DK234889A - Heteroaroylhydrazidderivater af monocycliske beta-lactamantibiotika og farmaceutisk acceptable salte deraf samt mellemprodukter ved deres fremstilling - Google Patents

Heteroaroylhydrazidderivater af monocycliske beta-lactamantibiotika og farmaceutisk acceptable salte deraf samt mellemprodukter ved deres fremstilling Download PDF

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Publication number
DK234889A
DK234889A DK234889A DK234889A DK234889A DK 234889 A DK234889 A DK 234889A DK 234889 A DK234889 A DK 234889A DK 234889 A DK234889 A DK 234889A DK 234889 A DK234889 A DK 234889A
Authority
DK
Denmark
Prior art keywords
lactamantibiotics
heteroaroyl
intermediates
preparation
acceptable salts
Prior art date
Application number
DK234889A
Other languages
English (en)
Other versions
DK234889D0 (da
Inventor
Joseph Edward Sundeen
Peter Has Ermann
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of DK234889D0 publication Critical patent/DK234889D0/da
Publication of DK234889A publication Critical patent/DK234889A/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/36Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
    • C07D241/38Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with only hydrogen or carbon atoms directly attached to the ring nitrogen atoms
    • C07D241/40Benzopyrazines
    • C07D241/44Benzopyrazines with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK234889A 1988-05-16 1989-05-12 Heteroaroylhydrazidderivater af monocycliske beta-lactamantibiotika og farmaceutisk acceptable salte deraf samt mellemprodukter ved deres fremstilling DK234889A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/194,355 US4904775A (en) 1988-05-16 1988-05-16 Heteroaroylhydrazide derivatives of monocyclic beta-lactam antibiotics

Publications (2)

Publication Number Publication Date
DK234889D0 DK234889D0 (da) 1989-05-12
DK234889A true DK234889A (da) 1989-11-17

Family

ID=22717261

Family Applications (1)

Application Number Title Priority Date Filing Date
DK234889A DK234889A (da) 1988-05-16 1989-05-12 Heteroaroylhydrazidderivater af monocycliske beta-lactamantibiotika og farmaceutisk acceptable salte deraf samt mellemprodukter ved deres fremstilling

Country Status (7)

Country Link
US (1) US4904775A (da)
EP (1) EP0342423A3 (da)
JP (1) JPH0217189A (da)
AU (2) AU618598B2 (da)
DK (1) DK234889A (da)
NZ (1) NZ228880A (da)
ZA (1) ZA893483B (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5232918A (en) * 1987-07-23 1993-08-03 Imperial Chemical Industries Plc Cephalosporin derivatives
US5037983A (en) * 1988-05-16 1991-08-06 E. R. Squibb & Sons, Inc. 6,7-dihydroxyquinoxalines as intermediates to beta-lactam antibiotics
US5112968A (en) * 1989-07-28 1992-05-12 E. R. Squibb & Sons, Inc. Monobactam hydrazide derivatives
CA2024282A1 (en) * 1989-09-21 1991-03-22 Peter H. Ermann Heterocyclic hydrazide derivatives of monocyclic beta-lactam antibiotics
US5194604A (en) * 1990-06-29 1993-03-16 E. R. Squibb & Sons, Inc. Process and intermediates for beta-lactams having aminothiazole(iminooxyacetic acid)acetic acid sidechains
ZA918014B (en) * 1990-11-05 1992-07-29 Squibb & Sons Inc Heteroaroyl derivatives of monocyclic beta-lactam antibiotics
US5250691A (en) * 1991-09-09 1993-10-05 E. R. Squibb & Sons, Inc. Heteroaryl derivatives of monocyclic beta-lactam antibiotics
JP3749628B2 (ja) 1997-12-26 2006-03-01 キッコーマン株式会社 ルシフェラーゼおよびそれを用いる細胞内atpの測定法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4217453A (en) * 1978-07-24 1980-08-12 Merck & Co., Inc. 6-Amido-3-substituted-amino-1-azabicyclo[3.2.0]hept-2-en-7-one-2-carboxylic acid
PH15791A (en) * 1978-10-20 1983-03-25 Lilly Co Eli Pharmaceutical composition containing 3,4-dihydro-3-oxoquinoxalines
US4224336A (en) * 1979-04-17 1980-09-23 Merck & Co., Inc. 3-(2-Aminoethylthio)-6-amido-7-oxo-1-azabicyclo[3.2.0]-hept-2-ene-2-carboxylic acid
DE3372768D1 (de) * 1982-06-03 1987-09-03 Hoffmann La Roche 1-sulfo-2-oxoazetidine derivatives
US4610824A (en) * 1984-10-09 1986-09-09 E. R. Squibb & Sons, Inc. Hydrazide derivatives of monocyclic beta-lactam antibiotics
US4638062A (en) * 1985-06-17 1987-01-20 E. R. Squibb & Sons, Inc. 3-acylamino-2-oxo-1-azetidinesulfonic acids
FI872879A7 (fi) * 1986-07-21 1988-01-22 Sankei Yakuhin Kk --laktamfoerening, foerfarande foer dess framstaellning, denna innehaollande laekemedelskomposition foer behandling av sjukdom med bakterieinfektion samt mellanprodukter foer dess syntes.
GB8816519D0 (en) * 1987-07-23 1988-08-17 Ici Plc Antibiotic compounds
US4777252A (en) * 1987-08-13 1988-10-11 E. R. Squibb & Sons, Inc. 2-oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines

Also Published As

Publication number Publication date
AU640531B2 (en) 1993-08-26
JPH0217189A (ja) 1990-01-22
US4904775A (en) 1990-02-27
AU8576891A (en) 1991-12-05
ZA893483B (en) 1990-01-31
AU3484789A (en) 1989-11-16
AU618598B2 (en) 1992-01-02
DK234889D0 (da) 1989-05-12
EP0342423A3 (en) 1991-04-17
EP0342423A2 (en) 1989-11-23
NZ228880A (en) 1991-04-26

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