1 (hu) 1999-10-08 2015-05-28 Debiopharm International Sa Fab I inhibitorok
US6413969B1 (en) * 2000-09-13 2002-07-02 Bristol-Myers Squibb Company Gatifloxacin pentahydrate
EP1560584B1 (en) * 2001-04-06 2009-01-14 Affinium Pharmaceuticals, Inc. Fab i inhibitors
US6589955B2 (en) * 2001-06-20 2003-07-08 Bristol-Myers Squibb Company Pediatric formulation of gatifloxacin
EP1575951B1 (en) * 2002-12-06 2014-06-25 Debiopharm International SA Heterocyclic compounds, methods of making them and their use in therapy
WO2004082586A2 (en) 2003-03-17 2004-09-30 Affinium Pharmaceuticals, Inc. Phamaceutical compositions comprising inhibitors of fab i and further antibiotics
US20050031683A1 (en) * 2003-08-04 2005-02-10 Ashish Kapoor Solid pharmaceutical composition
WO2005021000A1 (en) * 2003-08-28 2005-03-10 Ranbaxy Laboratories Limited Solid oral dosage forms of gatifloxacin
PE20142101A1 (es) * 2004-03-17 2014-12-27 Novartis Ag Composiciones farmaceuticas de aliskiren
DK1828167T3 (da) * 2004-06-04 2014-10-20 Debiopharm Int Sa Acrylamidderivater som antibiotiske midler
US20060247255A1 (en) * 2005-05-02 2006-11-02 Patel Satishkumar A Method for preparing a stable gatifloxacin composition
AU2006275439A1 (en) * 2005-08-02 2007-02-08 Baxter Healthcare S.A. Medical products and parenteral formulations
KR20080075027A (ko) * 2005-12-05 2008-08-13 아피늄 파마슈티컬스, 인크. Ｆａｂｉ 억제제 및 항박테리아제로서의헤테로시클릴아크릴아미드 화합물
JP5468899B2 (ja) 2006-07-20 2014-04-09 アフィニウム ファーマシューティカルズ， インク． Ｆａｂｉインヒビターとしてのアクリルアミド誘導体
CN100415212C (zh) * 2006-07-21 2008-09-03 哈药集团制药总厂 一种含乳酸卡德沙星的口服制剂
CA2563690C (en) * 2006-10-12 2014-10-07 Pharmascience Inc. Pharmaceutical compositions comprising intra- and extra- granular fractions
EP2125802A4 (en) 2007-02-16 2014-08-20 Debiopharm Int Sa SALTS, PRODRUGS AND POLYMORPHES OF FAB I INHIBITORS
AU2013279021C1 (en) 2012-06-19 2017-03-16 Debiopharm International Sa Prodrug derivatives of (E)-N-methyl-N-((3-methylbenzofuran-2-yl)methyl)-3-(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)acrylamide
RS61312B1 (sr) 2016-02-26 2021-02-26 Debiopharm Int Sa Lek za lečenje infekcija dijabetskog stopala
TN2021000159A1 (en) 2019-02-14 2023-04-04 Debiopharm Int Sa Afabicin formulation, method for making the same and uses thereof
SG11202113174SA (en) 2019-06-14 2021-12-30 Debiopharm Int Sa Medicament and use thereof for treating bacterial infections involving biofilm

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH089597B2 (ja) * 1986-01-21 1996-01-31 杏林製薬株式会社 選択毒性に優れた８‐アルコキシキノロンカルボン酸およびその塩並びにその製造方法
DE3887179T2 (de) * 1987-03-02 1994-06-16 Brocades Pharma Bv Pharmazeutische Zusammensetzung, pharmazeutisches Granulat und Verfahren zu ihrer Herstellung.
MY110880A (en) * 1991-01-30 1999-06-30 The Wellcome Foundation Ltd Water-dispersible tablets
GB9109862D0 (en) * 1991-05-08 1991-07-03 Beecham Lab Sa Pharmaceutical formulations
JP2647338B2 (ja) * 1993-02-10 1997-08-27 武田薬品工業株式会社 素錠およびその製造方法
US5436253A (en) * 1993-09-08 1995-07-25 Daiichi Pharmaceutical Co., Ltd. Pyridonecarboxylic acid derivatives and mycotic infections
ATE251896T1 (de) * 1994-12-19 2003-11-15 Daiichi Seiyaku Co Granulat-präparate mit kontinuierlicher freisetzung und verfahren zur herstellung
JP3449658B2 (ja) * 1994-12-21 2003-09-22 杏林製薬株式会社 安定性に優れた８−アルコキシキノロンカルボン酸水和物並びにその製造方法
US5945124A (en) * 1995-07-05 1999-08-31 Byk Gulden Chemische Fabrik Gmbh Oral pharmaceutical composition with delayed release of active ingredient for pantoprazole
US5837292A (en) * 1996-07-03 1998-11-17 Yamanouchi Europe B.V. Granulate for the preparation of fast-disintegrating and fast-dissolving compositions containing a high amount of drug
CA2311734C (en) * 2000-04-12 2011-03-08 Bristol-Myers Squibb Company Flash-melt oral dosage formulation

Also Published As

Publication number Publication date
KR20010043408A (ko) 2001-05-25
SK16772000A3 (sk) 2001-05-10
IL139512A0 (en) 2001-11-25
CO5050341A1 (es) 2001-06-27
NO20005385L (no) 2000-10-26
ES2195573T3 (es) 2003-12-01
EP1077703A1 (de) 2001-02-28
BR9910350A (pt) 2001-09-25
PT1077703E (pt) 2003-08-29
WO1999058129A1 (de) 1999-11-18
NZ507968A (en) 2002-12-20
EP1077703B1 (de) 2003-03-26
NO20005385D0 (no) 2000-10-26
HK1033281A1 (en) 2001-08-24
CN1300216A (zh) 2001-06-20
MY118569A (en) 2004-12-31
AU4035299A (en) 1999-11-29
US6291462B1 (en) 2001-09-18
HUP0101597A3 (en) 2003-01-28
PL343936A1 (en) 2001-09-10
CA2325636A1 (en) 1999-11-18
KR100587210B1 (ko) 2006-06-08
PE20000480A1 (es) 2000-05-20
AU753482B2 (en) 2002-10-17
UA60364C2 (uk) 2003-10-15
ZA200006440B (en) 2002-02-08
CN1198615C (zh) 2005-04-27
JP2002514600A (ja) 2002-05-21
DE59904737D1 (de) 2003-04-30
HUP0101597A2 (hu) 2001-11-28
AR019279A1 (es) 2002-02-13
ATE235242T1 (de) 2003-04-15
RU2226394C2 (ru) 2004-04-10
DE19820801A1 (de) 1999-11-25

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