DK132778A - Pyrido(2,1-b) quinazolin-derivater deres fremstilling og anvendelser - Google Patents

Pyrido(2,1-b) quinazolin-derivater deres fremstilling og anvendelser

Info

Publication number: DK132778A
Authority: DK; Denmark
Prior art keywords: pyrido; preparation; quinazoline derivatives; quinazoline; derivatives
Prior art date: 1977-03-24

Application number

DK132778A

Other languages

English (en)

Inventor

R W Kierstead

J W Tilley

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-03-24

Filing date

1978-03-22

Publication date

1978-09-25

1978-03-22 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

1978-09-25 Publication of DK132778A publication Critical patent/DK132778A/da

Links

QBEIZCZOJLXENV-UHFFFAOYSA-N 9h-pyrido[2,1-b]quinazoline Chemical class C1=CC=CC2=CN3CC=CC=C3N=C21 QBEIZCZOJLXENV-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
- C07D213/82—Amides; Imides in position 3
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
- C07C205/49—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups
- C07C205/57—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
- C07C205/59—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton the carbon skeleton being further substituted by singly-bound oxygen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/61—Halogen atoms or nitro radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/89—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pulmonology (AREA)
Engineering & Computer Science (AREA)
Immunology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)

DK132778A 1977-03-24 1978-03-22 Pyrido(2,1-b) quinazolin-derivater deres fremstilling og anvendelser DK132778A (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US78093977A	1977-03-24	1977-03-24
US87156478A	1978-01-23	1978-01-23

Publications (1)

Publication Number	Publication Date
DK132778A true DK132778A (da)	1978-09-25

Family

ID=27119777

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
DK132778A DK132778A (da)	1977-03-24	1978-03-22	Pyrido(2,1-b) quinazolin-derivater deres fremstilling og anvendelser
DK128878A DK128878A (da)	1977-03-24	1978-03-22	Pyrido(2,1-b) quinazoliner deres fremstilling og anvendelser

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
DK128878A DK128878A (da)	1977-03-24	1978-03-22	Pyrido(2,1-b) quinazoliner deres fremstilling og anvendelser

Country Status (23)

Country	Link
JP (2)	JPS53119896A (da)
AR (3)	AR218480A1 (da)
AT (2)	AT367050B (da)
AU (2)	AU521352B2 (da)
DE (2)	DE2812585A1 (da)
DK (2)	DK132778A (da)
ES (13)	ES468127A1 (da)
FI (2)	FI780918A7 (da)
FR (2)	FR2384771A1 (da)
GB (2)	GB1601371A (da)
GR (2)	GR72948B (da)
HU (1)	HU180782B (da)
IE (1)	IE46505B1 (da)
IL (2)	IL54328A (da)
IT (2)	IT1093710B (da)
LU (2)	LU79290A1 (da)
MC (2)	MC1185A1 (da)
NL (2)	NL7803122A (da)
NO (2)	NO781051L (da)
NZ (2)	NZ186760A (da)
PH (2)	PH14130A (da)
PT (2)	PT67821B (da)
SE (2)	SE7803419L (da)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DK154297B (da) *	1978-10-18	1988-10-31	Schering Ag	Analogifremgangsmaade til fremstilling af optisk aktive eller racemiske pyridooe2,1-baa-quinazolinonderivater

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE2557425C2 (de) *	1975-12-19	1987-03-19	C.H. Boehringer Sohn, 6507 Ingelheim	11-Oxo-11-H-pyrido[2,1-b]-chinazolin-2-carbonsäure und ihre Salze, Verfahren zu ihrer Herstellung und Arzneimittel
US4395549A (en)	1981-10-02	1983-07-26	Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt.	6-Hydrazono-pyrido[2,1-b] quinazoline-11 ones
ES8306729A1 (es) *	1982-04-30	1983-06-01	Lafarquim	"procedimiento de obtencion de 2-isopropil pirido (2-1-b) quinazolinas y sus sales no toxicas con actividad antianafilactica".
US4551460A (en) *	1982-05-10	1985-11-05	Hoffmann-La Roche Inc.	Pyrido[2,1-b]quinazoline derivatives useful as agents for treatment of allergic conditions and vascular disorders involving thrombosis
DE3300477A1 (de) *	1983-01-08	1984-07-12	Boehringer Ingelheim KG, 6507 Ingelheim	Neue heterocyclische verbindungen, ihre herstellung und verwendung
JPS62238264A (ja) *	1986-04-04	1987-10-19	Nippon Tokushu Noyaku Seizo Kk	２−ハロ−５−アセチルピリジン

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4012387A (en) *	1975-09-18	1977-03-15	Warner-Lambert Company	Benzo-[g]pyrido[2,1-b]quinazolinones
US4033961A (en) *	1975-10-07	1977-07-05	Warner-Lambert Company	Pyrido[2-1-b]quinazolin-ones and their methods of preparation

1978
- 1978-03-22 DE DE19782812585 patent/DE2812585A1/de not_active Withdrawn
- 1978-03-22 IL IL54328A patent/IL54328A/xx unknown
- 1978-03-22 LU LU79290A patent/LU79290A1/de unknown
- 1978-03-22 DK DK132778A patent/DK132778A/da not_active IP Right Cessation
- 1978-03-22 FR FR7808317A patent/FR2384771A1/fr active Granted
- 1978-03-22 NZ NZ186760A patent/NZ186760A/xx unknown
- 1978-03-22 IL IL54326A patent/IL54326A/xx unknown
- 1978-03-22 DE DE19782812586 patent/DE2812586A1/de not_active Withdrawn
- 1978-03-22 NZ NZ186759A patent/NZ186759A/xx unknown
- 1978-03-22 NO NO781051A patent/NO781051L/no unknown
- 1978-03-22 LU LU79293A patent/LU79293A1/de unknown
- 1978-03-22 PH PH20918A patent/PH14130A/en unknown
- 1978-03-22 FR FR7808316A patent/FR2384770A1/fr active Granted
- 1978-03-22 NO NO781053A patent/NO781053L/no unknown
- 1978-03-22 PH PH20917A patent/PH13915A/en unknown
- 1978-03-22 ES ES468127A patent/ES468127A1/es not_active Expired
- 1978-03-22 HU HU78HO2058A patent/HU180782B/hu unknown
- 1978-03-22 ES ES468126A patent/ES468126A1/es not_active Expired
- 1978-03-22 NL NL7803122A patent/NL7803122A/xx not_active Application Discontinuation
- 1978-03-22 NL NL7803112A patent/NL7803112A/xx not_active Application Discontinuation
- 1978-03-22 MC MC781291A patent/MC1185A1/fr unknown
- 1978-03-22 DK DK128878A patent/DK128878A/da not_active Application Discontinuation
- 1978-03-22 MC MC781292A patent/MC1186A1/fr unknown
- 1978-03-23 PT PT67821A patent/PT67821B/pt unknown
- 1978-03-23 AU AU34474/78A patent/AU521352B2/en not_active Expired
- 1978-03-23 SE SE7803419A patent/SE7803419L/xx unknown
- 1978-03-23 FI FI780918A patent/FI780918A7/fi not_active Application Discontinuation
- 1978-03-23 FI FI780917A patent/FI780917A7/fi not_active Application Discontinuation
- 1978-03-23 GR GR55781A patent/GR72948B/el unknown
- 1978-03-23 IE IE582/78A patent/IE46505B1/en unknown
- 1978-03-23 AT AT0210278A patent/AT367050B/de not_active IP Right Cessation
- 1978-03-23 AT AT0210478A patent/AT367051B/de not_active IP Right Cessation
- 1978-03-23 SE SE7803418A patent/SE7803418L/xx unknown
- 1978-03-23 AU AU34475/78A patent/AU521096B2/en not_active Expired
- 1978-03-23 GR GR55782A patent/GR73170B/el unknown
- 1978-03-23 GB GB11704/78A patent/GB1601371A/en not_active Expired
- 1978-03-23 PT PT67820A patent/PT67820A/pt unknown
- 1978-03-23 IT IT7821578A patent/IT1093710B/it active
- 1978-03-23 GB GB11705/78A patent/GB1601991A/en not_active Expired
- 1978-03-24 JP JP3320578A patent/JPS53119896A/ja active Pending
- 1978-03-24 JP JP3400278A patent/JPS53119897A/ja active Pending
- 1978-03-24 IT IT21655/78A patent/IT1095493B/it active
- 1978-03-27 AR AR271537A patent/AR218480A1/es active
- 1978-03-27 AR AR271538A patent/AR218060A1/es active
1979
- 1979-02-16 ES ES478324A patent/ES478324A1/es not_active Expired
- 1979-02-16 ES ES478329A patent/ES478329A1/es not_active Expired
- 1979-02-16 ES ES478328A patent/ES478328A1/es not_active Expired
- 1979-02-16 ES ES478330A patent/ES478330A1/es not_active Expired
- 1979-02-16 ES ES478331A patent/ES478331A1/es not_active Expired
- 1979-02-16 ES ES478325A patent/ES478325A1/es not_active Expired
- 1979-02-16 ES ES478323A patent/ES478323A1/es not_active Expired
- 1979-02-16 ES ES478333A patent/ES478333A1/es not_active Expired
- 1979-02-16 ES ES478326A patent/ES478326A1/es not_active Expired
- 1979-02-16 ES ES478327A patent/ES478327A1/es not_active Expired
- 1979-02-16 ES ES478332A patent/ES478332A1/es not_active Expired
- 1979-05-10 AR AR276467A patent/AR225415A1/es active

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DK154297B (da) *	1978-10-18	1988-10-31	Schering Ag	Analogifremgangsmaade til fremstilling af optisk aktive eller racemiske pyridooe2,1-baa-quinazolinonderivater

Also Published As

Publication number	Publication date
ES478326A1 (es)	1979-11-01
FR2384770A1 (fr)	1978-10-20
FR2384771A1 (fr)	1978-10-20
AU521096B2 (en)	1982-03-18
IL54328A0 (en)	1978-06-15
DE2812585A1 (de)	1978-09-28
ES468126A1 (es)	1979-09-01
IE46505B1 (en)	1983-06-29
GB1601991A (en)	1981-11-04
IL54326A0 (en)	1978-06-15
PT67821B (en)	1980-03-04
FI780917A7 (fi)	1978-09-25
ES478323A1 (es)	1979-11-01
NL7803122A (nl)	1978-09-26
ES478328A1 (es)	1979-11-01
AT367050B (de)	1982-05-25
ES478325A1 (es)	1979-11-01
PH14130A (en)	1981-02-26
LU79293A1 (de)	1979-05-25
NZ186760A (en)	1981-03-16
IT7821578A0 (it)	1978-03-23
MC1186A1 (fr)	1978-12-22
AR225415A1 (es)	1982-03-31
ES478332A1 (es)	1979-11-16
IT7821655A0 (it)	1978-03-24
ATA210478A (de)	1981-10-15
GB1601371A (en)	1981-10-28
NO781051L (no)	1978-09-26
NL7803112A (nl)	1978-09-26
ES468127A1 (es)	1979-09-16
MC1185A1 (fr)	1978-12-22
JPS53119896A (en)	1978-10-19
ES478331A1 (es)	1979-11-16
SE7803419L (sv)	1978-09-25
FR2384771B1 (da)	1980-04-04
IL54326A (en)	1982-04-30
AR218060A1 (es)	1980-05-15
AR218480A1 (es)	1980-06-13
ES478329A1 (es)	1979-11-01
ES478330A1 (es)	1979-11-01
AT367051B (de)	1982-05-25
NZ186759A (en)	1981-03-16
PT67820A (en)	1978-04-01
FI780918A7 (fi)	1978-09-25
IT1095493B (it)	1985-08-10
PH13915A (en)	1980-11-04
ATA210278A (de)	1981-10-15
IE780582L (en)	1978-09-24
LU79290A1 (de)	1979-05-25
HU180782B (en)	1983-04-29
JPS53119897A (en)	1978-10-19
ES478324A1 (es)	1979-11-01
GR73170B (da)	1983-02-14
FR2384770B1 (da)	1980-10-24
SE7803418L (sv)	1978-09-25
IL54328A (en)	1982-03-31
IT1093710B (it)	1985-07-26
NO781053L (no)	1978-09-26
GR72948B (da)	1984-01-17
AU521352B2 (en)	1982-04-01
ES478327A1 (es)	1979-11-01
PT67821A (en)	1978-04-01
AU3447478A (en)	1979-09-27
ES478333A1 (es)	1979-11-16
DE2812586A1 (de)	1978-09-28
DK128878A (da)	1978-09-25
AU3447578A (en)	1979-09-27

Legal Events

Date	Code	Title	Description
1985-09-23	AHS	Application shelved for other reasons than non-payment
1990-10-22	PUP	Patent expired

Publication	Publication Date	Title
DK377678A (da)	1979-02-28	3,4,5-trihydroxypiperidinderivater deres fremstilling og anvendelse
DK450776A (da)	1977-04-08	Pyrido(2,1-b)quinazolinoner samt deres fremstilling og anvendelse
DK569087A (da)	1988-05-01	Quinolin-derivater, deres fremstilling og anvendelse
NL7802671A (nl)	1978-09-14	Cefemderivaten en hun bereiding.
DK462187D0 (da)	1987-09-04	Pyridinyl-pyrimidin-derivater, deres fremstilling og anvendelse.
DK279578A (da)	1979-02-02	Sulfonamidderivater og deres anvendelse som herbicider
DK547378A (da)	1979-06-03	1-n-4,6-di-o(aminoglycosyl-)-1,3-dimino-cyclitol-derivater deres fremstilling og anvendelse
DK239378A (da)	1978-12-01	5,11-dihydro-6h-pyrido(2,3-b)(1,4)-benzodiazepin-6-oner, der er substitueret i 11-stillingen og femgangsmaade til deres fremstilling
NO150275C (no)	1984-09-19	Organiske nitrogenholdige forbindelser og fremgangsmaate til deres fremsilling, samt anvendelse av forbindelsene i sjampo
DK239578A (da)	1978-12-01	5-11-dihydro-6h-pyrido(2,3-b)(1,4)-benzodiazepin-6-oner der substitueret i 11-stillingen og fremgangsmaade til deres fremstilling
DK633287D0 (da)	1987-12-02	Carbamoylimidazo-derivater, deres fremstilling og anvendelse
DK239478A (da)	1978-12-01	5,11-dihydro-6h-pyrido(2,3-b)(1,4)-benzodiazepin-6-oner der er substituerede i 11-stillingen og fremgangsmaade til deres fremstilling
DK28685A (da)	1985-07-24	Azolyl-aryl-alkanol-derivater, deres fremstilling og anvendelse
DK582578A (da)	1979-06-30	2,4-thiazolidindion-derivater og fremgangsmaade til deres fremstilling
DK132778A (da)	1978-09-25	Pyrido(2,1-b) quinazolin-derivater deres fremstilling og anvendelser
DK235787D0 (da)	1987-05-08	Tripeptidderivater, deres fremstilling og anvendelse
DK270077A (da)	1977-12-22	6,7-benzomorphanderivater og fremgangsmade til deres fremstillling
DK319478A (da)	1979-01-19	Angiotensinpeptider og deres fremstilling
DK213387A (da)	1987-10-29	Benzothiazinon-derivater, deres fremstilling og anvendelse
DK482877A (da)	1978-05-02	8-(1h-tetrazol-5-yl)-11h-pyrido (2,1-b) quinazolin-11-oner samt deres fremstilling og anvendelse
DK212687D0 (da)	1987-04-27	Benzothiazinon-derivater, deres fremstilling og anvendelse
DK607787A (da)	1988-05-21	12-halogenerede forskolin-derivater, deres fremstilling og anvendelse
DK546578A (da)	1979-06-23	2-oxo-hexahydroazepin-, -piperidin- og- pyrrolinderivater samt deres fremstilling og anvendelse
DK610787D0 (da)	1987-11-20	Substituerede thienoimidazoltoluidin-derivater, deres fremstilling og anvendelse
DK477778A (da)	1979-04-27	17alfa-(3-jodbenzoyloxy)-9alfa-4-pregnen-3,20-dioner deres d-homoanaloge og fremgangsmaade til deres fremstilling og deres anvendelse

DK132778A - Pyrido(2,1-b) quinazolin-derivater deres fremstilling og anvendelser - Google Patents

Info

Links

Classifications

Landscapes

Applications Claiming Priority (2)

Publications (1)

Family

ID=27119777

Family Applications (2)

Family Applications After (1)

Country Status (23)

Cited By (1)

Families Citing this family (6)

Family Cites Families (2)

Cited By (1)

Also Published As

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