DK142987A - Hidtil ukendte vitamin d-analoger - Google Patents

Hidtil ukendte vitamin d-analoger

Info

Publication number
DK142987A
DK142987A DK142987A DK142987A DK142987A DK 142987 A DK142987 A DK 142987A DK 142987 A DK142987 A DK 142987A DK 142987 A DK142987 A DK 142987A DK 142987 A DK142987 A DK 142987A
Authority
DK
Denmark
Prior art keywords
lower alkyl
hydroxyl
halogen
denotes hydrogen
optionally substituted
Prior art date
Application number
DK142987A
Other languages
English (en)
Other versions
DK166617B1 (da
DK142987D0 (da
Inventor
Martin John Calverley
Ernst Torndal Binderup
Original Assignee
Leo Pharm Prod Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26289597&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK142987(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB858519502A external-priority patent/GB8519502D0/en
Application filed by Leo Pharm Prod Ltd filed Critical Leo Pharm Prod Ltd
Publication of DK142987D0 publication Critical patent/DK142987D0/da
Publication of DK142987A publication Critical patent/DK142987A/da
Application granted granted Critical
Publication of DK166617B1 publication Critical patent/DK166617B1/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C401/00—Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DK142987A 1985-08-02 1987-03-20 24-hydroxylerede d-vitamin-derivater og farmaceutiske praeparater indeholdende disse DK166617B1 (da)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
GB8519502 1985-08-02
GB858519502A GB8519502D0 (en) 1985-08-02 1985-08-02 Chemical compounds
DK8600081 1986-07-14
PCT/DK1986/000081 WO1987000834A1 (en) 1985-08-02 1986-07-14 Novel vitamin d analogues
PH34061A PH25496A (en) 1985-08-02 1986-08-11 New vitamin d analogues
PH3406186 1986-08-11

Publications (3)

Publication Number Publication Date
DK142987D0 DK142987D0 (da) 1987-03-20
DK142987A true DK142987A (da) 1987-03-20
DK166617B1 DK166617B1 (da) 1993-06-21

Family

ID=26289597

Family Applications (1)

Application Number Title Priority Date Filing Date
DK142987A DK166617B1 (da) 1985-08-02 1987-03-20 24-hydroxylerede d-vitamin-derivater og farmaceutiske praeparater indeholdende disse

Country Status (16)

Country Link
US (1) US4866048A (da)
EP (1) EP0227826B1 (da)
JP (1) JPH07100685B2 (da)
KR (1) KR940010767B1 (da)
AU (1) AU603340B2 (da)
CA (1) CA1307288C (da)
DE (1) DE3666587D1 (da)
DK (1) DK166617B1 (da)
ES (1) ES2000823A6 (da)
GR (1) GR862029B (da)
HK (1) HK63492A (da)
IE (1) IE58545B1 (da)
PH (1) PH25496A (da)
PT (1) PT83119B (da)
SG (1) SG64192G (da)
WO (1) WO1987000834A1 (da)

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US5260290A (en) * 1990-02-14 1993-11-09 Wisconsin Alumni Research Foundation Homologated vitamin D2 compounds and the corresponding 1α-hydroxylated derivatives
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US5763428A (en) * 1990-09-21 1998-06-09 Bone Care International, Inc. Methods of treating skin disorders with novel 1a-hydroxy vitamin D4 compounds and derivatives thereof
US5801164A (en) * 1990-09-21 1998-09-01 Bone Care International, Inc. Methods of treating osteoporosis prophylactically or therapeutically
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US5786348A (en) * 1991-01-08 1998-07-28 Bone Care International, Inc. Methods for preparation and use of 1α,24(S)-dihydroxy vitamin D2
US20040009958A1 (en) * 1991-01-08 2004-01-15 Bone Care International, Inc. Methods for preparation and use of 1alpha,24(S)-dihydroxyvitamin D2
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US6503893B2 (en) 1996-12-30 2003-01-07 Bone Care International, Inc. Method of treating hyperproliferative diseases using active vitamin D analogues
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CN105348164B (zh) * 2015-10-29 2017-03-29 无锡福祈制药有限公司 一种1α‑羟基维生素D2的制备方法
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CN107501150A (zh) * 2016-06-14 2017-12-22 江苏吉贝尔药业股份有限公司 两种他卡西醇中间体的制备方法
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CN110156836A (zh) * 2019-06-10 2019-08-23 成家钢 一种环丙基羰基亚甲基三苯基磷的制备方法
CN111662221B (zh) * 2020-06-29 2022-04-19 重庆华邦胜凯制药有限公司 一种卡泊三醇杂质的制备方法
CN115177586A (zh) * 2022-08-31 2022-10-14 江苏知原药业股份有限公司 一种卡泊三醇组合物

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Also Published As

Publication number Publication date
AU603340B2 (en) 1990-11-15
DK166617B1 (da) 1993-06-21
DK142987D0 (da) 1987-03-20
PH25496A (en) 1991-07-24
PT83119B (pt) 1989-03-30
IE861894L (en) 1987-02-02
HK63492A (en) 1992-08-28
EP0227826B1 (en) 1989-10-25
SG64192G (en) 1992-09-04
GR862029B (en) 1986-12-24
PT83119A (en) 1986-09-01
WO1987000834A1 (en) 1987-02-12
EP0227826A1 (en) 1987-07-08
ES2000823A6 (es) 1988-03-16
AU6196186A (en) 1987-03-05
IE58545B1 (en) 1993-10-06
KR870700600A (ko) 1987-12-30
CA1307288C (en) 1992-09-08
DE3666587D1 (en) 1989-11-30
JPS63500661A (ja) 1988-03-10
KR940010767B1 (ko) 1994-11-11
US4866048A (en) 1989-09-12
JPH07100685B2 (ja) 1995-11-01

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