DK1434570T3 - Farmaceutiske formuleringer til kontrolleret frigivelse af 4-amino-6,7-dimethoxy-2-(5-methansulfonamido-1,2,3,4-tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazolin - Google Patents

Farmaceutiske formuleringer til kontrolleret frigivelse af 4-amino-6,7-dimethoxy-2-(5-methansulfonamido-1,2,3,4-tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazolin

Info

Publication number: DK1434570T3
Authority: DK; Denmark
Prior art keywords: tetrahydroisoquinol; methanesulfonamido; quinazoline; dimethoxy; pyridyl
Prior art date: 2001-10-11

Application number

DK02775048T

Other languages

English (en)

Inventor

John D Davis

Michael J Humphrey

Ross J Macrae

Janet S Smith

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-10-11

Filing date

2002-09-30

Publication date

2005-11-07

2002-09-30 Application filed by Pfizer filed Critical Pfizer

2005-11-07 Application granted granted Critical

2005-11-07 Publication of DK1434570T3 publication Critical patent/DK1434570T3/da

Links

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Molecular Biology (AREA)
Biophysics (AREA)
Urology & Nephrology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Plural Heterocyclic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

DK02775048T 2001-10-11 2002-09-30 Farmaceutiske formuleringer til kontrolleret frigivelse af 4-amino-6,7-dimethoxy-2-(5-methansulfonamido-1,2,3,4-tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazolin DK1434570T3 (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GBGB0124455.7A GB0124455D0 (en)	2001-10-11	2001-10-11	Pharmaceutical formulations

Publications (1)

Publication Number	Publication Date
DK1434570T3 true DK1434570T3 (da)	2005-11-07

Family

ID=9923660

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK02775048T DK1434570T3 (da)	2001-10-11	2002-09-30	Farmaceutiske formuleringer til kontrolleret frigivelse af 4-amino-6,7-dimethoxy-2-(5-methansulfonamido-1,2,3,4-tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazolin

Country Status (33)

Country	Link
EP (1)	EP1434570B8 (da)
JP (1)	JP4131471B2 (da)
KR (1)	KR20050032510A (da)
CN (1)	CN1568180A (da)
AP (1)	AP2004003001A0 (da)
AR (1)	AR036782A1 (da)
AT (1)	ATE303135T1 (da)
BR (1)	BR0213196A (da)
CA (1)	CA2461168A1 (da)
CO (1)	CO5560534A2 (da)
DE (1)	DE60205925T2 (da)
DK (1)	DK1434570T3 (da)
DO (1)	DOP2002000464A (da)
EA (1)	EA006168B1 (da)
ES (1)	ES2246017T3 (da)
GB (1)	GB0124455D0 (da)
GT (1)	GT200200184A (da)
HR (1)	HRP20040261A2 (da)
HU (1)	HUP0600064A3 (da)
IL (1)	IL160969A0 (da)
IS (1)	IS7179A (da)
MA (1)	MA27075A1 (da)
MX (1)	MXPA04003293A (da)
NO (1)	NO20041520L (da)
OA (1)	OA12709A (da)
PA (1)	PA8556001A1 (da)
PE (1)	PE20030551A1 (da)
PL (1)	PL369666A1 (da)
PY (1)	PY0223360A (da)
SV (1)	SV2004001279A (da)
UY (1)	UY27477A1 (da)
WO (1)	WO2003032956A1 (da)
ZA (1)	ZA200401976B (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0317663D0 (en) *	2003-07-29	2003-09-03	Astrazeneca Ab	Pharmaceutical composition
EP3821882A1 (en)	2013-03-14	2021-05-19	Amgen Inc.	Heterocyclic compounds and their uses
KR101943592B1 (ko)	2017-08-31	2019-01-30	조현우	데이터 마이닝 기법을 이용한 전자가계부 시스템

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0466986B1 (en) *	1990-07-02	1994-04-27	Bend Research, Inc.	Asymmetric microporous beads for controlled release
FR2752737B1 (fr) *	1996-08-29	1998-10-02	Synthelabo	Comprime a liberation controlee de chlorhydrate d'alfuzosine
GB9700504D0 (en) *	1997-01-11	1997-02-26	Pfizer Ltd	Pharmaceutical compounds
IL141235A (en) *	2000-02-09	2012-04-30	Novartis Int Pharm Ltd	Combined use of an alpha-adrenoceptor antagonist and a muscarinic antagonist in the preparation of a drug for the treatment of non-malignant prostatic hyperplasia
AU779118B2 (en) *	2000-03-03	2005-01-06	Pfizer Inc.	4-amino-6,7-dimethoxy-2-(5-methanesulfonamido-1,2,3, 4-tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazoline mesylate and polymorphs

2001
- 2001-10-11 GB GBGB0124455.7A patent/GB0124455D0/en not_active Ceased
2002
- 2002-09-12 DO DO2002000464A patent/DOP2002000464A/es unknown
- 2002-09-17 GT GT200200184A patent/GT200200184A/es unknown
- 2002-09-25 PY PY200200223360A patent/PY0223360A/es unknown
- 2002-09-30 AP APAP/P/2004/003001A patent/AP2004003001A0/en unknown
- 2002-09-30 WO PCT/IB2002/004040 patent/WO2003032956A1/en not_active Ceased
- 2002-09-30 KR KR1020047005316A patent/KR20050032510A/ko not_active Ceased
- 2002-09-30 OA OA1200400094A patent/OA12709A/en unknown
- 2002-09-30 EA EA200400431A patent/EA006168B1/ru not_active IP Right Cessation
- 2002-09-30 DK DK02775048T patent/DK1434570T3/da active
- 2002-09-30 ES ES02775048T patent/ES2246017T3/es not_active Expired - Lifetime
- 2002-09-30 IL IL16096902A patent/IL160969A0/xx unknown
- 2002-09-30 PL PL02369666A patent/PL369666A1/xx not_active Application Discontinuation
- 2002-09-30 AT AT02775048T patent/ATE303135T1/de not_active IP Right Cessation
- 2002-09-30 MX MXPA04003293A patent/MXPA04003293A/es active IP Right Grant
- 2002-09-30 DE DE60205925T patent/DE60205925T2/de not_active Expired - Lifetime
- 2002-09-30 HU HU0600064A patent/HUP0600064A3/hu unknown
- 2002-09-30 CA CA002461168A patent/CA2461168A1/en not_active Abandoned
- 2002-09-30 BR BR0213196-0A patent/BR0213196A/pt not_active IP Right Cessation
- 2002-09-30 EP EP02775048A patent/EP1434570B8/en not_active Expired - Lifetime
- 2002-09-30 CN CNA02820042XA patent/CN1568180A/zh active Pending
- 2002-09-30 HR HR20040261A patent/HRP20040261A2/hr not_active Application Discontinuation
- 2002-09-30 JP JP2003535760A patent/JP4131471B2/ja not_active Expired - Fee Related
- 2002-10-09 UY UY27477A patent/UY27477A1/es not_active Application Discontinuation
- 2002-10-09 AR ARP020103805A patent/AR036782A1/es unknown
- 2002-10-09 PE PE2002000996A patent/PE20030551A1/es not_active Application Discontinuation
- 2002-10-10 PA PA20028556001A patent/PA8556001A1/es unknown
- 2002-10-10 SV SV2002001279A patent/SV2004001279A/es not_active Application Discontinuation
2004
- 2004-03-11 ZA ZA200401976A patent/ZA200401976B/en unknown
- 2004-03-11 IS IS7179A patent/IS7179A/is unknown
- 2004-03-18 CO CO04025929A patent/CO5560534A2/es not_active Application Discontinuation
- 2004-04-05 NO NO20041520A patent/NO20041520L/no unknown
- 2004-04-08 MA MA27623A patent/MA27075A1/fr unknown

Also Published As

Publication number	Publication date
ES2246017T3 (es)	2006-02-01
EP1434570B8 (en)	2005-10-26
MXPA04003293A (es)	2004-07-23
UY27477A1 (es)	2003-05-30
EA200400431A1 (ru)	2004-08-26
CO5560534A2 (es)	2005-09-30
HRP20040261A2 (en)	2004-08-31
AP2004003001A0 (en)	2004-03-31
DOP2002000464A (es)	2003-04-15
BR0213196A (pt)	2004-08-31
PL369666A1 (en)	2005-05-02
IL160969A0 (en)	2004-08-31
EP1434570B1 (en)	2005-08-31
SV2004001279A (es)	2004-02-19
CN1568180A (zh)	2005-01-19
IS7179A (is)	2004-03-11
NO20041520L (no)	2004-04-05
AR036782A1 (es)	2004-10-06
DE60205925T2 (de)	2006-06-08
CA2461168A1 (en)	2003-04-24
GT200200184A (es)	2003-05-23
DE60205925D1 (de)	2005-10-06
OA12709A (en)	2006-06-26
PE20030551A1 (es)	2003-06-26
HUP0600064A2 (en)	2006-06-28
EP1434570A1 (en)	2004-07-07
ATE303135T1 (de)	2005-09-15
EA006168B1 (ru)	2005-10-27
WO2003032956A1 (en)	2003-04-24
MA27075A1 (fr)	2004-12-20
GB0124455D0 (en)	2001-12-05
JP2005507909A (ja)	2005-03-24
PA8556001A1 (es)	2003-07-28
JP4131471B2 (ja)	2008-08-13
ZA200401976B (en)	2004-07-12
PY0223360A (es)	2004-04-01
HUP0600064A3 (en)	2007-02-28
KR20050032510A (ko)	2005-04-07

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