DK181285A - Heterocycliske bornanderivater, fremgangsmaade til fremstilling deraf og laegemiddel indeholdende saadanne forbindelser - Google Patents

Heterocycliske bornanderivater, fremgangsmaade til fremstilling deraf og laegemiddel indeholdende saadanne forbindelser Download PDF

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Publication number
DK181285A
DK181285A DK181285A DK181285A DK181285A DK 181285 A DK181285 A DK 181285A DK 181285 A DK181285 A DK 181285A DK 181285 A DK181285 A DK 181285A DK 181285 A DK181285 A DK 181285A
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DK
Denmark
Prior art keywords
compounds
bornand
heterocyclic
procedures
derivatives
Prior art date
Application number
DK181285A
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English (en)
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DK160832C (da
DK160832B (da
DK181285D0 (da
Inventor
Andre Esanu
Original Assignee
Scras
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Scras filed Critical Scras
Publication of DK181285D0 publication Critical patent/DK181285D0/da
Publication of DK181285A publication Critical patent/DK181285A/da
Publication of DK160832B publication Critical patent/DK160832B/da
Application granted granted Critical
Publication of DK160832C publication Critical patent/DK160832C/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • E—FIXED CONSTRUCTIONS
    • E04—BUILDING
    • E04H—BUILDINGS OR LIKE STRUCTURES FOR PARTICULAR PURPOSES; SWIMMING OR SPLASH BATHS OR POOLS; MASTS; FENCING; TENTS OR CANOPIES, IN GENERAL
    • E04H1/00—Buildings or groups of buildings for dwelling or office purposes; General layout, e.g. modular co-ordination or staggered storeys
    • E04H1/12—Small buildings or other erections for limited occupation, erected in the open air or arranged in buildings, e.g. kiosks, waiting shelters for bus stops or for filling stations, roofs for railway platforms, watchmen's huts or dressing cubicles
    • E04H1/1272—Exhibition stands
    • F—MECHANICAL ENGINEERING; LIGHTING; HEATING; WEAPONS; BLASTING
    • F16—ENGINEERING ELEMENTS AND UNITS; GENERAL MEASURES FOR PRODUCING AND MAINTAINING EFFECTIVE FUNCTIONING OF MACHINES OR INSTALLATIONS; THERMAL INSULATION IN GENERAL
    • F16B—DEVICES FOR FASTENING OR SECURING CONSTRUCTIONAL ELEMENTS OR MACHINE PARTS TOGETHER, e.g. NAILS, BOLTS, CIRCLIPS, CLAMPS, CLIPS OR WEDGES; JOINTS OR JOINTING
    • F16B2/00—Friction-grip releasable fastenings
    • F16B2/20—Clips, i.e. with gripping action effected solely by the inherent resistance to deformation of the material of the fastening

Landscapes

  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Architecture (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • General Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Structural Engineering (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Civil Engineering (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Mechanical Engineering (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrane Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Description

idet X = H, Cl eller Br, T = O eller S og Y er en arabinose-, xylose- eller riboserest, en acetyleret sådan med enten pyran- eller furankonfiguration og bundet som c- eller p-anomer, fremstilles ved reaktion mellen R-H og ose-forbindelsen i acetyleret form i støkiometrisk forhold i acetonitril under ^ og omrøring ved stuetemperatur i 12 - 24 timer og i nærvær af 1,1,1,3,3,3-hexanmethy1-disilanzan, trimethylchlorsilan og tintetrachlorid.
Forbindelserne er aktive over for vira og bakterier, og visse af dem indvirker på hjerte-kar-systemet, hvor for de anvendes i lægemidler især til bekæmpelse af virussygdomme .
DK181285A 1984-04-24 1985-04-23 Heterocycliske bornan-derivater, fremgangsmaade til fremstilling deraf og laegemiddel indeholdende saadanne forbindelser DK160832C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8410484 1984-04-24
GB848410484A GB8410484D0 (en) 1984-04-24 1984-04-24 Antiviral and antibacterial compounds

Publications (4)

Publication Number Publication Date
DK181285D0 DK181285D0 (da) 1985-04-23
DK181285A true DK181285A (da) 1985-10-25
DK160832B DK160832B (da) 1991-04-22
DK160832C DK160832C (da) 1991-10-07

Family

ID=10560013

Family Applications (2)

Application Number Title Priority Date Filing Date
DK181285A DK160832C (da) 1984-04-24 1985-04-23 Heterocycliske bornan-derivater, fremgangsmaade til fremstilling deraf og laegemiddel indeholdende saadanne forbindelser
DK181385A DK160833C (da) 1984-04-24 1985-04-23 Heterocycliske pyrano-derivater, fremgangsmaade til fremstilling deraf og laegemidler indeholdende saadanne forbindelser

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK181385A DK160833C (da) 1984-04-24 1985-04-23 Heterocycliske pyrano-derivater, fremgangsmaade til fremstilling deraf og laegemidler indeholdende saadanne forbindelser

Country Status (26)

Country Link
US (2) US4720487A (da)
JP (2) JPS60233095A (da)
AR (2) AR241917A1 (da)
AT (2) AT388558B (da)
BE (2) BE902232A (da)
CA (2) CA1265129A (da)
CH (2) CH664572A5 (da)
DE (2) DE3514637A1 (da)
DK (2) DK160832C (da)
DZ (1) DZ772A1 (da)
ES (2) ES8606380A1 (da)
FI (2) FI78301C (da)
FR (3) FR2563107B1 (da)
GB (3) GB8410484D0 (da)
HK (2) HK18788A (da)
IE (2) IE58322B1 (da)
IT (2) IT1215265B (da)
LU (2) LU85865A1 (da)
MA (2) MA20414A1 (da)
MY (1) MY102313A (da)
NL (2) NL193067C (da)
NO (2) NO161122C (da)
OA (2) OA08000A (da)
PT (2) PT80324B (da)
SE (2) SE462972B (da)
ZA (2) ZA852367B (da)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7622492B2 (en) 2005-08-31 2009-11-24 Hoffmann-La Roche Inc. Pyrazolones as inhibitors of 11β-hydroxysteroid dehydrogenase

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3868361A (en) * 1973-03-12 1975-02-25 Richard L Tolman s-Triazolo{8 2,3-A{9 {0 pryimidine nucleosides
DE3019322A1 (de) * 1980-05-21 1981-12-03 Merck Patent Gmbh, 6100 Darmstadt Psychopharmakon sowie verwendung von adenosinderivaten

Also Published As

Publication number Publication date
DE3514637A1 (de) 1985-10-24
HK18788A (en) 1988-03-18
NO161121B (no) 1989-03-28
GB2158436A (en) 1985-11-13
AR241917A1 (es) 1993-01-29
FR2563107A1 (fr) 1985-10-25
FI851577A0 (fi) 1985-04-22
NO161122C (no) 1989-07-05
NO161121C (no) 1989-07-05
MA20414A1 (fr) 1985-12-31
SE8501885D0 (sv) 1985-04-17
BE902232A (fr) 1985-08-16
DE3514641A1 (de) 1985-10-24
FI78302B (fi) 1989-03-31
OA07999A (fr) 1987-01-31
IE851030L (en) 1985-10-24
GB2158436B (en) 1987-08-05
ES8606379A1 (es) 1986-04-01
NL193109B (nl) 1998-07-01
US4704454A (en) 1987-11-03
DK181385A (da) 1985-10-25
FI78301C (fi) 1989-07-10
DK160832C (da) 1991-10-07
DE3514641C2 (da) 1989-02-23
ZA852367B (en) 1985-11-27
ATA122685A (de) 1988-12-15
JPH0129197B2 (da) 1989-06-08
GB8510329D0 (en) 1985-05-30
IT8520440A0 (it) 1985-04-22
FI78301B (fi) 1989-03-31
MY102313A (en) 1992-05-28
HK10289A (en) 1989-02-10
FR2563106A1 (fr) 1985-10-25
DZ772A1 (fr) 2004-09-13
IE58322B1 (en) 1993-09-08
GB2157690B (en) 1988-01-27
FR2563224B1 (fr) 1986-12-19
IE851029L (en) 1985-10-24
SE8501885L (sv) 1985-10-25
GB8510328D0 (en) 1985-05-30
JPH0129198B2 (da) 1989-06-08
GB2157690A (en) 1985-10-30
DK160832B (da) 1991-04-22
AT388557B (de) 1989-07-25
FI851577L (fi) 1985-10-25
SE8501884L (sv) 1985-10-25
ZA852366B (en) 1985-11-27
SE8501884D0 (sv) 1985-04-17
NL193067C (nl) 1998-09-08
FR2563107B1 (fr) 1986-12-19
NO851619L (no) 1985-10-25
DK181285D0 (da) 1985-04-23
NL193067B (nl) 1998-05-06
DK160833C (da) 1991-10-07
LU85865A1 (fr) 1985-12-16
FR2563106B1 (fr) 1986-12-19
DE3514637C2 (da) 1989-04-13
MA20415A1 (fr) 1985-12-31
AR241916A1 (es) 1993-01-29
DK160833B (da) 1991-04-22
IE58323B1 (en) 1993-09-08
PT80325B (pt) 1987-11-11
ES542486A0 (es) 1986-04-01
FI851576A0 (fi) 1985-04-22
NO161122B (no) 1989-03-28
IT1201415B (it) 1989-02-02
FR2563224A1 (fr) 1985-10-25
SE462973B (sv) 1990-09-24
CA1241649A (en) 1988-09-06
DK181385D0 (da) 1985-04-23
CA1265129A (en) 1990-01-30
JPS60233096A (ja) 1985-11-19
US4720487A (en) 1988-01-19
IT8520439A0 (it) 1985-04-22
ES542485A0 (es) 1986-04-01
JPS60233095A (ja) 1985-11-19
OA08000A (fr) 1987-01-31
ATA122585A (de) 1988-12-15
LU85864A1 (fr) 1985-12-16
CH664572A5 (fr) 1988-03-15
BE902231A (fr) 1985-08-16
NO851620L (no) 1985-10-25
FI851576L (fi) 1985-10-25
PT80324B (pt) 1987-11-11
FI78302C (fi) 1989-07-10
AT388558B (de) 1989-07-25
PT80325A (en) 1985-05-01
ES8606380A1 (es) 1986-04-01
GB8410484D0 (en) 1984-05-31
IT1215265B (it) 1990-01-31
SE462972B (sv) 1990-09-24
CH665837A5 (fr) 1988-06-15
PT80324A (en) 1985-05-01
NL8501171A (nl) 1985-11-18
NL8501170A (nl) 1985-11-18

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