DK1858878T3 - Konvertering af 2-pyrazoliner til pyrazoler ved hjælp af brom - Google Patents
Konvertering af 2-pyrazoliner til pyrazoler ved hjælp af bromInfo
- Publication number
- DK1858878T3 DK1858878T3 DK06738651.6T DK06738651T DK1858878T3 DK 1858878 T3 DK1858878 T3 DK 1858878T3 DK 06738651 T DK06738651 T DK 06738651T DK 1858878 T3 DK1858878 T3 DK 1858878T3
- Authority
- DK
- Denmark
- Prior art keywords
- formula
- bromine
- pyrazolines
- pyrazoles
- conversion
- Prior art date
Links
- MCGBIXXDQFWVDW-UHFFFAOYSA-N 4,5-dihydro-1h-pyrazole Chemical class C1CC=NN1 MCGBIXXDQFWVDW-UHFFFAOYSA-N 0.000 title abstract 2
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical compound [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 title abstract 2
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Substances BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 title abstract 2
- 229910052794 bromium Inorganic materials 0.000 title abstract 2
- 238000006243 chemical reaction Methods 0.000 title 1
- 150000003217 pyrazoles Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 4
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/16—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Chemical Treatment Of Metals (AREA)
- Enzymes And Modification Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US66341005P | 2005-03-18 | 2005-03-18 | |
| PCT/US2006/009617 WO2006102025A1 (en) | 2005-03-18 | 2006-03-14 | Conversion of 2-pyrazolines to pyrazoles using bromine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1858878T3 true DK1858878T3 (da) | 2012-08-06 |
Family
ID=36592996
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK06738651.6T DK1858878T3 (da) | 2005-03-18 | 2006-03-14 | Konvertering af 2-pyrazoliner til pyrazoler ved hjælp af brom |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US7951953B2 (da) |
| EP (1) | EP1858878B1 (da) |
| JP (1) | JP5086987B2 (da) |
| KR (1) | KR101337159B1 (da) |
| CN (1) | CN101142207B (da) |
| AT (1) | ATE555103T1 (da) |
| AU (1) | AU2006227484B2 (da) |
| BR (1) | BRPI0609844B1 (da) |
| CA (1) | CA2601870C (da) |
| DK (1) | DK1858878T3 (da) |
| ES (1) | ES2385496T3 (da) |
| IL (1) | IL185329A (da) |
| MX (1) | MX2007011162A (da) |
| PL (1) | PL1858878T3 (da) |
| RS (2) | RS52344B (da) |
| RU (1) | RU2410381C2 (da) |
| TW (1) | TWI371449B (da) |
| UA (1) | UA93869C2 (da) |
| WO (1) | WO2006102025A1 (da) |
| ZA (1) | ZA200707470B (da) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101243067A (zh) * | 2005-08-24 | 2008-08-13 | 杜邦公司 | 用于防治无脊椎害虫的新的邻氨基苯甲酰胺 |
| CN101550130B (zh) * | 2008-04-01 | 2012-11-07 | 中国中化股份有限公司 | 一种制备3-卤代-1-(3-氯-2-吡啶基)-1h-吡唑-5-甲酰卤的方法 |
| CN101863874B (zh) * | 2009-04-14 | 2013-11-06 | 中国中化股份有限公司 | 一种吡唑亚胺类化合物及其应用 |
| WO2011157654A1 (de) | 2010-06-15 | 2011-12-22 | Bayer Cropscience Ag | Anthranilsäurediamid-derivate |
| TWI849253B (zh) * | 2019-11-11 | 2024-07-21 | 美商富曼西公司 | 用於製備3-溴-1- (3-氯吡啶-2-基) -1h-吡唑-5-羧酸乙酯的方法 |
| TWI884201B (zh) * | 2020-01-08 | 2025-05-21 | 美商富曼西公司 | 用於製備3-溴-1-(3-氯吡啶-2-基)-1h-吡唑-5-羧酸乙酯的方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5281571A (en) * | 1990-10-18 | 1994-01-25 | Monsanto Company | Herbicidal benzoxazinone- and benzothiazinone-substituted pyrazoles |
| TWI356822B (en) * | 2001-08-13 | 2012-01-21 | Du Pont | Novel substituted dihydro 3-halo-1h-pyrazole-5-car |
| TWI325302B (en) | 2001-08-13 | 2010-06-01 | Du Pont | Benzoxazinone compounds |
| TWI343376B (en) | 2002-07-31 | 2011-06-11 | Du Pont | Method for preparing 3-halo-4, 5-dihydro-1h-pyrazoles |
-
2006
- 2006-03-14 EP EP06738651A patent/EP1858878B1/en not_active Expired - Lifetime
- 2006-03-14 AU AU2006227484A patent/AU2006227484B2/en not_active Expired
- 2006-03-14 MX MX2007011162A patent/MX2007011162A/es active IP Right Grant
- 2006-03-14 ZA ZA200707470A patent/ZA200707470B/xx unknown
- 2006-03-14 KR KR1020077023792A patent/KR101337159B1/ko not_active Expired - Lifetime
- 2006-03-14 CN CN2006800087738A patent/CN101142207B/zh not_active Expired - Lifetime
- 2006-03-14 DK DK06738651.6T patent/DK1858878T3/da active
- 2006-03-14 AT AT06738651T patent/ATE555103T1/de active
- 2006-03-14 ES ES06738651T patent/ES2385496T3/es not_active Expired - Lifetime
- 2006-03-14 RU RU2007138552/04A patent/RU2410381C2/ru active
- 2006-03-14 PL PL06738651T patent/PL1858878T3/pl unknown
- 2006-03-14 WO PCT/US2006/009617 patent/WO2006102025A1/en not_active Ceased
- 2006-03-14 US US11/885,325 patent/US7951953B2/en active Active
- 2006-03-14 CA CA2601870A patent/CA2601870C/en not_active Expired - Fee Related
- 2006-03-14 RS RS20120261A patent/RS52344B/sr unknown
- 2006-03-14 BR BRPI0609844-4A patent/BRPI0609844B1/pt active IP Right Grant
- 2006-03-14 JP JP2008502077A patent/JP5086987B2/ja not_active Expired - Lifetime
- 2006-03-14 UA UAA200709764A patent/UA93869C2/ru unknown
- 2006-03-14 RS RSP-2007/0369A patent/RS20070369A/sr unknown
- 2006-03-14 TW TW095108602A patent/TWI371449B/zh not_active IP Right Cessation
-
2007
- 2007-08-16 IL IL185329A patent/IL185329A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| KR101337159B1 (ko) | 2013-12-05 |
| CN101142207B (zh) | 2011-10-05 |
| AU2006227484A1 (en) | 2006-09-28 |
| JP5086987B2 (ja) | 2012-11-28 |
| BRPI0609844B1 (pt) | 2015-06-30 |
| TW200700407A (en) | 2007-01-01 |
| US7951953B2 (en) | 2011-05-31 |
| ATE555103T1 (de) | 2012-05-15 |
| EP1858878B1 (en) | 2012-04-25 |
| UA93869C2 (en) | 2011-03-25 |
| BRPI0609844A2 (pt) | 2010-05-04 |
| US20080177078A1 (en) | 2008-07-24 |
| MX2007011162A (es) | 2007-10-17 |
| ZA200707470B (en) | 2008-12-31 |
| RU2410381C2 (ru) | 2011-01-27 |
| CN101142207A (zh) | 2008-03-12 |
| RS20070369A (sr) | 2009-01-22 |
| ES2385496T3 (es) | 2012-07-25 |
| JP2008533169A (ja) | 2008-08-21 |
| RS52344B (sr) | 2012-12-31 |
| IL185329A (en) | 2013-04-30 |
| TWI371449B (en) | 2012-09-01 |
| CA2601870A1 (en) | 2006-09-28 |
| AU2006227484B2 (en) | 2011-08-11 |
| WO2006102025A1 (en) | 2006-09-28 |
| RU2007138552A (ru) | 2009-04-27 |
| IL185329A0 (en) | 2008-02-09 |
| PL1858878T3 (pl) | 2012-09-28 |
| EP1858878A1 (en) | 2007-11-28 |
| KR20070112292A (ko) | 2007-11-22 |
| CA2601870C (en) | 2013-06-11 |
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