DK168524B1 - Fremgangsmåde til fremstilling af 23-desoxy-makrolidforbindelser - Google Patents

Fremgangsmåde til fremstilling af 23-desoxy-makrolidforbindelser Download PDF

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Publication number
DK168524B1
DK168524B1 DK504788A DK504788A DK168524B1 DK 168524 B1 DK168524 B1 DK 168524B1 DK 504788 A DK504788 A DK 504788A DK 504788 A DK504788 A DK 504788A DK 168524 B1 DK168524 B1 DK 168524B1
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DK
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Prior art keywords
compound
formula
group
prepared
solvent
Prior art date
Application number
DK504788A
Other languages
Danish (da)
English (en)
Other versions
DK504788A (da
DK504788D0 (da
Inventor
Michael V J Ramsay
Anthony H Shingler
Simon C Dolan
Stephen Freeman
Oswy Z Pereira
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of DK504788D0 publication Critical patent/DK504788D0/da
Publication of DK504788A publication Critical patent/DK504788A/da
Application granted granted Critical
Publication of DK168524B1 publication Critical patent/DK168524B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Cephalosporin Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Physical Or Chemical Processes And Apparatus (AREA)
DK504788A 1987-09-11 1988-09-09 Fremgangsmåde til fremstilling af 23-desoxy-makrolidforbindelser DK168524B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8721373 1987-09-11
GB878721373A GB8721373D0 (en) 1987-09-11 1987-09-11 Chemical process

Publications (3)

Publication Number Publication Date
DK504788D0 DK504788D0 (da) 1988-09-09
DK504788A DK504788A (da) 1989-03-12
DK168524B1 true DK168524B1 (da) 1994-04-11

Family

ID=10623610

Family Applications (1)

Application Number Title Priority Date Filing Date
DK504788A DK168524B1 (da) 1987-09-11 1988-09-09 Fremgangsmåde til fremstilling af 23-desoxy-makrolidforbindelser

Country Status (17)

Country Link
EP (1) EP0307221B1 (de)
JP (1) JPH01163182A (de)
KR (1) KR890005116A (de)
AT (1) ATE90101T1 (de)
AU (1) AU621063B2 (de)
BR (1) BR8804664A (de)
CA (1) CA1333600C (de)
DD (1) DD274421A5 (de)
DE (1) DE3881458T2 (de)
DK (1) DK168524B1 (de)
ES (1) ES2040863T3 (de)
GB (1) GB8721373D0 (de)
HU (2) HU203353B (de)
IE (1) IE62759B1 (de)
NZ (1) NZ226118A (de)
PT (1) PT88468B (de)
ZA (1) ZA886739B (de)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4429209A (en) * 1981-10-19 1984-01-31 Duro Dyne Corporation Resistance welding pin
ES8802229A1 (es) * 1985-04-30 1988-04-16 Glaxo Group Ltd Un procedimiento para preparar nuevos derivados lactonicos macrociclicos.
DE3782481T2 (de) * 1986-09-12 1993-05-19 American Cyanamid Co 23-deoxy-derivate von ll-f28249-verbindungen.
US4806527A (en) * 1987-03-16 1989-02-21 Merck & Co., Inc. Avermectin derivatives

Also Published As

Publication number Publication date
GB8721373D0 (en) 1987-10-21
HU203353B (en) 1991-07-29
ES2040863T3 (es) 1993-11-01
DE3881458D1 (de) 1993-07-08
DE3881458T2 (de) 1993-10-14
PT88468A (pt) 1988-10-01
DK504788A (da) 1989-03-12
DK504788D0 (da) 1988-09-09
EP0307221A3 (en) 1989-10-25
PT88468B (pt) 1992-11-30
KR890005116A (ko) 1989-05-11
BR8804664A (pt) 1989-04-18
IE882745L (en) 1989-03-11
EP0307221B1 (de) 1993-06-02
AU621063B2 (en) 1992-03-05
ZA886739B (en) 1989-08-30
IE62759B1 (en) 1995-02-22
JPH01163182A (ja) 1989-06-27
HU207085B (en) 1993-03-01
AU2208988A (en) 1989-03-16
CA1333600C (en) 1994-12-20
HUT48258A (en) 1989-05-29
HU903199D0 (en) 1990-10-28
DD274421A5 (de) 1989-12-20
NZ226118A (en) 1989-12-21
EP0307221A2 (de) 1989-03-15
ATE90101T1 (de) 1993-06-15

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PBP Patent lapsed