DK11593A - Fremgangsmaade til fremstilling af (s)-citalopram og forbindelser der kan anvendes som mellemprodukt ved fremgangsmaaden - Google Patents

Fremgangsmaade til fremstilling af (s)-citalopram og forbindelser der kan anvendes som mellemprodukt ved fremgangsmaaden

Info

Publication number
DK11593A
DK11593A DK011593A DK11593A DK11593A DK 11593 A DK11593 A DK 11593A DK 011593 A DK011593 A DK 011593A DK 11593 A DK11593 A DK 11593A DK 11593 A DK11593 A DK 11593A
Authority
DK
Denmark
Prior art keywords
procedure
preparation
relationships
capital program
well
Prior art date
Application number
DK011593A
Other languages
English (en)
Other versions
DK170280B1 (da
DK11593D0 (da
Inventor
Klaus Peter Boegesoe
Jens Kristian Perregaard
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10638616&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK11593(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of DK11593A publication Critical patent/DK11593A/da
Publication of DK11593D0 publication Critical patent/DK11593D0/da
Application granted granted Critical
Publication of DK170280B1 publication Critical patent/DK170280B1/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Psychiatry (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Addiction (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Silicon Compounds (AREA)
DK011593A 1988-06-14 1993-02-01 Fremgangsmåde til fremstilling af (+)-citalopram og forbindelser der kan anvendes som mellemprodukt ved fremgangsmåden DK170280B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB888814057A GB8814057D0 (en) 1988-06-14 1988-06-14 New enantiomers & their isolation
GB8814057 1988-06-14

Publications (3)

Publication Number Publication Date
DK11593A true DK11593A (da) 1993-02-01
DK11593D0 DK11593D0 (da) 1993-02-01
DK170280B1 DK170280B1 (da) 1995-07-24

Family

ID=10638616

Family Applications (2)

Application Number Title Priority Date Filing Date
DK259989A DK259989A (da) 1988-06-14 1989-05-29 Nye enantiomere og deres isolering
DK011593A DK170280B1 (da) 1988-06-14 1993-02-01 Fremgangsmåde til fremstilling af (+)-citalopram og forbindelser der kan anvendes som mellemprodukt ved fremgangsmåden

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK259989A DK259989A (da) 1988-06-14 1989-05-29 Nye enantiomere og deres isolering

Country Status (24)

Country Link
US (2) US4943590A (da)
EP (1) EP0347066B1 (da)
JP (2) JP3044253B2 (da)
AT (1) ATE119896T1 (da)
AU (1) AU623144B2 (da)
CA (2) CA1339452C (da)
CY (2) CY2081B1 (da)
DE (2) DE68921672T2 (da)
DK (2) DK259989A (da)
ES (1) ES2068891T4 (da)
FI (4) FI98627C (da)
GB (1) GB8814057D0 (da)
GR (1) GR3015889T3 (da)
HK (1) HK139596A (da)
HU (1) HU211460A9 (da)
IE (1) IE65734B1 (da)
IL (1) IL90465A (da)
LU (1) LU90999I2 (da)
MX (1) MX9203346A (da)
NL (1) NL300155I2 (da)
NO (2) NO172892C (da)
NZ (1) NZ229426A (da)
PT (1) PT90845B (da)
ZA (1) ZA894476B (da)

Families Citing this family (148)

* Cited by examiner, † Cited by third party
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DE4439836C1 (de) * 1994-11-08 1996-06-05 Hoechst Ag cis-4-(2,2,3,3-Tetrafluorpropoxy)-zimtsäurenitril und trans-4-(2,2,3,3-Tetrafluorpropoxy)- zimtsäurenitril und ein Verfahren zu ihrer Herstellung
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AR021155A1 (es) * 1999-07-08 2002-06-12 Lundbeck & Co As H Tratamiento de desordenes neuroticos
US6759437B2 (en) 1999-10-04 2004-07-06 Martin C. Hinz Comprehensive pharmacologic therapy for treatment of obesity including cysteine
US6403657B1 (en) 1999-10-04 2002-06-11 Martin C. Hinz Comprehensive pharmacologic therapy for treatment of obesity
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GB2357762B (en) * 2000-03-13 2002-01-30 Lundbeck & Co As H Crystalline base of citalopram
KR20020080485A (ko) * 2000-03-13 2002-10-23 하. 룬트벡 아크티에 셀스카브 5-치환 1-(4-플루오로페닐)-1,3-디히드로이소벤조푸란의단계적 알킬화
ES2214400T3 (es) 2000-03-14 2004-09-16 H. Lundbeck A/S Metodo para la preparacion de citalopram.
DE10190485T1 (de) * 2000-03-16 2002-03-21 Lundbeck & Co As H Verfahren zur Herstellung von 5-Cyano-1-(4-fluorphenyl)-1,3-dihydroisobenzofuranen
AR032455A1 (es) 2000-05-12 2003-11-12 Lundbeck & Co As H Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
EA008372B1 (ru) * 2000-07-07 2007-04-27 Х.Лундбекк А/С Применение эсциталопрама для лечения расстройства, связанного с социальной тревогой
EA008373B1 (ru) * 2000-07-07 2007-04-27 Х. Лундбекк А/С Применение эсциталопрама для лечения расстройства, связанного с посттравматическим стрессом
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US20030109577A1 (en) * 2000-10-27 2003-06-12 Ken Liljegren Pharmaceutical composition containing citalopram
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CZ20033267A3 (en) * 2001-05-01 2004-06-16 H. Lundbeck A/S The use of enantiomeric pure escitalopram
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PT1522539E (pt) * 2001-07-31 2007-03-30 Lundbeck & Co As H Composição cristalina contendo escitalopram
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MEP5808A (xx) * 2002-12-23 2010-02-10 Lundbeck & Co As H Ecitalopram bromhidrat i postupak za njegovo pripremanje
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DE10399030I1 (de) 2004-01-08
PT90845B (pt) 1994-11-30
CA1339568C (en) 1997-12-02
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FI98627C (fi) 1997-07-25
JP3038204B2 (ja) 2000-05-08
DE10399030I2 (de) 2004-08-12
DK259989D0 (da) 1989-05-29
FI20041359A7 (fi) 2004-10-20
NO172892B (no) 1993-06-14
DE68921672D1 (de) 1995-04-20
HK139596A (en) 1996-08-02
NL300155I2 (nl) 2005-09-01
ES2068891T3 (es) 1995-05-01
GB8814057D0 (en) 1988-07-20
JPH11292867A (ja) 1999-10-26
CA1339452C (en) 1997-09-09
ZA894476B (en) 1990-04-25
ATE119896T1 (de) 1995-04-15
MX9203346A (es) 1992-08-31
AU623144C (en) 1990-01-04
CY2007004I2 (el) 2009-11-04
NO172892C (no) 1993-09-22
JP3044253B2 (ja) 2000-05-22
IL90465A (en) 1995-01-24
EP0347066B1 (en) 1995-03-15
FI20000507L (fi) 2000-03-06
FI941829A0 (fi) 1994-04-20
JPH0236177A (ja) 1990-02-06
FI20041359L (fi) 2004-10-20
CY2007004I1 (el) 2009-11-04
FI892823A0 (fi) 1989-06-08
EP0347066A1 (en) 1989-12-20
FI20000507A7 (fi) 2000-03-06
NZ229426A (en) 1990-12-21
CY2081B1 (en) 1998-10-16
LU90999I2 (fr) 2003-03-17
DK170280B1 (da) 1995-07-24
DK11593D0 (da) 1993-02-01
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FI91527B (fi) 1994-03-31
FI113762B (fi) 2004-06-15
GR3015889T3 (en) 1995-07-31
US4943590A (en) 1990-07-24
FI892823L (fi) 1989-12-15
FI941829L (fi) 1994-04-20
AU623144B2 (en) 1992-05-07
IE65734B1 (en) 1995-11-15
DE68921672T2 (de) 1995-07-27
HU211460A9 (en) 1995-11-28
PT90845A (pt) 1989-12-29
AU3629589A (en) 1990-01-04
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USRE34712E (en) 1994-08-30
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B1 Patent granted (law 1993)
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Spc suppl protection certif: CA 2002 00011

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Free format text: PRODUCT NAME: ESCITALOPRAM; NAT. REGISTRATION NO/DATE: 33407, 33408, 33409, 33411 20020523; FIRST REGISTRATION: SE 17084-17087 20011207

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