DK1208095T3 - Dibenzopyraner som glucocorticoidreceptorantagonister til behandling af diabetes - Google Patents

Dibenzopyraner som glucocorticoidreceptorantagonister til behandling af diabetes

Info

Publication number
DK1208095T3
DK1208095T3 DK00959835T DK00959835T DK1208095T3 DK 1208095 T3 DK1208095 T3 DK 1208095T3 DK 00959835 T DK00959835 T DK 00959835T DK 00959835 T DK00959835 T DK 00959835T DK 1208095 T3 DK1208095 T3 DK 1208095T3
Authority
DK
Denmark
Prior art keywords
dibenzopyrans
diabetes
treatment
receptor antagonists
glucocorticoid receptor
Prior art date
Application number
DK00959835T
Other languages
English (en)
Inventor
Philip R Kym
Benjamin C Lane
John K Pratt
Geldern Tom Von
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Lab filed Critical Abbott Lab
Application granted granted Critical
Publication of DK1208095T3 publication Critical patent/DK1208095T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78—Ring systems having three or more relevant rings
    • C07D311/80—Dibenzopyrans; Hydrogenated dibenzopyrans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrane Compounds (AREA)
DK00959835T 1999-09-01 2000-09-01 Dibenzopyraner som glucocorticoidreceptorantagonister til behandling af diabetes DK1208095T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US38825199A 1999-09-01 1999-09-01
PCT/US2000/024234 WO2001016128A1 (en) 1999-09-01 2000-09-01 Dibenzopyrans as glucocorticoid receptor antagonists for treatment of diabetes

Publications (1)

Publication Number Publication Date
DK1208095T3 true DK1208095T3 (da) 2004-09-20

Family

ID=23533319

Family Applications (1)

Application Number Title Priority Date Filing Date
DK00959835T DK1208095T3 (da) 1999-09-01 2000-09-01 Dibenzopyraner som glucocorticoidreceptorantagonister til behandling af diabetes

Country Status (15)

Country Link
EP (1) EP1208095B1 (da)
JP (1) JP2003508393A (da)
AR (1) AR034096A1 (da)
AT (1) ATE266655T1 (da)
AU (1) AU7109000A (da)
BR (1) BR0009320A (da)
CA (1) CA2381239A1 (da)
CO (1) CO5180649A1 (da)
DE (1) DE60010722T2 (da)
DK (1) DK1208095T3 (da)
ES (1) ES2220529T3 (da)
HK (1) HK1047580B (da)
MX (1) MXPA02002110A (da)
PT (1) PT1208095E (da)
WO (1) WO2001016128A1 (da)

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US20120029054A1 (en) 2009-03-19 2012-02-02 Merck Sharp & Dohme Corp. RNA Interference Mediated Inhibition of GATA Binding Protein 3 (GATA3) Gene Expression Using Short Intefering Nucleic Acid (siNA)
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WO2011067365A1 (en) 2009-12-03 2011-06-09 Glaxo Group Limited Benzpyrazole derivatives as inhibitors of p13 kinases
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Also Published As

Publication number Publication date
CA2381239A1 (en) 2001-03-08
AU7109000A (en) 2001-03-26
DE60010722T2 (de) 2005-05-12
JP2003508393A (ja) 2003-03-04
ES2220529T3 (es) 2004-12-16
AR034096A1 (es) 2004-02-04
EP1208095A1 (en) 2002-05-29
WO2001016128A1 (en) 2001-03-08
CO5180649A1 (es) 2002-07-30
ATE266655T1 (de) 2004-05-15
HK1047580A1 (en) 2003-02-28
HK1047580B (en) 2005-04-01
DE60010722D1 (de) 2004-06-17
EP1208095B1 (en) 2004-05-12
PT1208095E (pt) 2004-09-30
BR0009320A (pt) 2002-02-05
MXPA02002110A (es) 2002-11-07

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