DK1691808T3 - Farmeceutisk sammensætning til oral indgivelse af et pyrazol-3-carboxamid - Google Patents

Farmeceutisk sammensætning til oral indgivelse af et pyrazol-3-carboxamid

Info

Publication number
DK1691808T3
DK1691808T3 DK04805418T DK04805418T DK1691808T3 DK 1691808 T3 DK1691808 T3 DK 1691808T3 DK 04805418 T DK04805418 T DK 04805418T DK 04805418 T DK04805418 T DK 04805418T DK 1691808 T3 DK1691808 T3 DK 1691808T3
Authority
DK
Denmark
Prior art keywords
carboxamide
pyrazole
pharmaceutical composition
oral administration
oral
Prior art date
Application number
DK04805418T
Other languages
Danish (da)
English (en)
Inventor
Thierry Breul
Jean Claude Gautier
Olivier Saslawski
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Application granted granted Critical
Publication of DK1691808T3 publication Critical patent/DK1691808T3/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Dispersion Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK04805418T 2003-11-10 2004-11-09 Farmeceutisk sammensætning til oral indgivelse af et pyrazol-3-carboxamid DK1691808T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0313259A FR2861992B1 (fr) 2003-11-10 2003-11-10 Composition pharmaceutique destinee a l'administration orale d'un derive de pyrazole-3-carboxamide.
PCT/FR2004/002875 WO2005046690A1 (fr) 2003-11-10 2004-11-09 Composition pharmaceutique destinee a l'administration orale d'un derive de pyrazole-3­carboxamide

Publications (1)

Publication Number Publication Date
DK1691808T3 true DK1691808T3 (da) 2009-08-03

Family

ID=34508418

Family Applications (1)

Application Number Title Priority Date Filing Date
DK04805418T DK1691808T3 (da) 2003-11-10 2004-11-09 Farmeceutisk sammensætning til oral indgivelse af et pyrazol-3-carboxamid

Country Status (27)

Country Link
US (2) US20060264469A1 (de)
EP (1) EP1691808B1 (de)
JP (1) JP4767171B2 (de)
KR (1) KR20060108668A (de)
CN (1) CN100528158C (de)
AR (1) AR047237A1 (de)
AT (1) ATE429227T1 (de)
AU (1) AU2004289086A1 (de)
BR (1) BRPI0416341A (de)
CA (1) CA2544413A1 (de)
CY (1) CY1110478T1 (de)
DE (1) DE602004020797D1 (de)
DK (1) DK1691808T3 (de)
ES (1) ES2325373T3 (de)
FR (1) FR2861992B1 (de)
HR (1) HRP20090393T1 (de)
IL (1) IL175556A (de)
MA (1) MA28419B1 (de)
NO (1) NO20062609L (de)
NZ (1) NZ547763A (de)
PL (1) PL1691808T3 (de)
PT (1) PT1691808E (de)
RU (1) RU2321404C1 (de)
SI (1) SI1691808T1 (de)
TW (1) TWI280129B (de)
WO (1) WO2005046690A1 (de)
ZA (1) ZA200604451B (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1880715A1 (de) * 2006-07-19 2008-01-23 Abbott GmbH & Co. KG Pharmazeutisch annehmbare lösungsvermittelnde Zusammensetzung und diese enthaltende pharmazeutische Darreichungsform
EP1920767A1 (de) * 2006-11-09 2008-05-14 Abbott GmbH & Co. KG Schmelzverarbeitete Darreichungsform mit Imatinib
US8536208B2 (en) * 2007-08-21 2013-09-17 Basilea Pharmaceutica Ag Antifungal composition
MY158809A (en) * 2010-09-22 2016-11-15 Craun Res Sdn Bhd Pharmaceutical compositions for calanolides, their derivatives and analogues, and process for producing the same
US20130317117A1 (en) * 2010-11-24 2013-11-28 Pharmaceutics International, Inc. Self micro-emulsifying drug delivery system with increased bioavailability

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5059691A (en) * 1990-01-22 1991-10-22 American Cyanamid Company N-((dialkylamino)methylene)-substituted pyrazolo (1,5-A)-pyrimidine-3-carboxamides and N-((dialkylamino)methylene)-substituted-4,5-dihydropyrazolo-(1,5-A)-pyrimidine-3-carboxamides
FR2692575B1 (fr) * 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
SI1033128T2 (sl) * 1993-09-28 2012-02-29 Scherer Gmbh R P Izdelava mehke Ĺľelatinaste kapsule
GB9405304D0 (en) * 1994-03-16 1994-04-27 Scherer Ltd R P Delivery systems for hydrophobic drugs
JPH11504028A (ja) * 1995-04-24 1999-04-06 イースム リサーチ ディベロップメント カンパニー オブ ザ ヒーブル ユニバーシティ オブ エルサレム 油/水エマルジョンを作り出す自己乳化性配合物
WO1996036316A1 (en) * 1995-05-19 1996-11-21 Abbott Laboratories Self-emulsifying formulations of lipophilic drugs
US5993858A (en) * 1996-06-14 1999-11-30 Port Systems L.L.C. Method and formulation for increasing the bioavailability of poorly water-soluble drugs
US6197774B1 (en) * 1997-03-14 2001-03-06 Otsuka Pharmaceutical Co., Ltd. Pyrimidine derivative
FR2761266B1 (fr) * 1997-03-28 1999-07-02 Sanofi Sa Composition pharmaceutique formee par granulation humide pour l'administration orale d'un derive du n-piperidino-3- pyrazolecarboxamide, de ses sels et de leurs solvates
FR2761265B1 (fr) * 1997-03-28 1999-07-02 Sanofi Sa Composition pharmaceutique pour l'administration orale d'un derive du n-piperidino-3-pyrazolecarboxamide, de ses sels et de leurs solvates
US6617426B1 (en) * 1999-06-22 2003-09-09 Merck & Co Inc Cysteinyl protease inhibitors
JP2001151669A (ja) * 1999-11-24 2001-06-05 Nippon Kayaku Co Ltd 経口用自己乳化製剤
GEP20053427B (en) * 1999-12-23 2005-01-25 Pfizer Prod Inc Pharmaceutical Compositions Providing Enhanced Drug Concentrations
GB0001928D0 (en) * 2000-01-27 2000-03-22 Novartis Ag Organic compounds
FR2831883B1 (fr) * 2001-11-08 2004-07-23 Sanofi Synthelabo Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant
ES2283756T3 (es) * 2002-03-01 2007-11-01 Novagali Pharma Sa Sistemas autoemulsionantes de administracion de farmaco para taxoides.
GB0216700D0 (en) * 2002-07-18 2002-08-28 Astrazeneca Ab Process

Also Published As

Publication number Publication date
ES2325373T3 (es) 2009-09-02
NO20062609L (no) 2006-06-06
EP1691808B1 (de) 2009-04-22
CN100528158C (zh) 2009-08-19
BRPI0416341A (pt) 2007-02-27
HK1102021A1 (en) 2007-11-02
NZ547763A (en) 2009-08-28
PT1691808E (pt) 2009-07-14
ATE429227T1 (de) 2009-05-15
JP2007516960A (ja) 2007-06-28
FR2861992B1 (fr) 2007-07-20
RU2321404C1 (ru) 2008-04-10
DE602004020797D1 (de) 2009-06-04
SI1691808T1 (sl) 2009-10-31
IL175556A (en) 2010-11-30
HRP20090393T1 (en) 2009-08-31
CY1110478T1 (el) 2015-04-29
IL175556A0 (en) 2008-04-13
FR2861992A1 (fr) 2005-05-13
KR20060108668A (ko) 2006-10-18
MA28419B1 (fr) 2007-02-01
RU2006120447A (ru) 2007-12-20
PL1691808T3 (pl) 2009-09-30
US20090004261A1 (en) 2009-01-01
US20060264469A1 (en) 2006-11-23
JP4767171B2 (ja) 2011-09-07
CA2544413A1 (fr) 2005-05-26
AR047237A1 (es) 2006-01-11
EP1691808A1 (de) 2006-08-23
ZA200604451B (en) 2007-10-31
AU2004289086A1 (en) 2005-05-26
WO2005046690A1 (fr) 2005-05-26
TWI280129B (en) 2007-05-01
TW200524597A (en) 2005-08-01
CN1925856A (zh) 2007-03-07

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