DK158670C - Fremgangsmaade til fremstilling af 6beta-halogensubstituerede penicillansyrederivater - Google Patents

Fremgangsmaade til fremstilling af 6beta-halogensubstituerede penicillansyrederivater

Info

Publication number: DK158670C
Authority: DK; Denmark
Prior art keywords: 6beta; halogen; procedure; preparation; acid derivatives
Prior art date: 1979-05-21

Application number

DK562589A

Other languages

English (en)

Other versions

DK562589D0 (da

DK562589A (da

DK158670B (da

Inventor

Welf Von Daehne

Original Assignee

Leo Pharm Prod Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1979-05-21

Filing date

1989-11-10

Publication date

1991-01-07

1989-11-10 Application filed by Leo Pharm Prod Ltd filed Critical Leo Pharm Prod Ltd

1989-11-10 Publication of DK562589D0 publication Critical patent/DK562589D0/da

1989-11-10 Publication of DK562589A publication Critical patent/DK562589A/da

1990-07-02 Publication of DK158670B publication Critical patent/DK158670B/da

1991-01-07 Application granted granted Critical

1991-01-07 Publication of DK158670C publication Critical patent/DK158670C/da

Links

RBKMMJSQKNKNEV-RITPCOANSA-N penicillanic acid Chemical class OC(=O)[C@H]1C(C)(C)S[C@@H]2CC(=O)N21 RBKMMJSQKNKNEV-RITPCOANSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DK562589A 1979-05-21 1989-11-10 Fremgangsmaade til fremstilling af 6beta-halogensubstituerede penicillansyrederivater DK158670C (da)

Applications Claiming Priority (8)

Application Number	Priority Date	Filing Date	Title
GB7917665		1979-05-21
GB7917665		1979-05-21
GB7930819		1979-09-05
GB7930819		1979-09-05
GB7941252		1979-11-29
GB7941252		1979-11-29
GB8006681		1980-02-27
GB8006681		1980-02-27

Publications (4)

Publication Number	Publication Date
DK562589D0 DK562589D0 (da)	1989-11-10
DK562589A DK562589A (da)	1989-11-10
DK158670B DK158670B (da)	1990-07-02
DK158670C true DK158670C (da)	1991-01-07

Family

ID=27449123

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
DK218580A DK158669C (da)	1979-05-21	1980-05-20	Fremgangsmaade til fremstilling af 6beta-halogensubstituerede penicillansyrederivater.
DK562589A DK158670C (da)	1979-05-21	1989-11-10	Fremgangsmaade til fremstilling af 6beta-halogensubstituerede penicillansyrederivater

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
DK218580A DK158669C (da)	1979-05-21	1980-05-20	Fremgangsmaade til fremstilling af 6beta-halogensubstituerede penicillansyrederivater.

Country Status (19)

Country	Link
US (3)	US4446144A (da)
JP (1)	JPS55154977A (da)
AU (3)	AU534754B2 (da)
BE (1)	BE883390A (da)
CA (1)	CA1265787A (da)
DE (3)	DE3051037C2 (da)
DK (2)	DK158669C (da)
FI (1)	FI801618A7 (da)
FR (2)	FR2457294A1 (da)
GR (1)	GR68372B (da)
IE (2)	IE49768B1 (da)
IL (1)	IL59948A0 (da)
IT (1)	IT1133091B (da)
LU (1)	LU82468A1 (da)
NL (1)	NL8002911A (da)
NZ (1)	NZ193597A (da)
PH (2)	PH17959A (da)
PT (1)	PT71273A (da)
SE (3)	SE452465B (da)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4432970A (en) *	1979-11-23	1984-02-21	Pfizer Inc.	6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors
IE51846B1 (en) *	1980-11-17	1987-04-15	Leo Pharm Prod Ltd	Pharmaceutical preparation for veterinary use and an appliance containing it
US4521533A (en) *	1984-07-12	1985-06-04	Pfizer Inc.	Salts of 6-alpha-(aminomethyl)penicillanic acid 1,1-dioxide esters and beta-lactam antibiotics
GB8522156D0 (en) *	1985-09-06	1985-10-09	Leo Pharm Prod Ltd	Producing chemical compounds
US5589354A (en) *	1994-12-20	1996-12-31	Biopure Corporation	Halogenation of cephalexin with haloperoxidase from Rathayibacter biopuresis
US5695951A (en) *	1994-12-20	1997-12-09	Biopure Corporation	Chlorination of cephalexin with chloroperoxidase from Rathayibacter biopuresis
DK0971690T4 (da)	1996-12-18	2015-07-13	Bimeda Res & Dev Ltd	Antiinfektionsmiddelfri intramammal veterinærsammensætning.
US20020035107A1 (en) *	2000-06-20	2002-03-21	Stefan Henke	Highly concentrated stable meloxicam solutions
PL208585B1 (pl) *	2002-10-25	2011-05-31	Intervet Int Bv	Kompozycja farmaceutyczna o przedłużonym uwalnianiu zawierająca cefquinom, sposób jej wytwarzania i zastosowanie cefquinomu
EP1568369A1 (en)	2004-02-23	2005-08-31	Boehringer Ingelheim Vetmedica Gmbh	Use of meloxicam for the treatment of respiratory diseases in pigs
DE102004025324A1 (de) *	2004-05-19	2005-12-08	Boehringer Ingelheim Vetmedica Gmbh	Flüssige Zubereitung für die Veterinärmedizin, Verfahren zu deren Herstellung und deren Verwendung
US9452155B2 (en)	2012-07-17	2016-09-27	Bayer New Zealand Ltd	Injectable antibiotic formulations and their methods of use
PL2874624T3 (pl) *	2012-07-17	2020-07-27	Bayer New Zealand Limited 3 Argus Place Hillcrest, Auckland 0627 / NZ	Wstrzykiwalne formulacje antybiotykowe i sposoby ich zastosowania
ES2729328T3 (es) *	2012-12-20	2019-10-31	Alleva Animal Health Ltd	Formulaciones inyectables veterinarias de penetamato
EP4265241A1 (en) *	2022-04-20	2023-10-25	Bilim Ilac Sanayii Ve Ticaret A.S.	Tablet formulations for the treatment of urinary system infections and method for the preparation of such formulations

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3206469A (en) *	1961-08-15	1965-09-14	Lepetit Spa	6-halopenicillanic acid
GB1297555A (da) *	1970-09-22	1972-11-22
GB1377817A (en) *	1971-06-09	1974-12-18	Beecham Group Ltd	Penicillins and cephalosporins
US4234579A (en) *	1977-06-07	1980-11-18	Pfizer Inc.	Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
IN149747B (da) *	1977-06-07	1982-04-03	Pfizer
US4180506A (en) *	1978-01-18	1979-12-25	Rex Pratt	6β-Bromo penicillanic acid
US4203992A (en) *	1978-12-11	1980-05-20	E. R. Squibb & Sons, Inc.	β-Bromopenicillanic acid sulfone
CA1158639A (en) *	1978-12-11	1983-12-13	Eric M. Gordon	6-bromopenicillanic acid sulfone
EP0013617B1 (en) *	1979-01-10	1984-07-04	Beecham Group Plc	Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
IL59081A0 (en) *	1979-01-10	1980-05-30	Schering Corp	2-penem compounds and a method for preparing them
US4518530A (en) *	1979-03-05	1985-05-21	Pfizer Inc.	6-β-Substituted penicillanic acids as β-lactamase inhibitors
US4397783A (en) *	1979-03-05	1983-08-09	Pfizer Inc.	Process for converting 6,6-disubstituted penicillanic acid derivatives to the 6-β-congeners
US4287181A (en) *	1979-10-22	1981-09-01	Pfizer Inc.	Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors
US4432970A (en) *	1979-11-23	1984-02-21	Pfizer Inc.	6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors

1980
- 1980-04-29 IE IE868/80A patent/IE49768B1/en not_active IP Right Cessation
- 1980-04-29 IE IE2559/84A patent/IE49770B1/en unknown
- 1980-04-29 IL IL59948A patent/IL59948A0/xx unknown
- 1980-05-01 NZ NZ193597A patent/NZ193597A/en unknown
- 1980-05-05 PH PH23982A patent/PH17959A/en unknown
- 1980-05-12 GR GR61906A patent/GR68372B/el unknown
- 1980-05-19 SE SE8003722A patent/SE452465B/sv not_active IP Right Cessation
- 1980-05-20 BE BE0/200687A patent/BE883390A/fr not_active IP Right Cessation
- 1980-05-20 DE DE19803051037 patent/DE3051037C2/de not_active Expired
- 1980-05-20 IT IT67790/80A patent/IT1133091B/it active
- 1980-05-20 PT PT71273A patent/PT71273A/pt unknown
- 1980-05-20 DE DE19803019244 patent/DE3019244A1/de active Granted
- 1980-05-20 DK DK218580A patent/DK158669C/da not_active IP Right Cessation
- 1980-05-20 JP JP6768580A patent/JPS55154977A/ja active Granted
- 1980-05-20 AU AU58584/80A patent/AU534754B2/en not_active Ceased
- 1980-05-20 LU LU82468A patent/LU82468A1/fr unknown
- 1980-05-20 CA CA000352237A patent/CA1265787A/en not_active Expired - Lifetime
- 1980-05-20 FI FI801618A patent/FI801618A7/fi not_active Application Discontinuation
- 1980-05-20 FR FR8011263A patent/FR2457294A1/fr active Granted
- 1980-05-20 NL NL8002911A patent/NL8002911A/nl not_active Application Discontinuation
- 1980-05-20 DE DE19803051038 patent/DE3051038C2/de not_active Expired
- 1980-11-17 US US06/207,614 patent/US4446144A/en not_active Expired - Lifetime
1982
- 1982-03-04 FR FR8203636A patent/FR2499575A1/fr active Granted
1983
- 1983-08-26 AU AU18486/83A patent/AU541322B2/en not_active Ceased
- 1983-08-26 PH PH29453A patent/PH19005A/en unknown
- 1983-08-26 AU AU18487/83A patent/AU541323B2/en not_active Ceased
- 1983-12-23 US US06/564,901 patent/US4594246A/en not_active Expired - Fee Related
1984
- 1984-12-06 SE SE8406201A patent/SE462096B/sv not_active IP Right Cessation
- 1984-12-06 SE SE8406202A patent/SE462097B/sv not_active IP Right Cessation
1986
- 1986-03-31 US US06/845,941 patent/US4672114A/en not_active Expired - Fee Related
1989
- 1989-11-10 DK DK562589A patent/DK158670C/da not_active IP Right Cessation

Also Published As

Publication number	Publication date
DK562589D0 (da)	1989-11-10
BE883390A (fr)	1980-11-20
FR2499575B1 (da)	1985-03-01
DK562589A (da)	1989-11-10
AU1848783A (en)	1983-12-22
SE452465B (sv)	1987-11-30
SE462096B (sv)	1990-05-07
DE3019244A1 (de)	1980-12-04
AU541322B2 (en)	1985-01-03
PH17959A (en)	1985-02-20
SE8406202D0 (sv)	1984-12-06
IE49768B1 (en)	1985-12-11
SE8406202L (sv)	1984-12-06
NZ193597A (en)	1985-04-30
LU82468A1 (fr)	1980-12-16
SE8003722L (sv)	1980-11-22
DE3051038C2 (da)	1989-04-13
GR68372B (da)	1981-12-28
PH19005A (en)	1985-12-03
IT8067790A0 (it)	1980-05-20
IE842559L (en)	1980-11-21
AU541323B2 (en)	1985-01-03
IE800868L (en)	1980-11-21
DE3019244C2 (da)	1989-04-06
DK218580A (da)	1980-11-22
AU534754B2 (en)	1984-02-16
AU1848683A (en)	1983-12-22
DE3051037C2 (da)	1989-03-30
US4446144A (en)	1984-05-01
IT1133091B (it)	1986-07-09
FR2457294B1 (da)	1984-01-13
US4672114A (en)	1987-06-09
NL8002911A (nl)	1980-11-25
JPS55154977A (en)	1980-12-02
DK158670B (da)	1990-07-02
CA1265787A (en)	1990-02-13
SE8406201D0 (sv)	1984-12-06
JPH0140837B2 (da)	1989-08-31
DK158669B (da)	1990-07-02
SE8406201L (sv)	1984-12-06
FR2457294A1 (fr)	1980-12-19
US4594246A (en)	1986-06-10
IL59948A0 (en)	1980-06-30
IE49770B1 (en)	1985-12-11
PT71273A (en)	1980-06-01
AU5858480A (en)	1980-11-27
DE3051038A1 (da)	1986-03-20
DK158669C (da)	1991-01-21
SE462097B (sv)	1990-05-07
FI801618A7 (fi)	1981-01-01
FR2499575A1 (fr)	1982-08-13

Legal Events

Date	Code	Title	Description
1996-01-22	PBP	Patent lapsed

Publication	Publication Date	Title
DK46079A (da)	1979-08-07	Fremgangsmaade til fremstilling af alkylendiaminderivater
DK129578A (da)	1978-09-26	Fremgangsmaade til fremstilling af oximderivater af 3-acetoxymethyl-7-aminothiazolylacetamidocephalosporansyre
DK266479A (da)	1980-02-04	Fremgangsmaade til fremstilling af 3-aminopropoxyarylderivater
DK303079A (da)	1980-01-27	Fremgangsmaade til fremstilling af imidazolderivater
DK77679A (da)	1979-08-23	Fremgangsmaade til fremstilling af hidtil ukendte propanonderivater
DK377680A (da)	1981-03-07	Fremgangsmaade til fremstilling af kanelsyrederivater
DK310779A (da)	1980-02-29	Fremgangsmaade til fremstilling af pyrimidinonderivater
DK562589D0 (da)	1989-11-10	Fremgangsmaade til fremstilling af 6beta-halogensubstituerede penicillansyrederivater
DK186179A (da)	1979-12-10	Fremgangsmaade til fremstilling af carbapenemderivater
DK129678A (da)	1978-09-26	Fremgangsmaade til fremstilling af oximderivater af 7-aminothiazolylacetamidocephalosporansyre
DK20279A (da)	1979-07-19	Fremgangsmaade til fremstilling af 4-pyridon-3-carboxylsyrederivater
DK415379A (da)	1980-04-05	Fremgangsmaade til fremstilling af chromanolderivater
DK34781A (da)	1981-07-29	Fremgangsmaade til fremstilling af phenylalkansyrederivater
DK12477A (da)	1977-07-15	Fremgangsmade til fremstilling af 7-aminothiazolylacetamidocephalosporansyrederivater
DK331679A (da)	1980-02-09	Fremgangsmaade til fremstilling af phenylalkansyrederivater
DK512379A (da)	1980-06-08	Fremgangsmaade til chlorering af pyridinderivater
DK257779A (da)	1979-12-22	Fremgangsmaade til fremstilling af chlor-styryl-cyclopropan-carboxylsyrederivater
DK73379A (da)	1979-08-22	Fremgangsmaade til fremstilling af halogensubstituerede mercaptoacylaminsyrer
DK68978A (da)	1978-08-19	Fremgangsmaade til fremstilling af oximderivater af 3-thiadiazolythiomethyl-7-aminothiazolylacetamidocephalosporansyre
DK160281C (da)	1991-07-29	Fremgangsmaade til fremstilling af steroid-s-thioesterderivater
DK282379A (da)	1980-01-06	Fremgangsmaade til fremstilling af phenylpiperidinderivater isaer substituerede eventuelt enkeltmaettede 1-benzylphenylpiperidiner
DK150879A (da)	1979-10-15	Fremgangsmaade til fremstilling af oximderivater af 3-azidomethyl-7-aminothiazolylacetamidocephalosporansyre
DK424080A (da)	1981-04-12	Fremgangsmaade til fremstilling af penicillansyrederivater
DK428079A (da)	1980-04-12	Fremgangsmaade til fremstilling af cyclohexadienderivater
DK348179A (da)	1980-02-22	Fremgangsmaade til fremstilling af carbazolyderivater