DK149490D0 - Antiemetiske ergolinderivater - Google Patents

Antiemetiske ergolinderivater

Info

Publication number: DK149490D0
Authority: DK; Denmark
Prior art keywords: antiemetic; ergoline derivatives; ergoline; derivatives; antiemetic ergoline
Prior art date: 1988-10-21

Application number

DK149490A

Other languages

English (en)

Other versions

DK149490A (da

Inventor

Alessandro Rossi

Metilde Buonamici

Lorenzo Pergrassi

Enzo Brambilla

Original Assignee

Erba Carlo Spa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1988-10-21

Filing date

1990-06-19

Publication date

1990-06-19

1990-06-19 Application filed by Erba Carlo Spa filed Critical Erba Carlo Spa

1990-06-19 Publication of DK149490D0 publication Critical patent/DK149490D0/da

1990-08-16 Publication of DK149490A publication Critical patent/DK149490A/da

Links

AWFDCTXCTHGORH-HGHGUNKESA-N 6-[4-[(6ar,9r,10ar)-5-bromo-7-methyl-6,6a,8,9,10,10a-hexahydro-4h-indolo[4,3-fg]quinoline-9-carbonyl]piperazin-1-yl]-1-methylpyridin-2-one Chemical class O=C([C@H]1CN([C@H]2[C@@H](C=3C=CC=C4NC(Br)=C(C=34)C2)C1)C)N(CC1)CCN1C1=CC=CC(=O)N1C AWFDCTXCTHGORH-HGHGUNKESA-N 0.000 title 1
230000003474 anti-emetic effect Effects 0.000 title 1
239000002111 antiemetic agent Substances 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/48—Ergoline derivatives, e.g. lysergic acid, ergotamine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics

Landscapes

Health & Medical Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Epidemiology (AREA)
Otolaryngology (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Hospice & Palliative Care (AREA)
Engineering & Computer Science (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

DK149490A 1988-10-21 1990-06-19 Antiemetiske ergolinderivater DK149490A (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB888824744A GB8824744D0 (en)	1988-10-21	1988-10-21	Antiemesis ergoline derivatives
PCT/EP1989/001263 WO1990004396A1 (en)	1988-10-21	1989-10-20	Antiemesis ergoline derivatives

Publications (2)

Publication Number	Publication Date
DK149490D0 true DK149490D0 (da)	1990-06-19
DK149490A DK149490A (da)	1990-08-16

Family

ID=10645610

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK149490A DK149490A (da)	1988-10-21	1990-06-19	Antiemetiske ergolinderivater

Country Status (12)

Country	Link
US (1)	US5202325A (da)
EP (2)	EP0371246A1 (da)
JP (1)	JPH03502802A (da)
KR (1)	KR900701273A (da)
AU (1)	AU626358B2 (da)
CA (1)	CA2001004C (da)
DK (1)	DK149490A (da)
GB (1)	GB8824744D0 (da)
HU (1)	HU208077B (da)
IE (1)	IE63194B1 (da)
IL (1)	IL91999A0 (da)
WO (1)	WO1990004396A1 (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5364856A (en) *	1991-03-28	1994-11-15	Eli Lilly And Company	6-heterocyclic-4-amino-1,3,4,5-tetrahydrobenz[CD]indoles
US5347013A (en) *	1991-03-28	1994-09-13	Eli Lilly And Company	6-heterocyclic-4-amino-1,2,2a,3,4,5-hexahydrobenz[cd]indoles
US5648356A (en) *	1991-03-28	1997-07-15	Eli Lilly And Company	6-heterocyclic-4-amino-1,2,2a,3,4,5-hexahydrobenz[CD]indoles
EP0628042B1 (en) *	1992-12-24	2001-08-16	PHARMACIA & UPJOHN S.p.A.	Serotoninergic ergoline derivatives
EP1053752A1 (en)	1998-02-10	2000-11-22	Yoshitomi Pharmaceutical Industries, Ltd.	Preparations with controlled release

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
HU172479B (hu) *	1976-03-09	1978-09-28	Gyogyszerkutato Intezet	Sposob poluchenija novykh soedinenij s ehrgolenovymi i
DE3101535A1 (de) *	1981-01-14	1982-08-12	Schering Ag, 1000 Berlin Und 4619 Bergkamen	Neue (2-halogen-ergolinyl)-n'.n'-diethyl-harnstoffderivate, verfahren zu ihrer herstellung und deren verwendung als arzneimittel
HU197569B (en) *	1984-01-12	1989-04-28	Sandoz Ag	Process for producing 8alpha-acylaminoergoline derivatives and pharmaceuticals comprising such compounds
GB8501078D0 (en) *	1985-01-16	1985-02-20	Erba Farmitalia	Piperazin-1-yl-ergo-line derivatives
IL80193A0 (en) *	1985-10-01	1986-12-31	Lilly Co Eli	Esters of dihydrolysergic acid
US4713384A (en) *	1985-10-01	1987-12-15	Eli Lilly And Company	Selective method for blocking 5HT2 receptors

1988
- 1988-10-21 GB GB888824744A patent/GB8824744D0/en active Pending
1989
- 1989-10-16 IL IL91999A patent/IL91999A0/xx not_active IP Right Cessation
- 1989-10-19 CA CA002001004A patent/CA2001004C/en not_active Expired - Fee Related
- 1989-10-19 IE IE335889A patent/IE63194B1/en not_active IP Right Cessation
- 1989-10-20 JP JP2500032A patent/JPH03502802A/ja active Pending
- 1989-10-20 AU AU46336/89A patent/AU626358B2/en not_active Ceased
- 1989-10-20 EP EP89119544A patent/EP0371246A1/en active Pending
- 1989-10-20 US US07/499,413 patent/US5202325A/en not_active Expired - Fee Related
- 1989-10-20 KR KR1019900701311A patent/KR900701273A/ko not_active Ceased
- 1989-10-20 HU HU896835A patent/HU208077B/hu not_active IP Right Cessation
- 1989-10-20 WO PCT/EP1989/001263 patent/WO1990004396A1/en not_active Ceased
- 1989-10-20 EP EP89913149A patent/EP0418327B1/en not_active Expired - Lifetime
1990
- 1990-06-19 DK DK149490A patent/DK149490A/da not_active Application Discontinuation

Also Published As

Publication number	Publication date
CA2001004C (en)	1996-01-30
HU896835D0 (en)	1990-11-28
EP0371246A1 (en)	1990-06-06
IE893358L (en)	1990-04-21
US5202325A (en)	1993-04-13
AU4633689A (en)	1990-05-14
GB8824744D0 (en)	1988-11-30
HU208077B (en)	1993-08-30
KR900701273A (ko)	1990-12-01
JPH03502802A (ja)	1991-06-27
HUT54049A (en)	1991-01-28
EP0418327B1 (en)	1993-05-26
WO1990004396A1 (en)	1990-05-03
CA2001004A1 (en)	1990-04-21
DK149490A (da)	1990-08-16
AU626358B2 (en)	1992-07-30
IL91999A0 (en)	1990-07-12
EP0418327A1 (en)	1991-03-27
IE63194B1 (en)	1995-04-05

Legal Events

Date	Code	Title	Description
1997-06-16	AHB	Application shelved due to non-payment

Publication	Publication Date	Title
TR26815A (tr)	1994-08-09	Azolilmetil-sikropil türevleri
DE68927948D1 (de)	1997-05-15	Trehalosderivate
DE68925161D1 (de)	1996-02-01	Alkylavermectin-Derivate
DK491389A (da)	1990-04-07	Substituerede 9h-purinderivater
DE68927610D1 (de)	1997-02-13	Antikörper-Arzneimittel Konjugale
DK19789A (da)	1989-07-21	Dehydrocholcalciferolderivater
TR24894A (tr)	1992-07-20	N-FENILPIRAZOL TüREVLERI
DK507188A (da)	1989-03-15	Cholecalciferolderivater
DE68927657D1 (de)	1997-02-27	Butynylaminderivate
DK486089D0 (da)	1989-10-03	Pyranobenzoxadiazolderivater
DK378088D0 (da)	1988-07-07	Alkenderivater
DK49688D0 (da)	1988-02-01	Propiolophenonderivater
DK81989A (da)	1989-08-26	Substituerede quinolinderivater
DK82189A (da)	1989-08-26	Substituerede quinolinderivater
FI895871A7 (fi)	1990-06-10	Uusia bentsopyranyylipyrrolinonijohdannaisia
DK35787D0 (da)	1987-01-22	Ergolinderivater
ATA48389A (de)	1995-04-15	Antiemetikum
DK271088A (da)	1988-11-20	Tienopyridinderivater
DK160389A (da)	1989-10-05	Aryldionderivater
DK149490A (da)	1990-08-16	Antiemetiske ergolinderivater
FI893041A7 (fi)	1989-06-21	Substituoidut atsasykloheksyylijohdannaiset
ATA155589A (de)	1994-02-15	Mitomycinphosphat-derivate
DK695788A (da)	1989-06-18	Naphtalenderivater
DK324489D0 (da)	1989-06-29	Substituerede azacyclohexylderivater
DK82089D0 (da)	1989-02-22	Substituerede quinolinderivater