DK147855C - Analogifremgangsmaade til fremstilling af 3,4-dihydro-quinazolinderivatereller salte deraf - Google Patents

Analogifremgangsmaade til fremstilling af 3,4-dihydro-quinazolinderivatereller salte deraf

Info

Publication number
DK147855C
DK147855C DK546776A DK546776A DK147855C DK 147855 C DK147855 C DK 147855C DK 546776 A DK546776 A DK 546776A DK 546776 A DK546776 A DK 546776A DK 147855 C DK147855 C DK 147855C
Authority
DK
Denmark
Prior art keywords
dihydro
preparing
quinazoline derivatives
analogy procedure
derivatives salts
Prior art date
Application number
DK546776A
Other languages
Danish (da)
English (en)
Other versions
DK546776A (da
DK147855B (da
Inventor
Gianfederico Doria
Ciriaco Romeo
Piernicola Giraldi
Francesco Lauria
Maria Luisa Corno
Piero Sberze
Marcello Tibolla
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of DK546776A publication Critical patent/DK546776A/da
Publication of DK147855B publication Critical patent/DK147855B/da
Application granted granted Critical
Publication of DK147855C publication Critical patent/DK147855C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C07D239/91—Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C07D239/90—Oxygen atoms with acyclic radicals attached in position 2 or 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/93—Sulfur atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Immunology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK546776A 1975-12-05 1976-12-03 Analogifremgangsmaade til fremstilling af 3,4-dihydro-quinazolinderivatereller salte deraf DK147855C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT2999875 1975-12-05
IT29998/75A IT1050750B (it) 1975-12-05 1975-12-05 Derivati della 3.4 di idro chinazolina

Publications (3)

Publication Number Publication Date
DK546776A DK546776A (da) 1977-06-06
DK147855B DK147855B (da) 1984-12-24
DK147855C true DK147855C (da) 1985-06-10

Family

ID=11228830

Family Applications (1)

Application Number Title Priority Date Filing Date
DK546776A DK147855C (da) 1975-12-05 1976-12-03 Analogifremgangsmaade til fremstilling af 3,4-dihydro-quinazolinderivatereller salte deraf

Country Status (22)

Country Link
US (1) US4251531A (cs)
JP (1) JPS5271485A (cs)
AT (1) AT355029B (cs)
AU (1) AU505660B2 (cs)
BE (1) BE848696A (cs)
CA (1) CA1084051A (cs)
CH (2) CH626073A5 (cs)
CS (1) CS194786B2 (cs)
DE (1) DE2654215A1 (cs)
DK (1) DK147855C (cs)
FI (1) FI64359C (cs)
FR (1) FR2333511A1 (cs)
GB (1) GB1523081A (cs)
HU (1) HU177817B (cs)
IL (1) IL50849A (cs)
IT (1) IT1050750B (cs)
NL (1) NL7613450A (cs)
NO (1) NO146095C (cs)
NZ (1) NZ182778A (cs)
SE (1) SE7613588L (cs)
SU (1) SU786894A3 (cs)
ZA (1) ZA766745B (cs)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4419357A (en) 1982-01-18 1983-12-06 The Dow Chemical Company 3-(1H-Tetrazol-5-yl)-4(3H)-quinazolinones
IL69274A (en) * 1982-08-05 1986-08-31 Erba Farmitalia (substituted amino)derivatives of 3-benzylidene-pyrrolo(2,1-b)quinazolin-9-ones and 6-benzylidene-pyrido(2,1-b)quinazolin-11-ones,their preparation and pharmaceutical compositions containing them
US4666913A (en) * 1985-11-22 1987-05-19 William H. Rorer, Inc. Hydroxy and aminothiazolyl-benzodiazinone compounds, cardiotonic compositions including the same, and their uses
GB8827988D0 (en) * 1988-11-30 1989-01-05 Smith Kline French Lab Chemical compounds
US5430148A (en) * 1992-03-31 1995-07-04 Agouron Pharmaceuticals, Inc. Antiproliferative quinazolines
US6632961B1 (en) * 1998-05-22 2003-10-14 Abbott Laboratories Antiangiogenic drug to treat cancer, arthritis and retinopathy
CA2332535C (en) * 1998-05-22 2006-02-28 Abbott Laboratories Antiangiogenic drug to treat cancer, arthritis and retinopathy
CO5170498A1 (es) * 1999-05-28 2002-06-27 Abbott Lab Biaril sulfonamidas son utiles como inhibidores de proliferacion celular
US7893071B2 (en) * 2001-04-23 2011-02-22 University Of Virginia Patent Foundation Synthesis and evaluation of novel phthalimide mimics as anti-angiogenic
CN101152185B (zh) * 2003-06-06 2010-12-08 阿里克斯股份公司 杂环化合物作为scce抑制剂的用途
CN100518740C (zh) * 2003-06-06 2009-07-29 阿里克斯股份公司 杂环化合物作为scce抑制剂的制药用途
KR101419075B1 (ko) * 2006-08-08 2014-07-11 아스카 세이야쿠 가부시키가이샤 퀴나졸린 유도체
PT2118074E (pt) 2007-02-01 2014-03-20 Resverlogix Corp Compostos para a prevenção e tratamento de doenças cardiovasculares
NZ617779A (en) 2009-03-18 2015-08-28 Resverlogix Corp Novel anti-inflammatory agents
US9757368B2 (en) 2009-04-22 2017-09-12 Resverlogix Corp. Anti-inflammatory agents
CN114984016A (zh) 2015-03-13 2022-09-02 雷斯韦洛吉克斯公司 用于治疗补体相关疾病之组合物及治疗方法
GB201510254D0 (en) * 2015-06-12 2015-07-29 Syngenta Participations Ag Improvements in or relating to organic compounds
WO2020004594A1 (ja) * 2018-06-27 2020-01-02 株式会社リボルナバイオサイエンス 脊髄性筋萎縮症の予防または治療剤

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3696102A (en) 1970-03-09 1972-10-03 Pfizer & Co C Process for the synthesis of substituted quinazolin-4-ones
GB1301319A (cs) 1970-07-13 1972-12-29

Also Published As

Publication number Publication date
ATA894376A (de) 1979-07-15
NO146095B (no) 1982-04-19
ZA766745B (en) 1977-10-26
FI64359B (fi) 1983-07-29
IL50849A (en) 1980-11-30
SE7613588L (sv) 1977-06-06
FR2333511B1 (cs) 1979-03-02
AU1947276A (en) 1978-05-18
DK546776A (da) 1977-06-06
AU505660B2 (en) 1979-11-29
NL7613450A (nl) 1977-06-07
IL50849A0 (en) 1977-01-31
FR2333511A1 (fr) 1977-07-01
BE848696A (fr) 1977-03-16
NZ182778A (en) 1978-07-28
US4251531A (en) 1981-02-17
CS194786B2 (en) 1979-12-31
GB1523081A (en) 1978-08-31
DK147855B (da) 1984-12-24
CH626073A5 (cs) 1981-10-30
CH626075A5 (cs) 1981-10-30
FI763391A7 (cs) 1977-06-06
SU786894A3 (ru) 1980-12-07
HU177817B (en) 1981-12-28
JPS5271485A (en) 1977-06-14
NO146095C (no) 1982-08-11
NO764135L (cs) 1977-06-07
AT355029B (de) 1980-02-11
JPS5543464B2 (cs) 1980-11-06
IT1050750B (it) 1981-03-20
FI64359C (fi) 1983-11-10
CA1084051A (en) 1980-08-19
DE2654215A1 (de) 1977-06-16

Similar Documents

Publication Publication Date Title
DK298176A (da) Fremgangsmade til fremstilling af 1,4-dihydropyrinderivater
DK141845C (da) Analogifremgangsmaade til fremstilling af 2-acyl-4-oxo-pyrazino(2,1-a)isoquinolinderivater
DK145228C (da) Analogifremgangsmaade til fremstilling af 3-amino-4-deoxo-4-iminorifamycinderivater
DK148260C (da) Analogifremgangsmaade til fremstilling af 1,3,8-trisubstituerede xantinderivater eller salte deraf
DK143708C (da) Analogifremgangsmaade til fremstilling af 17alfa-acyloxy-9alfa,21-dihalogen-11beta-hydroxy-6alfa-fluor-16alfa-methyl-pregna-1,4-dien-3,20-dion-forbindelser
DK147068C (da) Analogifremgangsmaade til fremstilling af 1-naphthylmethyl-cinnamyl-aminderivater
DK144525C (da) Analogifremgangsmaade til fremstilling af 5-halogenpyrimid-2-oner eller salte deraf
DK144702C (da) Analogifremgangsmaade til fremstilling af 2,3-dihydro-imidazo(2,1-b)-thiazolderivater
DK5976A (da) Fremgangsmade til fremstilling af biphenyloxyderivater eller salte heraf
DK415676A (da) Fremgangsmade til fremstilling af pilocarpiniumsalte
DK153150C (da) Analogifremgangsmaade til fremstilling af 4-oxo-1,6,7,8-tetrahydro-4h-pyridooe1,2aaapyrimidinderivater
DK153489C (da) Analogifremgangsmaade til fremstilling af 7-aminothiazolylacetamidocephalosporansyrederivater
DK20077A (da) Fremgangsmade til fremstilling af salte af 3,3-dimethyl-2-oxo-smorsyre
DK150484C (da) Analogifremgangsmaade til fremstilling af 4-amino-3-thiophencarboxylsyrederivater
DK147623C (da) Analogifremgangsmaade til fremstilling af azapurinderivater eller salte deraf
DK153479C (da) Analogifremgangsmaade til fremstilling af 1,4-benzodiazepin-2-on-derivater
SE422579B (sv) Forfarande for framstellning av 4-oxo-hexahydro-pyrazino(2,1-a)isokinolinderivat
DK146822C (da) Analogifremgangsmaade til fremstilling af derivater af 4-desacetyl-vinblastin eller salte deraf
DK154888C (da) Analogifremgangsmaade til fremstilling af 6-substituerede-6-methoxypenicillansyrederivater
DK153843C (da) Analogifremgangsmaade til fremstilling af 5-substituerede 10,11-dihydro-5h-dibenzooea,daacyclohepten-5,10-iminer eller salte deraf
DK219776A (da) Fremgangsmade til fremstilling af 1,2-benzothiazin-oxadiazolforbindelse
DK150543C (da) Analogifremgangsmaade til fremstilling af 4-phenyl-3-oxo-1,2,4-oxadiazinderivater
DK146624C (da) Analogifremgangsmaade til fremstilling af 1-aminoalkyl-3,4-diphenyl-1h-pyrazoler
DK205676A (da) Fremgangsmade til fremstilling af 2-substituerede 1,4-benzodiazepinderivater
DK145060C (da) Analogifremgangsmaade til fremstilling af 6-acylamino-2,2-dimethyl-3-phosphonopenam-forbindelser eller salte deraf

Legal Events

Date Code Title Description
PBP Patent lapsed