IS7179A - Lyfjafræðilegar samsetningar til leysnistýringar á 4-amínó-6,7-dímetoxý-2-(5-metansúlfónamídó-1,2,3,4,-tetrahýdróísókínól-2-ýl)-5-(2-pýridýl) kínasólíni - Google Patents

Lyfjafræðilegar samsetningar til leysnistýringar á 4-amínó-6,7-dímetoxý-2-(5-metansúlfónamídó-1,2,3,4,-tetrahýdróísókínól-2-ýl)-5-(2-pýridýl) kínasólíni

Info

Publication number
IS7179A
IS7179A IS7179A IS7179A IS7179A IS 7179 A IS7179 A IS 7179A IS 7179 A IS7179 A IS 7179A IS 7179 A IS7179 A IS 7179A IS 7179 A IS7179 A IS 7179A
Authority
IS
Iceland
Prior art keywords
tetrahydroisoquinol
methanesulfonamido
quinazoline
dimethoxy
pyridyl
Prior art date
Application number
IS7179A
Other languages
English (en)
Inventor
Douglas Davis John
John Humphrey Michael
James Macrae Ross
Sarah Smith Janet
Original Assignee
Pfizer Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc. filed Critical Pfizer Inc.
Publication of IS7179A publication Critical patent/IS7179A/is

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5026Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Urology & Nephrology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
IS7179A 2001-10-11 2004-03-11 Lyfjafræðilegar samsetningar til leysnistýringar á 4-amínó-6,7-dímetoxý-2-(5-metansúlfónamídó-1,2,3,4,-tetrahýdróísókínól-2-ýl)-5-(2-pýridýl) kínasólíni IS7179A (is)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0124455.7A GB0124455D0 (en) 2001-10-11 2001-10-11 Pharmaceutical formulations
PCT/IB2002/004040 WO2003032956A1 (en) 2001-10-11 2002-09-30 Pharmaceutical formulations for the controlled release of 4-amino-6,7-dimethoxy-2-(5-methanesulfonamido-1,2,3,4-tetrahydroisoquinol-2-yl)-5-(2-pyridyl) quinazoline

Publications (1)

Publication Number Publication Date
IS7179A true IS7179A (is) 2004-03-11

Family

ID=9923660

Family Applications (1)

Application Number Title Priority Date Filing Date
IS7179A IS7179A (is) 2001-10-11 2004-03-11 Lyfjafræðilegar samsetningar til leysnistýringar á 4-amínó-6,7-dímetoxý-2-(5-metansúlfónamídó-1,2,3,4,-tetrahýdróísókínól-2-ýl)-5-(2-pýridýl) kínasólíni

Country Status (33)

Country Link
EP (1) EP1434570B8 (is)
JP (1) JP4131471B2 (is)
KR (1) KR20050032510A (is)
CN (1) CN1568180A (is)
AP (1) AP2004003001A0 (is)
AR (1) AR036782A1 (is)
AT (1) ATE303135T1 (is)
BR (1) BR0213196A (is)
CA (1) CA2461168A1 (is)
CO (1) CO5560534A2 (is)
DE (1) DE60205925T2 (is)
DK (1) DK1434570T3 (is)
DO (1) DOP2002000464A (is)
EA (1) EA006168B1 (is)
ES (1) ES2246017T3 (is)
GB (1) GB0124455D0 (is)
GT (1) GT200200184A (is)
HR (1) HRP20040261A2 (is)
HU (1) HUP0600064A3 (is)
IL (1) IL160969A0 (is)
IS (1) IS7179A (is)
MA (1) MA27075A1 (is)
MX (1) MXPA04003293A (is)
NO (1) NO20041520L (is)
OA (1) OA12709A (is)
PA (1) PA8556001A1 (is)
PE (1) PE20030551A1 (is)
PL (1) PL369666A1 (is)
PY (1) PY0223360A (is)
SV (1) SV2004001279A (is)
UY (1) UY27477A1 (is)
WO (1) WO2003032956A1 (is)
ZA (1) ZA200401976B (is)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0317663D0 (en) * 2003-07-29 2003-09-03 Astrazeneca Ab Pharmaceutical composition
SG11201507258PA (en) 2013-03-14 2015-10-29 Amgen Inc Heterocyclic compounds and their uses
KR101943592B1 (ko) 2017-08-31 2019-01-30 조현우 데이터 마이닝 기법을 이용한 전자가계부 시스템

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2053120T3 (es) * 1990-07-02 1994-07-16 Bend Res Inc Perlas microporosas asimetricas para liberacion controlada.
FR2752737B1 (fr) * 1996-08-29 1998-10-02 Synthelabo Comprime a liberation controlee de chlorhydrate d'alfuzosine
GB9700504D0 (en) * 1997-01-11 1997-02-26 Pfizer Ltd Pharmaceutical compounds
IL141235A (en) * 2000-02-09 2012-04-30 Novartis Int Pharm Ltd Combined use of an alpha-adrenoceptor antagonist and a muscarinic antagonist in the preparation of a drug for the treatment of non-malignant prostatic hyperplasia
IL150634A0 (en) * 2000-03-03 2003-02-12 Pfizer 4-amino-6,7-dimethoxy-2-(5-methanesulfonamido-1,2,3,4-tetrahydroisoquinol-2-yl)-5-(2-pyridyl)quinazoline mesylate and polymorphs

Also Published As

Publication number Publication date
DOP2002000464A (es) 2003-04-15
UY27477A1 (es) 2003-05-30
PE20030551A1 (es) 2003-06-26
AP2004003001A0 (en) 2004-03-31
ATE303135T1 (de) 2005-09-15
GB0124455D0 (en) 2001-12-05
CA2461168A1 (en) 2003-04-24
JP4131471B2 (ja) 2008-08-13
GT200200184A (es) 2003-05-23
ES2246017T3 (es) 2006-02-01
MXPA04003293A (es) 2004-07-23
KR20050032510A (ko) 2005-04-07
EP1434570B1 (en) 2005-08-31
EP1434570A1 (en) 2004-07-07
IL160969A0 (en) 2004-08-31
DE60205925T2 (de) 2006-06-08
JP2005507909A (ja) 2005-03-24
WO2003032956A1 (en) 2003-04-24
MA27075A1 (fr) 2004-12-20
BR0213196A (pt) 2004-08-31
HUP0600064A2 (en) 2006-06-28
DE60205925D1 (de) 2005-10-06
PL369666A1 (en) 2005-05-02
ZA200401976B (en) 2004-07-12
HUP0600064A3 (en) 2007-02-28
EA006168B1 (ru) 2005-10-27
SV2004001279A (es) 2004-02-19
NO20041520L (no) 2004-04-05
CO5560534A2 (es) 2005-09-30
HRP20040261A2 (en) 2004-08-31
CN1568180A (zh) 2005-01-19
DK1434570T3 (da) 2005-11-07
EA200400431A1 (ru) 2004-08-26
OA12709A (en) 2006-06-26
AR036782A1 (es) 2004-10-06
EP1434570B8 (en) 2005-10-26
PA8556001A1 (es) 2003-07-28
PY0223360A (es) 2004-04-01

Similar Documents

Publication Publication Date Title
DK1292594T3 (da) Quinazolinderivater til behandling af tumorer
ATE446093T1 (de) Substituierte chinazolin-derivate als aurora- kinase inhibitoren
DK1762567T3 (da) Pyrazolderivater til behandling af HIV
NO20052497D0 (no) Fremgangsmater for selektiv inhibering av Janus tyrosinkinase 3 (JAK3).
IS6957A (is) Tatrat sölt af 5,8,14,-tríasatetrasýkló[10.3.1.02,11.04,9]-hexadeka-2(11),3,5,7,9,-pentaen og lyfjafræðilegar samsetningar af þeim
EE200200201A (et) Trüosiinkinaasi pärssiv ühend, seda sisaldav farmatseutiline kompositsioon ning raviotstarbeline kasutamine.
MXPA03008690A (es) Inhibidores novedosos de tirosina cinasa.
DZ3425A1 (fr) Derives de quinolinone en tant qu'inhibiteurs kinases de tyrosine
IL160714A0 (en) Heterocyclic substituted 2-(4-phenoxy) pyridine derivatives and pharmaceutical compositions containing the same
DK1326841T3 (da) Pyridinon-derivater til behandling af atherosklerose
IS7233A (is) Kínasólín afleiður til meðhöndlunar á afbrigðilegum frumuvexti
DK1202746T3 (da) NSAID- og EGFR-kinaseinhibitorerholdigt præparat til behandling eller inhibering af colonpolypper og colorektal cancer
DK1480983T3 (da) Heteroarylsubstituerede 2-pyridinyl- og 2-pyrimidinyl- 6,7,8,9-tetrahydropyrimido[1,2a]pyrimidin-4-onderivater
DK1408756T3 (da) Fremgangsmåde til bekæmpelse af ukrudt
EG24957A (en) Quinazoline derivatives as src tyrosine kinase inhibitors.
DK1458386T3 (da) Aroylpyrrolheteroaryl- og methanolforbindelser til behandling af en lidelse i centralnervesystemet
DK1475379T3 (da) Anvendelse af scopinesterderivater til fremstilling af lægemidler
IS7179A (is) Lyfjafræðilegar samsetningar til leysnistýringar á 4-amínó-6,7-dímetoxý-2-(5-metansúlfónamídó-1,2,3,4,-tetrahýdróísókínól-2-ýl)-5-(2-pýridýl) kínasólíni
NO20024195L (no) 4-amino-6,7-dimetoksy-2-(5-metansulfonamido-1,2,3,4- tetrahydroisoquinol-2-yl)-5-(2-pyridinyl)quinazolin-mesylat samtpolymorfer
ATA1092002A (de) Pflug
NO20040549L (no) Komplettering av laterale bronnboringer.
DK1451177T3 (da) Substituerede 2-pyrrolidin-2-yl-1H-indol-derivater til behandling af migræne
DE60225958D1 (de) Pflug
DE50201969D1 (de) Temperaturstabilisierte verstärkerschaltung
TH0001002776B (th) สารประกอบอินดาโซลและองค์ประกอบทางเภสัชภัณฑ์ในการยับยั้งโปรตีนไคเนสและวิธีใช้ประโยชน์