DK1226131T3 - Isoxazolcarboxamidderivater - Google Patents
IsoxazolcarboxamidderivaterInfo
- Publication number
- DK1226131T3 DK1226131T3 DK00992436T DK00992436T DK1226131T3 DK 1226131 T3 DK1226131 T3 DK 1226131T3 DK 00992436 T DK00992436 T DK 00992436T DK 00992436 T DK00992436 T DK 00992436T DK 1226131 T3 DK1226131 T3 DK 1226131T3
- Authority
- DK
- Denmark
- Prior art keywords
- carboxamide derivatives
- isoxazole carboxamide
- isoxazole
- derivatives
- carboxamide
- Prior art date
Links
- LKYNGTHMKCTTQC-UHFFFAOYSA-N 1,2-oxazole-3-carboxamide Chemical class NC(=O)C=1C=CON=1 LKYNGTHMKCTTQC-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D261/18—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Urology & Nephrology (AREA)
- Ophthalmology & Optometry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Cardiology (AREA)
- Gynecology & Obstetrics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT1999MI002173A IT1314191B1 (it) | 1999-10-18 | 1999-10-18 | Derivati isossazolcarbossamidici |
| PCT/EP2000/010144 WO2001029015A2 (en) | 1999-10-18 | 2000-10-16 | Isoxazolecarboxamide derivatives as alpha1-adrenergic receptor antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1226131T3 true DK1226131T3 (da) | 2004-04-19 |
Family
ID=11383797
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK00992436T DK1226131T3 (da) | 1999-10-18 | 2000-10-16 | Isoxazolcarboxamidderivater |
Country Status (25)
| Country | Link |
|---|---|
| EP (1) | EP1226131B1 (da) |
| JP (1) | JP2003512362A (da) |
| KR (1) | KR20020038944A (da) |
| CN (1) | CN1139579C (da) |
| AR (1) | AR029400A1 (da) |
| AT (1) | ATE256670T1 (da) |
| AU (1) | AU757614B2 (da) |
| BR (1) | BR0014851A (da) |
| CA (1) | CA2385472A1 (da) |
| DE (1) | DE60007347T2 (da) |
| DK (1) | DK1226131T3 (da) |
| ES (1) | ES2210033T3 (da) |
| HK (1) | HK1044940A1 (da) |
| HU (1) | HUP0203184A3 (da) |
| IL (1) | IL148837A0 (da) |
| IT (1) | IT1314191B1 (da) |
| MX (1) | MXPA02003432A (da) |
| MY (1) | MY120400A (da) |
| NO (1) | NO20021803L (da) |
| NZ (1) | NZ517884A (da) |
| PL (1) | PL356990A1 (da) |
| PT (1) | PT1226131E (da) |
| RU (1) | RU2002113096A (da) |
| WO (1) | WO2001029015A2 (da) |
| ZA (1) | ZA200203942B (da) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101277952B (zh) | 2005-10-11 | 2011-09-28 | 弗·哈夫曼-拉罗切有限公司 | 异*唑衍生物 |
| DE602006014185D1 (de) | 2005-11-09 | 2010-06-17 | Hoffmann La Roche | 3-arylisoxazol-4-carbonylbenzofuranderivative |
| RU2426731C2 (ru) | 2005-12-23 | 2011-08-20 | Ф. Хоффманн-Ля Рош Аг | Производные арил-изоксазоло-4-ил-оксадиазола |
| PL1968973T3 (pl) | 2005-12-27 | 2012-03-30 | Hoffmann La Roche | Pochodne aryloizoksazol-4-iloimidazolu |
| KR101062583B1 (ko) | 2006-01-17 | 2011-09-06 | 에프. 호프만-라 로슈 아게 | Ｇａｂａ 수용체에 의해 알츠하이머병의 치료에 유용한아릴-아이속사졸-4-일-이미다조[1,2-ａ]피리딘 |
| KR101119365B1 (ko) | 2006-05-31 | 2012-03-07 | 에프. 호프만-라 로슈 아게 | 아릴-4-에틴일-아이속사졸 유도체 |
| CN101965344B (zh) | 2007-06-22 | 2013-03-06 | 弗·哈夫曼-拉罗切有限公司 | 异*唑-咪唑衍生物 |
| US7902201B2 (en) | 2007-12-04 | 2011-03-08 | Hoffmann-La Roche Inc. | Isoxazolo-pyrazine derivatives |
| US7943619B2 (en) | 2007-12-04 | 2011-05-17 | Hoffmann-La Roche Inc. | Isoxazolo-pyridazine derivatives |
| US7618973B2 (en) | 2007-12-04 | 2009-11-17 | Hoffmann-La Roche Inc. | Isoxazolo-pyrazine derivatives |
| WO2010081851A1 (en) | 2009-01-14 | 2010-07-22 | Genoscience Pharma | Piperidin-4-ylpiperazine compounds for the treatment of hcv infection |
| TW201033201A (en) | 2009-02-19 | 2010-09-16 | Hoffmann La Roche | Isoxazole-isoxazole and isoxazole-isothiazole derivatives |
| US8389550B2 (en) | 2009-02-25 | 2013-03-05 | Hoffmann-La Roche Inc. | Isoxazoles / O-pyridines with ethyl and ethenyl linker |
| US8222246B2 (en) | 2009-04-02 | 2012-07-17 | Hoffmann-La Roche Inc. | Substituted isoxazoles |
| US8227461B2 (en) | 2009-04-30 | 2012-07-24 | Hoffmann-La Roche Inc. | Isoxazoles |
| ES2601181T3 (es) | 2009-05-05 | 2017-02-14 | F. Hoffmann-La Roche Ag | Derivados de isoxazol-tiazol como agonistas inversos del receptor GABA A para su uso en el tratamiento de trastornos cognitivos |
| BRPI1014454A2 (pt) | 2009-05-05 | 2016-04-05 | Hoffmann La Roche | derivados de isoxazol-pirazol |
| BRPI1013762A2 (pt) | 2009-05-05 | 2015-08-25 | Hoffmann La Roche | "derivados isoxazol-piridazina" |
| US8415379B2 (en) | 2009-05-05 | 2013-04-09 | Hoffmann-La Roche Inc. | Pyridines |
| KR101354416B1 (ko) | 2009-05-07 | 2014-02-19 | 에프. 호프만-라 로슈 아게 | 감마-아미노부티르산 조절제로서 이속사졸-피리딘 유도체 |
| US8785435B2 (en) | 2011-10-20 | 2014-07-22 | Hoffmann-La Roche Inc. | Solid forms |
| CN113121540B (zh) * | 2020-01-15 | 2024-01-26 | 鲁南制药集团股份有限公司 | 一种西格列汀游离碱的合成方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1254469B (it) * | 1992-02-25 | 1995-09-25 | Recordati Chem Pharm | Derivati benzopiranici e benzotiopiranici |
| IT1266582B1 (it) * | 1993-07-30 | 1997-01-09 | Recordati Chem Pharm | Derivati (di)azacicloesanici e diazacicloeptanici |
| DE4425146A1 (de) * | 1994-07-15 | 1996-01-18 | Basf Ag | Verwendung heterocyclischer Verbindungen |
-
1999
- 1999-10-18 IT IT1999MI002173A patent/IT1314191B1/it active
-
2000
- 2000-10-10 MY MYPI20004718A patent/MY120400A/en unknown
- 2000-10-16 ES ES00992436T patent/ES2210033T3/es not_active Expired - Lifetime
- 2000-10-16 BR BR0014851-2A patent/BR0014851A/pt not_active IP Right Cessation
- 2000-10-16 CN CNB008143226A patent/CN1139579C/zh not_active Expired - Fee Related
- 2000-10-16 RU RU2002113096/04A patent/RU2002113096A/ru not_active Application Discontinuation
- 2000-10-16 DK DK00992436T patent/DK1226131T3/da active
- 2000-10-16 PT PT00992436T patent/PT1226131E/pt unknown
- 2000-10-16 NZ NZ517884A patent/NZ517884A/en unknown
- 2000-10-16 AT AT00992436T patent/ATE256670T1/de not_active IP Right Cessation
- 2000-10-16 WO PCT/EP2000/010144 patent/WO2001029015A2/en not_active Ceased
- 2000-10-16 HK HK02105918.6A patent/HK1044940A1/zh unknown
- 2000-10-16 IL IL14883700A patent/IL148837A0/xx unknown
- 2000-10-16 AU AU28347/01A patent/AU757614B2/en not_active Ceased
- 2000-10-16 CA CA002385472A patent/CA2385472A1/en not_active Abandoned
- 2000-10-16 EP EP00992436A patent/EP1226131B1/en not_active Expired - Lifetime
- 2000-10-16 DE DE60007347T patent/DE60007347T2/de not_active Expired - Fee Related
- 2000-10-16 JP JP2001531815A patent/JP2003512362A/ja active Pending
- 2000-10-16 MX MXPA02003432A patent/MXPA02003432A/es not_active Application Discontinuation
- 2000-10-16 PL PL00356990A patent/PL356990A1/xx not_active Application Discontinuation
- 2000-10-16 KR KR1020027004663A patent/KR20020038944A/ko not_active Withdrawn
- 2000-10-16 HU HU0203184A patent/HUP0203184A3/hu unknown
- 2000-10-18 AR ARP000105475A patent/AR029400A1/es not_active Application Discontinuation
-
2002
- 2002-04-17 NO NO20021803A patent/NO20021803L/no not_active Application Discontinuation
- 2002-05-17 ZA ZA200203942A patent/ZA200203942B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL148837A0 (en) | 2002-09-12 |
| DE60007347T2 (de) | 2004-09-02 |
| NO20021803D0 (no) | 2002-04-17 |
| BR0014851A (pt) | 2002-06-11 |
| ES2210033T3 (es) | 2004-07-01 |
| WO2001029015A3 (en) | 2001-11-01 |
| EP1226131B1 (en) | 2003-12-17 |
| IT1314191B1 (it) | 2002-12-06 |
| ITMI992173A1 (it) | 2001-04-18 |
| HK1044940A1 (zh) | 2002-11-08 |
| DE60007347D1 (de) | 2004-01-29 |
| ATE256670T1 (de) | 2004-01-15 |
| PT1226131E (pt) | 2004-05-31 |
| WO2001029015A2 (en) | 2001-04-26 |
| EP1226131A2 (en) | 2002-07-31 |
| PL356990A1 (en) | 2004-07-12 |
| ITMI992173A0 (it) | 1999-10-18 |
| CN1379767A (zh) | 2002-11-13 |
| NZ517884A (en) | 2003-08-29 |
| MXPA02003432A (es) | 2002-08-20 |
| ZA200203942B (en) | 2003-01-02 |
| MY120400A (en) | 2005-10-31 |
| HUP0203184A3 (en) | 2004-12-28 |
| HUP0203184A2 (hu) | 2003-01-28 |
| CA2385472A1 (en) | 2001-04-26 |
| JP2003512362A (ja) | 2003-04-02 |
| RU2002113096A (ru) | 2003-11-10 |
| KR20020038944A (ko) | 2002-05-24 |
| AR029400A1 (es) | 2003-06-25 |
| AU757614B2 (en) | 2003-02-27 |
| CN1139579C (zh) | 2004-02-25 |
| NO20021803L (no) | 2002-06-17 |
| AU2834701A (en) | 2001-04-30 |
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